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MAP kinase p38 gamma Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
▲
▼
DoramapimodIC5030.0 [1], 102.0 [2], 296.0 [3]
Unii-I92MU0V408IC5040.0 [1], 402.0 [2]
N-[4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]pyridin-2-yl]acetamideIC50195.0 [1]
N-[4-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxypyridin-2-yl]-2-methoxyacetamideIC50344.0 [1]
TofacitinibIC5010000.0 [1]
Cyclohexanol, 4-(4-(4-fluorophenyl)-5-(2-methoxy-4-pyrimidinyl)-1H-imidazol-1-yl)-, trans-IC50100000.0 [1]
Benzamide, N-[4-[2-ethyl-4-(3-methylphenyl)-5-thiazolyl]-2-pyridinyl]-IC5010000.0 [1]
JNK Inhibitor VIIIKi7500.0 [1]
CID 44814409IC5010000.0 [1]
N-[2-Methyl-5-(methylcarbamoyl)phenyl]-2-{[(1R)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamideIC5030000.0 [1]
1-(5-Tert-Butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-[4-(2-pyridin-4-yl-ethoxy)-naphthalen-1-yl]-ureaIC50213.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)acetamideKi7500.0 [1]
4-Amino-5-chloro-6-ethoxy-pyridine-2-carboxylic acid 4-methanesulfonyl-benzylamideKi7500.0 [1]
7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrileKi7500.0 [1]
1-({4-[(3,4-Dichlorophenyl)methoxy]phenyl}methyl)azetidine-3-carboxylic acidIC5010000.0 [1]
6-Acetyl-8-cyclopentyl-5-methyl-2-(4-piperazin-1-yl-phenylamino)-8H-pyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
1-(5-Tert-Butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-[4-(2-imidazol-1-yl-ethoxy)-naphthalen-1-yl]-ureaIC502050.0 [1]
1-(5-Tert-Butyl-2-p-tolyl-2H-pyrazol-3-yl)-3-[4-(2-pyridin-3-yl-ethoxy)-naphthalen-1-yl]-ureaIC50616.0 [1]
3-[[5-Cyano-6-(cyclopentylamino)pyrimidin-4-yl]amino]-4-methyl-N-(1,2-oxazol-3-yl)benzamideIC5030000.0 [1]
7-Chloro-8-(3-hydroxypropoxy)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
7-Chloro-8-(3-hydroxypropyl)-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5(10),6,8,18(22),19-hexaene-19-carbonitrileKi10000.0 [1]
N-(7-Chloro-19-cyano-3-oxo-11,17-dioxa-2,4,20,22-tetrazatricyclo[16.3.1.05,10]docosa-1(21),5,7,9,18(22),19-hexaen-8-yl)methanesulfonamideKi10000.0 [1]
N-(4-Amino-5-cyano-6-ethoxypyridin-2-yl)-2-(2,5-dimethoxy-4-methylsulfonylphenyl)acetamideKi7500.0 [1]
N-(4-Amino-5-chloro-6-ethoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi7500.0 [1]
N-(4-Amino-5-cyano-6-isopropoxypyridin-2-yl)-2-(4-methanesulfonyl-2,5-dimethoxyphenyl)acetamideKi7500.0 [1]
N-(4-Amino-5-cyano-6-phenylpyridin-2-yl)acetamideKi7500.0 [1]
(13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dioneIC501000.0 [1]
N-Cyclopropyl-3-[1-(2,6-difluorophenyl)-7-methyl-6-oxopyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamideKi3500.0 [1]
5-(2-Aminoethyl)-7-(7-(benzo[b]thiophen-2-yl)-1H-indazol-5-yl)-5H-pyrrolo[3,2-d]pyrimidin-2-amineIC504000.0 [1]
N-[3-[5-[2-(3-Morpholin-4-ylanilino)pyrimidin-4-yl]imidazo[2,1-b][1,3]thiazol-6-yl]phenyl]-2-phenylacetamideIC501000.0 [1]
1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaIC5030000.0 [1]
9-Cyclopentyl-N2-[4-(4-methylpiperazin-1-yl)phenyl]-N8-phenyl-purine-2,8-diamineIC5010000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
CID 9811100IC5010000.0 [1]
3-[(6-Benzoyl-5-Methylpyrrolo[2,1-F][1,2,4]triazin-4-Yl)amino]-N-Cyclopropyl-4-MethylbenzamideIC5025000.0 [1]
5-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4-difluorophenyl)-1,3-oxazoleIC5010000.0 [1]
5-(3-Propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazoleIC5010000.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
N-[4-[2-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]pyridin-3-yl]acetamideIC50634.0 [1]
4-[2-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]-N-methylpyridine-2-carboxamideIC5017000.0 [1]
