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Melatonin receptor 1A Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
MelatoninKi0.08 [1], 0.12 [2], 0.29 [3], 0.3 [4]
N-(2-(5-Methoxybenzofuran-3-yl)ethyl)acetamideIC500.6 [1], 1.58 [2]
N-(2-(5-Methoxybenzofuran-3-yl)ethyl)acetamideKi0.15 [1]
N-[2-[7-[4-[8-(2-Acetamidoethyl)naphthalen-2-yl]oxybutoxy]naphthalen-1-yl]ethyl]acetamideKi0.6 [1], 3.1 [2]
N-[2-[7-[3-[8-(2-Acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamideKi0.5 [1], 3.9 [2], 112.0 [3]
2-IodomelatoninIC501.0 [1]
2-IodomelatoninKi0.01 [1], 0.07 [2], 0.08 [3]
N-[2-(11-Methoxy-6,7-dihydro-5H-indolo[2,1-a][2]benzazepin-13-yl)ethyl]butanamideKi66.0 [1], 66.07 [2], 66.1 [3]
CID 10428383Ki1288.25 [1], 1290.0 [2]
CID 9998187Ki27.0 [1], 40.6 [2], 40.74 [3]
N-[2-(2-Benzyl-5-methoxy-benzofuran-3-yl)-ethyl]-acetamideIC500.02 [1]
N-[2-(2-Benzyl-5-methoxy-benzofuran-3-yl)-ethyl]-acetamideKi1.27 [1]
N-[2-(7,17-Dimethoxy-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4(9),5,7,10,14(19),15,17-heptaen-10-yl)ethyl]acetamideKi1800.0 [1], 1819.7 [2]
LuzindoleKi158.0 [1], 603.0 [2], 794.33 [3]
4-P-PdotKi59.0 [1], 104.71 [2], 501.0 [3]
N-[(6-Methoxy-9-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaenyl)methyl]acetamideKi6.17 [1], 27.0 [2]
7-AzamelatoninIC50125.89 [1]
7-AzamelatoninKi40.0 [1]
4-AzamelatoninKi0.2 [1], 0.24 [2]
N-[2-(7-Methoxy-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4(9),5,7,10,14,16,18-heptaen-10-yl)ethyl]acetamideKi316.23 [1], 319.3 [2], 320.0 [3]
1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanoneIC501000.0 [1]
1-[1-(2,2-Diphenyl-ethyl)-6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl]-ethanoneKi1000.0 [1]
N-[3-[5-Methoxy-2-[(3-methoxyphenyl)methoxy]phenyl]propyl]propanamideKi121.0 [1], 1348.96 [2], 1350.0 [3]
5-Methoxycarbonylamino-N-acetyltryptamineIC50100.0 [1], 1000.0 [2]
N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)ethyl]butanamideKi4.47 [1]
N-[2-(5-Methoxy-1-methyl-1H-indol-3-yl)-ethyl]-acetamideKi2.24 [1], 2.6 [2]
N-[2-(2,7-Dimethoxy-naphthalen-1-yl)-ethyl]-propionamideKi0.1 [1]
N-[(6-Methoxy-9-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaenyl)methyl]propanamideKi1.35 [1], 1.4 [2]
N-[(4-Methoxy-1H-indol-2-yl)methyl]propanamideKi407.38 [1]
N-[2-(5-Methoxy-2-phenyl-benzofuran-3-yl)-ethyl]-acetamideKi0.01 [1]
N-[2-[5-Methoxy-2-[(3-methoxyphenyl)methyl]-1-benzofuran-3-yl]ethyl]but-3-enamideKi21.6 [1]
N-[2-(5-Methoxy-1H-indol-2-yl)ethyl]acetamideKi16218.1 [1]
N-[(4-Methoxy-1H-indol-2-yl)methyl]cyclobutanecarboxamideKi524.81 [1]
N-[(1-Benzyl-4-methoxyindol-2-yl)methyl]propanamideKi630.96 [1]
N-[2-(1-Benzyl-5-methoxyindol-3-yl)ethyl]acetamideKi141.25 [1]
Acetylaminoethyl-methyl-phenylbutoxyphenyl-amineKi1.17 [1]
Acetamide, N-[2-(1H-indol-2-yl)ethyl]-Ki2454.71 [1]
N-[2-(4-Methoxy-1H-indol-2-yl)ethyl]acetamideKi630.96 [1]
N-[2-(4-Methoxy-1-phenylindol-2-yl)ethyl]acetamideKi87.1 [1]
N-[2-(4-Methoxy-1-phenylindol-2-yl)ethyl]propanamideKi63.1 [1]
N-[2-(6-Methoxy-1H-indol-2-yl)ethyl]acetamideKi8511.38 [1]
N-[2-(4-Methoxy-1H-indol-2-yl)ethyl]propanamideKi134.9 [1]
N-[2-(3-Bromo-6-methoxy-1H-indol-2-yl)ethyl]acetamideKi3981.07 [1]
N-[2-(1-Benzyl-4-methoxyindol-2-yl)ethyl]propanamideKi831.76 [1]
Acetamide, N-[(4-methoxy-1H-indol-2-yl)methyl]-Ki1230.27 [1]
N-[3-(5-Methoxy-1H-indol-2-yl)propyl]acetamideKi2951.21 [1]
N-[2-(7-Methoxy-1H-indol-2-yl)ethyl]acetamideKi3801.89 [1]
N-[2-(6-Methoxy-1-methylindol-2-yl)ethyl]acetamideKi1819.7 [1]
N-(3-(3-Methoxyphenyl)-3-phenylallyl)acetamideKi2.69 [1], 230.0 [2]
