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Matrix metalloproteinase 13 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(2R)-N-Hydroxy-2-[(4-methoxyphenyl)sulfonyl-(pyridin-3-ylmethyl)amino]-3-methylbutanamide;hydrochlorideIC508.0 [1]
(2R)-N-Hydroxy-2-[(4-methoxyphenyl)sulfonyl-(pyridin-3-ylmethyl)amino]-3-methylbutanamide;hydrochlorideKi1.27 [1]
4-[4-(4-Chloro-phenoxy)-benzenesulfonylmethyl]-tetrahydro-pyran-4-carboxylic acid hydroxyamideIC500.3 [1]
4-[4-(4-Chloro-phenoxy)-benzenesulfonylmethyl]-tetrahydro-pyran-4-carboxylic acid hydroxyamideKi0.28 [1], 0.52 [2]
MarimastatIC502.0 [1]
PrinomastatIC500.2 [1], 0.4 [2], 0.5 [3], 1.5 [4]
PrinomastatKi0.04 [1]
CipemastatIC503.4 [1], 3.5 [2], 4.7 [3]
CipemastatKi0.53 [1], 1.0 [2], 3.0 [3]
Pyrimidine-4,6-dicarboxylic acid bis-(4-fluoro-3-methyl-benzylamide)IC508.0 [1]
Benzyl 6-Benzyl-5,7-Dioxo-6,7-Dihydro-5h-[1,3]thiazolo[3,2-C]pyrimidine-2-CarboxylateIC5023.0 [1], 30.0 [2], 51.0 [3]
Benzyl 6-Benzyl-5,7-Dioxo-6,7-Dihydro-5h-[1,3]thiazolo[3,2-C]pyrimidine-2-CarboxylateKi64.0 [1]
n-Hydroxy-2-[(4-methoxy-benzenesulfonyl)-pyridin-3-ylmethyl-amino]-3-methyl-benzamideIC507.94 [1], 8.0 [2]
2-[(4-Methylbenzyl)sulfanyl]-3,5,6,7-Tetrahydro-4h-Cyclopenta[d]pyrimidin-4-OneIC502400.0 [1]
2-[(4-Methylbenzyl)sulfanyl]-3,5,6,7-Tetrahydro-4h-Cyclopenta[d]pyrimidin-4-OneKi800.0 [1], 824.0 [2]
CID 6914621IC501417.0 [1]
CID 6914621Ki1417.0 [1]
4-{[1-Methyl-2,4-Dioxo-6-(3-Phenylprop-1-Yn-1-Yl)-1,4-Dihydroquinazolin-3(2h)-Yl]methyl}benzoic AcidIC500.67 [1], 14.0 [2]
4-[(4-But-2-ynoxyphenyl)sulfonylmethyl]-N-hydroxy-1-propan-2-ylsulfonylpiperidine-4-carboxamideIC50157.0 [1], 230.0 [2]
N-({4'-[(1-Benzofuran-2-ylcarbonyl)amino]-1,1'-biphenyl-4-YL}sulfonyl)-L-valineIC501.3 [1], 2.4 [2]
(2R,3R)-1-[4-[(2-Chloro-4-fluorophenyl)methoxy]phenyl]sulfonyl-N,3-dihydroxy-3-methylpiperidine-2-carboxamideIC500.9 [1], 1.0 [2], 10.0 [3]
(2R)-2-[[4-(4-Methoxyphenyl)phenyl]sulfonylamino]-2-[1-[(2-methylpropan-2-yl)oxycarbonyl]piperidin-4-yl]acetic acidIC500.4 [1], 0.5 [2], 11.0 [3]
5-[3-Fluoro-4-[(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)sulfanylmethyl]phenyl]-N-[(2S)-3-methyl-1-(methylamino)-1-oxobutan-2-yl]furan-2-carboxamideIC502.7 [1], 8.1 [2]
5-[3-Fluoro-4-[(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)sulfanylmethyl]phenyl]-N-[(2S)-3-methyl-1-(methylamino)-1-oxobutan-2-yl]furan-2-carboxamideKi1.7 [1]
4-[[[5-(2-Ethoxycarbonyl-1H-indol-5-yl)-1-methylpyrazole-3-carbonyl]amino]methyl]benzoic acidIC501.0 [1], 4.0 [2], 11.0 [3], 31.0 [4]
(3S)-4-{[4-(But-2-ynyloxy)phenyl]sulfonyl}-N-hydroxy-2,2-dimethylthiomorpholine-3-carboxamideIC502.4 [1], 3.0 [2]
