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MAP kinase p38 alpha Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazoleIC5048.0 [1]
4-(4-Fluorophenyl)-2-(4-methylsulfinylphenyl)-5-(4-pyridyl)-1H-imidazoleKi18.0 [1], 57.0 [2]
DoramapimodIC5017.0 [1]
DoramapimodKi0.1 [1], 6.4 [2], 22.0 [3], 46.0 [4]
NeflamapimodIC5051.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMAP kinase p38 alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/map-kinase-p38-alpha-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseMAP kinase p38 alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/map-kinase-p38-alpha-inhibitors-ic50-ki.
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