N-[1-[2-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]imidazol-2-yl]acetamideIC5017000.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-[[2-(methanesulfonamido)pyridin-4-yl]methoxy]naphthalen-1-yl]ureaIC50303.0 [1]
N-[4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]pyridin-2-yl]benzamideIC508359.0 [1]
4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]-N-(2-methoxyethyl)pyridine-2-carboxamideIC5016000.0 [1]
4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]-N-(2-morpholin-4-ylethyl)pyridine-2-carboxamideIC5015000.0 [1]
Methyl N-[4-[2-[4-[[5-tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]pyridin-2-yl]carbamateIC5017000.0 [1]
N-[4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]pyridin-2-yl]-2-phenylacetamideIC50378.0 [1]
4-[2-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]-N-(2-methoxyethyl)pyridine-2-carboxamideIC5016000.0 [1]
N-[4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]pyridin-2-yl]-2-methoxy-N-methylacetamideIC502438.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-(2-pyridin-2-ylethoxy)naphthalen-1-yl]ureaIC502950.0 [1]
N,4-Dimethyl-3-[[6-(methylamino)-1-phenylpyrazolo[3,4-d]pyrimidin-4-yl]amino]benzamideIC5030000.0 [1]
4-(2-Chloro-4-fluorophenyl)-5-(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-1,3-oxazoleIC5010000.0 [1]
N-Ethyl-6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-[1,2,4]triazolo[4,3-a]pyridin-3-amineIC5010000.0 [1]
6-[5-(2,5-Difluorophenyl)-1H-pyrazol-4-yl]-3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridineIC5010000.0 [1]
4-(2-Chloro-4-fluorophenyl)-8-(2,6-dichlorophenyl)-7-oxido-1,7-naphthyridin-7-iumIC5010000.0 [1]
1-(5-Tert-butyl-2-phenylpyrazol-3-yl)-3-[4-[(3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC5043.0 [1]
1-(5-Tert-butyl-2-phenylpyrazol-3-yl)-3-[4-[(2-methyl-3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC50100.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-[(3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC5072.0 [1]
4-Chloro-N-cyclopropyl-3-[[1-(4-fluorophenyl)-7-methyl-6-oxopyrazolo[3,4-b]pyridin-4-yl]amino]benzamideIC5010000.0 [1]
4-(4-(2-(Cyclopentylamino)pyrimidin-4-yl)-1H-pyrazol-3-yl)cyclohexanolIC506200.0 [1]
N-[4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]pyridin-2-yl]-2-(dimethylamino)acetamideIC50461.0 [1]
N-[4-[2-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]pyridin-2-yl]-2-methoxyacetamideIC50647.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-[2-[2-(methylcarbamoylamino)pyridin-4-yl]ethoxy]naphthalen-1-yl]ureaIC50169.0 [1]
N-[4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]pyridin-2-yl]-2-methylsulfanylacetamideIC50148.0 [1]
N-[4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]pyridin-2-yl]-2-morpholin-4-ylacetamideIC50352.0 [1]
1-(5-Tert-butyl-2-phenylpyrazol-3-yl)-3-[4-[(2-oxo-1,3-dihydroimidazo[4,5-b]pyridin-7-yl)oxy]naphthalen-1-yl]ureaIC5067.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-[(2-oxo-1,3-dihydroimidazo[4,5-b]pyridin-7-yl)oxy]naphthalen-1-yl]ureaIC5074.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-[(1-methyl-2-oxo-3H-imidazo[4,5-b]pyridin-7-yl)oxy]naphthalen-1-yl]ureaIC5024.0 [1]
1-(5-Tert-butyl-2-phenylpyrazol-3-yl)-3-[3-[(2-oxo-1,3-dihydrobenzimidazol-4-yl)oxy]phenyl]ureaIC501810.0 [1]
N-(5-Tert-butyl-2-phenylpyrazol-3-yl)-3-[(2-oxo-1,3-dihydrobenzimidazol-4-yl)oxy]benzamideIC5010000.0 [1]
3-(Trifluoromethoxy)-N-[2,3,4-trifluoro-5-[(2-oxo-1,3-dihydrobenzimidazol-4-yl)oxy]phenyl]benzamideIC5010000.0 [1]
N-[4-[2-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]pyridin-3-yl]-2-methoxyacetamideIC50354.0 [1]