2-[(4-Chlorophenyl)methylthio]-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-oneIC503400.0 [1], 10300.0 [2]
2-[(4-Chlorophenyl)methylthio]-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-4-oneKi3800.0 [1]
CID 10370504IC5073.0 [1]
2-[(4-Methoxyphenyl)methylthio]-6-methyl-1H-pyrimidin-4-oneIC501600.0 [1], 4300.0 [2], 20000.0 [3]
2-[(4-Phenylphenyl)sulfonylamino]pentanedioic acidIC50280.0 [1], 2100.0 [2], 13000.0 [3]
3-(4-Hexyloxy-phenyl)-succinamic acidIC501300.0 [1], 4800.0 [2], 27000.0 [3]
2-(Biphenyl-4-ylsulfonamido)-N-hydroxyacetamideIC502.4 [1], 2.8 [2]
2-(Biphenyl-4-ylsulfonamido)-N-hydroxyacetamideKi2.0 [1]
N-Hydroxy-4-(4-phenylsulfanylphenyl)sulfonyl-1-prop-2-ynylpiperidine-4-carboxamideIC500.4 [1], 1.0 [2]
(2S)-2-[[4-(4-Methoxyphenyl)phenyl]sulfonylamino]-3-methylbutanoic acidIC506.0 [1], 24.2 [2]
N-(3-Methoxybenzyl)-4-Oxo-3,4-Dihydroquinazoline-2-CarboxamideIC505.6 [1], 12.0 [2]
N-Hydroxy-2-[[4-(4-methoxyphenyl)phenyl]methyl]-1,1-dioxo-1,2-thiazolidine-3-carboxamideKi55.0 [1]
(2R,3R)-3-(Cyclopentylmethyl)-N-hydroxy-2-[[methyl(methylsulfonyl)amino]methyl]-4-oxo-4-piperidin-1-ylbutanamideIC50398.11 [1], 400.0 [2]
4-((6-(4-Methoxybenzylcarbamoyl)-4-oxopyrido[3,4-d]pyrimidin-3(4H)-yl)methyl)benzoic acidIC506.72 [1], 30.5 [2]
2-[Benzyl(4-methoxyphenylsulfonyl)amino]benzenecarbohydroximic acidIC50549.54 [1], 555.0 [2]
2-[Benzyl(4-methoxyphenylsulfonyl)amino]-3-methoxybenzenecarbohydroximic acidIC50138.0 [1], 138.04 [2]
2-[Methyl(4-methoxyphenylsulfonyl)amino]-3-methyl-5-bromobenzohydroximic acidIC5011.0 [1], 21.0 [2]
(2R)-2-[Benzyl-[4-(2-fluoroethoxy)phenyl]sulfonylamino]-N-hydroxy-3-methylbutanamideIC5011.0 [1]
1-[4-(4-Chlorophenoxy)phenyl]-1,7,9-triazaspiro[4.5]decane-2,6,8,10-tetroneKi0.95 [1], 1.0 [2]
2-[Methyl[4-(2-propynyloxy)phenylsulfonyl]amino]-3-methyl-5-bromobenzohydroximic acidIC5052.0 [1], 113.0 [2]
2-(4'-Methoxy-4-biphenylylsulfonylamino)-5-phenyl-4-pentynoic acidIC5020.89 [1], 21.0 [2]
N-[(1S)-1-Cyclohexyl-2-(methylamino)-2-oxoethyl]-5-[3-fluoro-4-[(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)sulfanylmethyl]phenyl]furan-2-carboxamideIC504.4 [1], 6.3 [2], 7.9 [3]
(2R)-2-[[5-(4-Ethoxyphenyl)thiophen-2-yl]sulfonylamino]-2-(1-propan-2-yloxycarbonylpiperidin-4-yl)acetic acidIC500.5 [1], 37.8 [2]
(2R)-2-[[5-(4-Ethoxyphenyl)thiophen-2-yl]sulfonylamino]-2-(1-propan-2-yloxycarbonylpiperidin-4-yl)acetic acidKi0.19 [1]
N-(2-Aminoethyl)-4-[4-[(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)sulfanylmethyl]phenyl]benzenesulfonamideIC503.4 [1], 8.3 [2]
