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Melatonin receptor Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
MelatoninIC502.2 [1]
MelatoninKi0.08 [1], 1.1 [2]
6-ChloromelatoninIC500.04 [1], 3.6 [2]
6-ChloromelatoninKi0.99 [1], 2.2 [2]
N-[2-(5-Methoxy-2-phenyl-1H-indol-3-yl)ethyl]acetamideIC500.06 [1]
N-[2-(5-Methoxy-2-phenyl-1H-indol-3-yl)ethyl]acetamideKi0.02 [1], 0.06 [2]
N-(2-(2-Bromo-5-methoxy-1H-indol-3-yl)ethyl)acetamideIC500.13 [1]
N-(2-(2-Bromo-5-methoxy-1H-indol-3-yl)ethyl)acetamideKi0.04 [1], 0.06 [2]
N-[2-(6-Methoxy-2-phenylindol-1-yl)ethyl]propanamideIC500.05 [1], 0.19 [2], 1.18 [3]
N-[2-(6-Methoxy-2-phenylindol-1-yl)ethyl]propanamideKi0.01 [1]
N-[2-(5-Methoxyindol-1-yl)ethyl]propanamideIC505400.0 [1], 10400.0 [2], 10500.0 [3]
N-[2-(5-Methoxyindol-1-yl)ethyl]propanamideKi1500.0 [1]
N-(2-Bromo-6-methoxy-1,3,4,5-tetrahydrobenzo[cd]indol-4-yl)acetamideIC5073.0 [1], 89.5 [2], 396.0 [3]
N-(2-Bromo-6-methoxy-1,3,4,5-tetrahydrobenzo[cd]indol-4-yl)acetamideKi20.0 [1]
N-(6-Methoxy-1,3,4,5-tetrahydrobenzo[cd]indol-4-yl)acetamideIC501200.0 [1], 3110.0 [2], 8970.0 [3]
N-(6-Methoxy-1,3,4,5-tetrahydrobenzo[cd]indol-4-yl)acetamideKi330.0 [1]
CID 44303129IC501.07 [1], 1.4 [2], 2.99 [3]
CID 44303129Ki0.39 [1]
N-(2-Indol-1-ylethyl)cyclopropanecarboxamideIC502250.0 [1], 3200.0 [2], 5700.0 [3]
N-(2-Indol-1-ylethyl)cyclopropanecarboxamideKi880.0 [1]
AgomelatineIC500.08 [1]
AgomelatineKi0.1 [1]
2-IodomelatoninIC500.01 [1]
2-IodomelatoninKi0.02 [1]
5-Hydroxyethoxy-N-acetyltryptamineIC501020.0 [1]
5-Hydroxyethoxy-N-acetyltryptamineKi289.0 [1]
3-AcetylaminocarbazoleIC503000.0 [1]
3-AcetylaminocarbazoleKi820.0 [1]
N-[2-(5-Methoxy-1-methyl-1H-indol-3-yl)-ethyl]-acetamideIC5025.5 [1]
N-[2-(5-Methoxy-1-methyl-1H-indol-3-yl)-ethyl]-acetamideKi6.72 [1]
6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carbolin-1-oneIC5033000.0 [1]
6-Methoxy-2,3,4,9-tetrahydro-1H-beta-carbolin-1-oneKi9100.0 [1]
N-[2-(5-Methoxy-1H-indol-3-yl)ethyl]cyclopropanecarboxamideIC500.0 [1]
N-[2-(5-Methoxy-1H-indol-3-yl)ethyl]cyclopropanecarboxamideKi2.2 [1]
N-[2-(2-Phenyl-1H-indol-3-yl)ethyl]cyclobutanecarboxamideIC507100.0 [1]
N-[2-(2-Phenyl-1H-indol-3-yl)ethyl]cyclobutanecarboxamideKi1900.0 [1]
Ethyl 3-(acetamidomethyl)-6-methoxy-1,3,4,5-tetrahydrobenzo[cd]indole-2-carboxylateIC501.7 [1]
Ethyl 3-(acetamidomethyl)-6-methoxy-1,3,4,5-tetrahydrobenzo[cd]indole-2-carboxylateKi0.48 [1]
N-[2-(2-Bromo-6-methoxyindol-1-yl)ethyl]propanamideIC500.16 [1]
N-[2-(2-Bromo-6-methoxyindol-1-yl)ethyl]propanamideKi0.04 [1]
N-[2-(6-Methoxyindol-1-yl)ethyl]propanamideIC507.1 [1]
N-[2-(6-Methoxyindol-1-yl)ethyl]propanamideKi1.9 [1]
N-[2-(1-Benzyl-5-methoxyindol-3-yl)ethyl]acetamideIC501090.0 [1]
N-[2-(1-Benzyl-5-methoxyindol-3-yl)ethyl]acetamideKi287.0 [1]
N-Acetyl-6-methoxytryptamineIC504800.0 [1]
N-Acetyl-6-methoxytryptamineKi1180.0 [1]
6-Methoxy-1-[2-(acetylamino)ethyl]-1H-benzimidazoleIC505260.0 [1]
6-Methoxy-1-[2-(acetylamino)ethyl]-1H-benzimidazoleKi5000.0 [1]
N-[2-(5-Methoxy-1-phenylindol-3-yl)ethyl]acetamideIC501470.0 [1]
N-[2-(5-Methoxy-1-phenylindol-3-yl)ethyl]acetamideKi380.0 [1]
N-[2-(2-Phenylindol-1-yl)ethyl]propanamideIC5082.0 [1]
N-[2-(2-Phenylindol-1-yl)ethyl]propanamideKi23.0 [1]
N-[2-(4,5,6-Trimethoxy-1H-indol-3-yl)ethyl]acetamideIC502460.0 [1]
N-[2-(4,5,6-Trimethoxy-1H-indol-3-yl)ethyl]acetamideKi617.0 [1]
