Structure | Compound Name | Standard Type | Standard Values (in nM) |
---|---|---|---|
Melatonin | IC50 | 2.2 [1] | |
Melatonin | Ki | 0.08 [1], 1.1 [2] | |
6-Chloromelatonin | IC50 | 0.04 [1], 3.6 [2] | |
6-Chloromelatonin | Ki | 0.99 [1], 2.2 [2] | |
N-[2-(5-Methoxy-2-phenyl-1H-indol-3-yl)ethyl]acetamide | IC50 | 0.06 [1] | |
MLA | "Quest Database™ Melatonin receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 Oct. 2025, https://www.aatbio.com/data-sets/melatonin-receptor-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, October 10). Quest Database™ Melatonin receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/melatonin-receptor-inhibitors-ic50-ki. | |
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