N-(2-Aminoethyl)-4-[4-[(4-oxo-3,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)sulfanylmethyl]phenyl]benzenesulfonamideKi13.5 [1]
IlomastatIC505.2 [1]
N-Isobutyl-N-[4-methoxyphenylsulfonyl]glycyl hydroxamic acidIC503.0 [1]
N-Isobutyl-N-[4-methoxyphenylsulfonyl]glycyl hydroxamic acidKi3.1 [1]
(S)-2-(4'-Bromo-[1,1'-biphenyl]-4-ylsulfonamido)-3-methylbutanoic acidIC508.0 [1]
N-Hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)acetamideIC5025.0 [1]
N-Hydroxy-2-(N-isopropoxybiphenyl-4-ylsulfonamido)acetamideKi20.0 [1]
cis-2-Aminocyclohexylcarbamoylphosphonic acidIC50100000.0 [1]
(3R)-3-[[(2S)-1-[[(1S)-2-Methoxy-1-phenylethyl]amino]-3,3-dimethyl-1-oxobutan-2-yl]carbamoyl]-6-(3-methyl-4-phenylphenyl)hexanoic acidIC502300.0 [1]
4-[[(4-Oxo-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)thio]methyl]benzoic acid methyl esterIC502800.0 [1]
4-[[(4-Oxo-1,5,6,7-tetrahydrocyclopenta[d]pyrimidin-2-yl)thio]methyl]benzoic acid methyl esterKi1526.0 [1]
(4S)-5-Amino-4-[[(2S)-2-[[(2S)-2-[[(4-bromophenyl)-hydroxyphosphoryl]methyl]-3-[3-[4-(3-chlorophenyl)phenyl]-1,2-oxazol-5-yl]propanoyl]amino]-4-carboxybutanoyl]amino]-5-oxopentanoic acidKi49.0 [1], 139.0 [2]
N-Hydroxy-1-(2-methoxyethyl)-4-[4-[4-(trifluoromethoxy)phenoxy]phenyl]sulfonylpiperidine-4-carboxamideIC500.1 [1]
(3R,4R)-N-Hydroxy-4-[[4-[[2-(trifluoromethyl)benzimidazol-1-yl]methyl]benzoyl]amino]oxane-3-carboxamideKi10000.0 [1]
4-Benzoyl-N-hydroxy-1-(4-methoxyphenylsulfonyl)piperazine-2-carboxamideIC503.0 [1], 3.02 [2]
(2S)-2-[[4-(4-Fluorophenyl)phenyl]sulfonylamino]-3-methylbutanoic acidIC5043.0 [1]
(2S)-2-[[8-(Methoxycarbonylamino)dibenzofuran-3-yl]sulfonylamino]-3-methylbutanoic acidIC50120.0 [1]
2-[4-[4-(Trifluoromethyl)phenoxy]piperidinosulfonyl]benzohydroximic acidIC5028.0 [1]
MMP-9/MMP-13 Inhibitor IIC500.89 [1], 0.9 [2]
(4-Benzylphenyl)methyl-[2-[[(2S)-3,3-dimethyl-1-(methylamino)-1-oxobutan-2-yl]carbamoyl]-4-phenylbutyl]phosphinic acidIC5014.0 [1], 21.0 [2]
2-[Methyl[4-(2-butynyloxy)phenylsulfonyl]amino]-3-methyl-5-bromobenzohydroximic acidIC50154.0 [1]
N-Hydroxy-4-[(4-methoxyphenyl)sulfonyl-(pyridin-3-ylmethyl)amino]-8-phenylquinoline-3-carboxamideIC504.0 [1]
(8S,11R,12S)-12-N-Hydroxy-8-N-(2-morpholin-4-yl-2-oxoethyl)-2,10-dioxo-11-[[4-[2-(trifluoromethyl)phenyl]phenyl]methyl]-1-oxa-3,9-diazacyclopentadecane-8,12-dicarboxamideKi653.0 [1]
4-Acetyl-N-hydroxy-1-(4-methoxyphenylsulfonyl)piperazine-2-carboxamideIC501.0 [1]
4-(Furan-2-carbonyl)-N-hydroxy-1-(4-methoxyphenylsulfonyl)piperazine-2-carboxamideIC502.5 [1], 2.51 [2]
4-(Cyclohexanecarbonyl)-N-hydroxy-1-(4-methoxyphenylsulfonyl)piperazine-2-carboxamideIC501.5 [1], 1.51 [2]