6-Methoxy-1-[2-(propionylamino)ethyl]-1H-indole-2-carboxylic acid methyl esterIC500.83 [1]
6-Methoxy-1-[2-(propionylamino)ethyl]-1H-indole-2-carboxylic acid methyl esterKi0.23 [1]
N-[2-(6-Methoxyindol-1-yl)ethyl]acetamideIC5012.0 [1]
N-[2-(6-Methoxyindol-1-yl)ethyl]acetamideKi3.4 [1]
N-[2-(5-Methoxy-1H-indol-4-yl)ethyl]acetamideIC501300.0 [1]
N-[2-(5-Methoxy-1H-indol-4-yl)ethyl]acetamideKi360.0 [1]
N-[2-(5,7-Dimethoxy-1H-indol-3-yl)ethyl]acetamideIC50491.0 [1]
N-[2-(5,7-Dimethoxy-1H-indol-3-yl)ethyl]acetamideKi121.0 [1]
N-[(6-Methoxy-1,3,4,5-tetrahydrobenzo[cd]indol-3-yl)methyl]acetamideIC509.9 [1]
N-[(6-Methoxy-1,3,4,5-tetrahydrobenzo[cd]indol-3-yl)methyl]acetamideKi2.7 [1]
3-(Acetylamino)-6-methoxy-9H-carbazoleIC50230.0 [1]
3-(Acetylamino)-6-methoxy-9H-carbazoleKi63.0 [1]
Propanamide,n-[2-(2-iodo-5-methoxy-1h-indol-1-yl)ethyl]-IC50360.0 [1]
Propanamide,n-[2-(2-iodo-5-methoxy-1h-indol-1-yl)ethyl]-Ki99.0 [1]
N-[2-(5-Chloro-1H-indol-3-yl)ethyl]acetamideIC50126.0 [1]
N-[2-(5-Chloro-1H-indol-3-yl)ethyl]acetamideKi30.0 [1]
N-[2-(7-Methoxy-1H-indol-3-yl)ethyl]acetamideIC502620.0 [1]
N-[2-(7-Methoxy-1H-indol-3-yl)ethyl]acetamideKi647.0 [1]
N-[2-(5-Bromo-1H-indol-3-yl)ethyl]acetamideIC5033.6 [1]
N-[2-(5-Bromo-1H-indol-3-yl)ethyl]acetamideKi8.91 [1]
N-[2-(4-Methoxy-1H-indol-3-yl)ethyl]acetamideIC50772.0 [1]
N-[2-(4-Methoxy-1H-indol-3-yl)ethyl]acetamideKi190.0 [1]
CID 44303043IC5029.0 [1]
CID 44303043Ki8.0 [1]
N-[2-(5-Fluoro-1H-indol-3-yl)ethyl]acetamideIC50295.0 [1]
N-[2-(5-Fluoro-1H-indol-3-yl)ethyl]acetamideKi72.8 [1]
N-[2-(5-Methyl-1H-indol-3-yl)ethyl]acetamideIC50719.0 [1]
N-[2-(5-Methyl-1H-indol-3-yl)ethyl]acetamideKi180.0 [1]
N-(2-Indol-1-ylethyl)cyclobutanecarboxamideIC5018000.0 [1]
N-(2-Indol-1-ylethyl)cyclobutanecarboxamideKi5000.0 [1]
2,2,2-Trifluoro-N-[2-(6-methoxyindol-1-yl)ethyl]acetamideIC5035.0 [1]
2,2,2-Trifluoro-N-[2-(6-methoxyindol-1-yl)ethyl]acetamideKi9.6 [1]
N-[2-(2,4-Dibromo-5-methoxy-1H-indol-3-yl)ethyl]acetamideIC5023.3 [1]
N-[2-(2,4-Dibromo-5-methoxy-1H-indol-3-yl)ethyl]acetamideKi5.75 [1]
N-[2-(2-Phenylindol-1-yl)ethyl]cyclobutanecarboxamideIC5010000.0 [1]
N-[2-(2-Phenylindol-1-yl)ethyl]cyclobutanecarboxamideKi2800.0 [1]
6-Methoxy-1-[3-(propionylamino)propyl]-1H-indole-2-carboxylic acid methyl esterIC504.8 [1]
6-Methoxy-1-[3-(propionylamino)propyl]-1H-indole-2-carboxylic acid methyl esterKi1.3 [1]
N-[2-(6-Methoxyindol-1-yl)ethyl]butanamideIC5011.0 [1]
N-[2-(6-Methoxyindol-1-yl)ethyl]butanamideKi3.0 [1]
N-[2-(6-Methoxyindol-1-yl)ethyl]cyclopropanecarboxamideIC5089.0 [1]
N-[2-(6-Methoxyindol-1-yl)ethyl]cyclopropanecarboxamideKi24.0 [1]
(4Ar,9bS)-7-chloro-8-methoxy-2,3,4,4a,5,9b-hexahydro-1H-indeno[1,2-b]pyridineKi10000.0 [1]
1-[(4Ar,9bS)-7-chloro-8-methoxy-2,3,4,4a,5,9b-hexahydroindeno[1,2-b]pyridin-1-yl]ethanoneKi10000.0 [1]
(4Ar,9bS)-7-chloro-N-ethyl-8-methoxy-2,3,4,4a,5,9b-hexahydroindeno[1,2-b]pyridine-1-carboxamideKi190.0 [1], 670.0 [2]
(2S,7R)-12,14-Dioxa-3-azatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),9,11(15)-trieneKi10000.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Melatonin receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/melatonin-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Melatonin receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/melatonin-receptor-inhibitors-ic50-ki.
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