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Melatonin receptor 1A Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
MelatoninKi0.08 [1], 0.12 [2], 0.29 [3], 0.3 [4]
N-(2-(5-Methoxybenzofuran-3-yl)ethyl)acetamideIC500.6 [1], 1.58 [2]
N-(2-(5-Methoxybenzofuran-3-yl)ethyl)acetamideKi0.15 [1]
N-[2-[7-[4-[8-(2-Acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]acetamideKi0.6 [1], 3.1 [2]
N-[2-[7-[3-[8-(2-Acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamideKi0.5 [1], 3.9 [2], 112.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMelatonin receptor 1A Inhibitors (IC50, Ki)." AAT Bioquest, Inc.18 Dec2025https://www.aatbio.com/data-sets/melatonin-receptor-1a-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 18). Quest DatabaseMelatonin receptor 1A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/melatonin-receptor-1a-inhibitors-ic50-ki.
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