Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| N-[6-[(Dimethylamino)methyl]-5,6,7,8-tetrahydronaphthalen-2-yl]-4-(4-fluorophenyl)benzamide | IC50 | 5.5 [1], 43.0 [2], 85.0 [3], 872.0 [4] | |
| N-[6-[(Dimethylamino)methyl]-5,6,7,8-tetrahydronaphthalen-2-yl]-4-(4-fluorophenyl)benzamide | Ki | 5.5 [1], 38.0 [2] | |
| N-(4-Methyl-2-(4-methylpiperazin-1-yl)quinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide | IC50 | 25.0 [1], 29.0 [2] | |
| 8-(Cyclohexylmethoxy)quinolin-2-amine | IC50 | 90.0 [1] | |
| 6-(4-Chlorophenyl)-3-(3-methoxy-4-(2-(pyrrolidin-1-yl)ethoxy)phenyl)thieno[3,2-d]pyrimidin-4(3H)-one | IC50 | 0.5 [1], 16.0 [2], 89.13 [3] | |
MLA | "Quest Database™ Melanin-concentrating hormone receptor 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 13 Nov. 2025, https://www.aatbio.com/data-sets/melanin-concentrating-hormone-receptor-1-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, November 13). Quest Database™ Melanin-concentrating hormone receptor 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/melanin-concentrating-hormone-receptor-1-inhibitors-ic50-ki. | |
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