N-Hydroxy-1-(4-methoxyphenylsulfonyl)-4-(2-phenoxyacetyl)piperazine-2-carboxamideIC502.1 [1], 2.19 [2]
N-Hydroxy-1-(4-methoxyphenylsulfonyl)-4-(thiophene-2-carbonyl)piperazine-2-carboxamideIC501.9 [1], 1.91 [2]
N-Hydroxy-1-(4-methoxyphenyl)sulfonylpiperazine-2-carboxamideIC501.7 [1]
N-Hydroxy-1-(4-methoxyphenyl)sulfonyl-4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)piperazine-2-carboxamideIC5026.92 [1], 27.0 [2]
((4'-Chloro-[1,1'-biphenyl]-4-yl)sulfonyl)valineIC5048.0 [1]
4-Hexanoyl-N-hydroxy-1-(4-methoxyphenylsulfonyl)piperazine-2-carboxamideIC501.7 [1]
(2S)-2-[[4-[4-[(5-Bromo-4-methoxy-3-methyl-1-benzofuran-2-carbonyl)amino]phenyl]phenyl]sulfonylamino]-3-methylbutanoic acidIC502.3 [1]
(2R,5R)-1-[4-[(2,4-Dichlorophenyl)methoxy]phenyl]sulfonyl-N,5-dihydroxy-3,3-dimethylpiperidine-2-carboxamideIC503.0 [1], 10.0 [2]
4-Benzoyl-N-hydroxy-1-(4-phenoxyphenylsulfonyl)-1,4-diazepane-2-carboxamideIC501.29 [1], 1.3 [2]
(3S)-N-Hydroxy-4-(4-methoxyphenyl)sulfonyl-2,2-dimethyl-1,1-dioxo-1,4-thiazepane-3-carboxamideIC502.1 [1]
5-Methyl-5-(4-phenoxy-phenyl)-pyrimidine-2,4,6-trioneIC5065.0 [1]
5-Methyl-5-(4-phenoxy-phenyl)-pyrimidine-2,4,6-trioneKi65.0 [1]
2-[Benzyl(4-methoxyphenylsulfonyl)amino]-3-methylbenzenecarbohydroximic acidIC5050.0 [1], 50.12 [2]
N-Hydroxy-2-[2-methylpropyl-(4-phenylphenyl)sulfonylamino]acetamideIC509.4 [1], 39.0 [2]
N,N'-Bis(pyridin-3-ylmethyl)pyrimidine-4,6-dicarboxamideIC506600.0 [1]
(R)-N-Hydroxy-2-(4-methoxyphenylsulfonyl)-2-methyl-3-(4-(2-(piperidin-1-yl)ethoxy)phenyl)propanamideIC501.0 [1]
N-[4-[2-(Hydroxyamino)-2-oxoethyl]oxan-4-yl]-4-[(2-methylquinolin-4-yl)methoxy]benzamideKi5025.0 [1]
2-[4-[4-(Trifluoromethoxy)phenoxy]piperidinosulfonyl]benzohydroximic acidIC5033.0 [1]
1-(4-Bromobenzyl)-N-hydroxy-4-(4-methoxyphenylsulfonyl)piperidine-4-carboxamideIC502.0 [1]
2-[Methyl[4-(2-butynyloxy)phenylsulfonyl]amino]acetohydroximic acidIC5099.0 [1]
2-[Methyl[4-(2-butynyloxy)phenylsulfonyl]amino]acetohydroximic acidKi17.0 [1]
(S)-N-Hydroxy-4-(4-methoxyphenylsulfonyl)-2,2-dimethyl-1,4-thiazepane-3-carboxamideIC500.9 [1]
N-Hydroxy-4-(4-methoxyphenyl)sulfonylthiomorpholine-3-carboxamideIC501.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Matrix metalloproteinase 13 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/matrix-metalloproteinase-13-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Matrix metalloproteinase 13 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/matrix-metalloproteinase-13-inhibitors-ic50-ki.
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