N-[2-(3,13-Diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-4,6,8,10,14,16,18-heptaen-10-yl)ethyl]acetamideKi1000.0 [1]
N-[2-(7-Phenyl-2,6-dihydro-1H-cyclopenta[e][1]benzofuran-8-yl)ethyl]acetamideKi0.01 [1]
N-[3-[2-(4-Phenylbutyl)-1,3-benzoxazol-7-yl]propyl]cyclopropanecarboxamideKi0.63 [1]
1-[6,7-Dimethoxy-1-(2-phenylethyl)-3,4-dihydro-1H-isoquinolin-2-yl]ethanoneIC501000.0 [1]
CID 44436051Ki7.24 [1], 40.74 [2]
N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]pyridin-1-yl)ethyl)acetamideKi1.4 [1]
N-[2-[7-[8-(2-Acetamidoethyl)naphthalen-2-yl]naphthalen-1-yl]ethyl]acetamideKi5.2 [1]
N-[2-(8-Methoxy-2-methyl-3,4-dihydro-1H-pyrazino[1,2-a]indol-10-yl)ethyl]butanamideIC503.14 [1]
N-[2-(8-Methoxy-2-methyl-3,4-dihydro-1H-pyrazino[1,2-a]indol-10-yl)ethyl]butanamideKi6.61 [1]
N-[3-Hydroxy-2-(7-methoxynaphthalen-1-yl)propyl]acetamideIC5019.95 [1]
N-[3-Hydroxy-2-(7-methoxynaphthalen-1-yl)propyl]acetamideKi10.96 [1]
N-[2-[5-(3-Phenoxypropoxy)-1H-indol-3-yl]ethyl]acetamideKi7.9 [1]
N-[2-(6-Hexoxy-3,4-dihydro-2H-chromen-4-yl)ethyl]acetamideKi1.2 [1], 3.4 [2]
DopamineKi7100.0 [1]
SerotoninKi100000.0 [1]
RamelteonKi0.01 [1]
N,N-Dimethyl-5-methoxytryptamineKi210.0 [1]
AurapteneKi1900.0 [1]
6-ChloromelatoninKi11.4 [1]
4-(4-Butylpiperidin-1-yl)-1-o-tolylbutan-1-oneKi1000.0 [1]
4-[[(E)-3,7-Dimethyl-2,6-octadienyl]oxy]-3-methoxycinnamic acidKi59000.0 [1]
7-PrenyloxycoumarinKi5200.0 [1]
7-(Benzyloxy)-2H-chromen-2-oneKi445.0 [1]
n-[(2r)-2-(6-Chloro-5-methoxy-1h-indol-3-yl)propyl]acetamideKi0.08 [1]
N-[2-(N-(4-Methoxyphenyl)anilino)ethyl]acetamideKi776.25 [1]
CID 44208891Ki90.4 [1]
5-MethoxyluzindoleKi32.7 [1]
N-Cyclopropylcarbonyl-2-(7-methoxy-1-naphthyl)ethylamineIC501.26 [1]
n-[2-(5,6-Dimethoxy-1h-indol-3-yl)ethyl]acetamideKi207.0 [1]
N-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-acetamideIC501995.26 [1]
Propanamide, N-(2-(7-methoxy-1-naphthalenyl)ethyl)-IC502.0 [1]
N-[2-(2-Phenyl-1H-indol-3-yl)ethyl]cyclobutanecarboxamideKi199.53 [1]
Acetamide,n-[2-(2-iodo-5-methoxy-1-methyl-4-nitro-1h-indol-3-yl)ethyl]-Ki1880.0 [1]
N-[(1-Benzyl-5-methoxy-3,4-dihydro-2H-quinolin-2-yl)methyl]propanamideKi17.0 [1]
N-[2-(N-(3-Methoxyphenyl)anilino)ethyl]acetamideKi4.17 [1]
Propanamide, N-(2-(7-methoxy-1-naphthalenyl)ethyl)-2-methyl-IC502.51 [1]
N-[1-[3-(3-Oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamideKi1000.0 [1]
N-[2-(6-Fluoro-5-methoxy-1H-indol-3-yl)ethyl]cyclopropanecarboxamideIC502.0 [1]
N-(3-(3-Methoxyphenyl)propyl)propionamideKi85.4 [1]
N-[3-(3-Methoxyphenyl)propyl]acetamideKi23.3 [1]
N-[2-(5-Methoxy-1-methyl-4-nitro-1H-indol-3-yl)-ethyl]-acetamideKi8560.0 [1]
N-(2-Phenoxyethyl)AcetamideKi11481.54 [1]
N-[2-(7-Methoxynaphthalen-1-yl)ethyl]hexanamideIC501995.26 [1]
N-[2-(7-Methoxynaphthalen-1-yl)ethyl]heptanamideIC50100000.0 [1]
N-[2-[3-(3-Aminophenyl)-7-methoxynaphthalen-1-yl]ethyl]acetamideKi82.0 [1]
N-[2-(3-Methoxy-N-methylanilino)ethyl]acetamideKi0.81 [1]
EfppeaKi0.06 [1]
N-(2-(7-Methoxynaphth-1-yl)ethyl)pyrrolidin-2-oneIC50100.0 [1]
1H-Indole-2-carboxamide, N-(2-(7-methoxy-1-naphthalenyl)ethyl)-IC502511.89 [1]
ACETAMIDE, N-(2-(5-METHOXYBENZO(b)THIEN-3-YL)ETHYL)-IC501.26 [1]
Items per page: 1 - 10 of 99
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References

This online tool may be cited as follows

MLA

"Quest Database™ Melatonin receptor 1A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/melatonin-receptor-1a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Melatonin receptor 1A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/melatonin-receptor-1a-inhibitors-ic50-ki.
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