N-[4-[1-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]pyridin-2-yl]-2-methoxyacetamideIC50902.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-[(2-methyl-3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC5099.0 [1]
N-[4-[[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxymethyl]pyridin-2-yl]-2-methylsulfonylacetamideIC5055.0 [1]
N-[4-[2-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxyethyl]pyridin-2-yl]acetamideIC50972.0 [1]
Infigratinib phosphateIC5010000.0 [1]
1-(4-(2-(2-Aminopyridin-4-yl)ethoxy)naphthalen-1-yl)-3-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)ureaIC501504.0 [1]
1-(4-(2-(3-Aminopyridin-4-yl)ethoxy)naphthalen-1-yl)-3-(3-tert-butyl-1-p-tolyl-1H-pyrazol-5-yl)ureaIC50591.0 [1]
N-[4-[2-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxypropan-2-yl]pyridin-2-yl]-2-methoxyacetamideIC501941.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC5010000.0 [1]
3-Isopropyl-6-(4-phenyl-oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridineIC5010000.0 [1]
5-(3-Tert-butyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4-(2,4,5-trifluorophenyl)-1,3-oxazoleIC5010000.0 [1]
1-[5-Tert-butyl-2-[4-(hydroxymethyl)phenyl]pyrazol-3-yl]-3-[2,3-dichloro-4-[(3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]phenyl]ureaIC5035.0 [1]
1-[5-Tert-butyl-2-[6-(hydroxymethyl)pyridin-3-yl]pyrazol-3-yl]-3-[4-[(3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC5044.0 [1]
1-(5-Tert-butyl-2-phenylpyrazol-3-yl)-3-[8-[(2-oxo-1,3-dihydroimidazo[4,5-b]pyridin-7-yl)oxy]quinolin-5-yl]ureaIC50214.0 [1]
N-[4-[4-[[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoylamino]naphthalen-1-yl]oxypyridin-2-yl]acetamideIC50146.0 [1]
1-[5-Tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-3-[4-[(2-oxo-1,3-dihydroimidazo[4,5-b]pyridin-7-yl)oxy]naphthalen-1-yl]ureaIC50119.0 [1]
1-[5-Tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-3-[4-[(1-methyl-2-oxo-3H-imidazo[4,5-b]pyridin-7-yl)oxy]naphthalen-1-yl]ureaIC5045.0 [1]
1-[5-Tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-3-[8-[(2-oxo-1,3-dihydroimidazo[4,5-b]pyridin-7-yl)oxy]quinolin-5-yl]ureaIC50180.0 [1]
1-[5-Tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-3-[4-[(1-ethyl-2-oxo-3H-imidazo[4,5-b]pyridin-7-yl)oxy]naphthalen-1-yl]ureaIC50348.0 [1]
1-[5-Tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-3-[4-[(2-oxo-1-propan-2-yl-3H-imidazo[4,5-b]pyridin-7-yl)oxy]naphthalen-1-yl]ureaIC50495.0 [1]
1-[5-Tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-3-[2,3-dichloro-4-[(1-methyl-2-oxo-3H-imidazo[4,5-b]pyridin-7-yl)oxy]phenyl]ureaIC5023.0 [1]
1-[5-Tert-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[4-[(8-oxo-7,9-dihydropurin-6-yl)oxy]naphthalen-1-yl]ureaIC50539.0 [1]
1-[5-Tert-butyl-2-(4-hydroxyphenyl)pyrazol-3-yl]-3-[4-[(3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC5045.0 [1]
1-[5-Tert-butyl-2-[4-(hydroxymethyl)phenyl]pyrazol-3-yl]-3-[4-[(3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC50318.0 [1]
1-[5-Tert-butyl-2-[4-(hydroxymethyl)-3-methoxyphenyl]pyrazol-3-yl]-3-[4-[(3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC5024.0 [1]
1-[5-Tert-butyl-2-(5-methylthiophen-2-yl)pyrazol-3-yl]-3-[4-[(3-oxo-4H-pyrido[2,3-b]pyrazin-8-yl)oxy]naphthalen-1-yl]ureaIC5041.0 [1]
1-[5-Tert-butyl-2-(4-methoxyphenyl)pyrazol-3-yl]-3-[4-[(7-oxo-8H-pteridin-4-yl)oxy]naphthalen-1-yl]ureaIC502620.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ MAP kinase p38 gamma Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/map-kinase-p38-gamma-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ MAP kinase p38 gamma Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/map-kinase-p38-gamma-inhibitors-ic50-ki.
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