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Melanocortin receptor 1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
Melanotan IIIC500.2 [1], 0.25 [2], 0.4 [3], 6.7 [4]
Melanotan IIKi0.11 [1]
ThiqIC502063.0 [1], 2067.0 [2]
ThiqKi300.0 [1], 760.0 [2], 1500.0 [3], 5000.0 [4]
Melanotan-1IC500.51 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMelanocortin receptor 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/melanocortin-receptor-1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseMelanocortin receptor 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/melanocortin-receptor-1-inhibitors-ic50-ki.
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