Membrane-bound transcription factor site-1 protease Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(R)-4-((Diethylamino)methyl)-N-(2-methoxyphenethyl)-N-(pyrrolidin-3-yl)benzamide	IC50	170.0 [1]
	CID 44433047	IC50	8.0 [1]
	N-(2-Chlorophenethyl)-4-isopropoxy-N-(pyrrolidin-3-yl)benzamide	IC50	1400.0 [1]
	N-(2-Fluorophenethyl)-4-isopropoxy-N-(pyrrolidin-3-yl)benzamide	IC50	9000.0 [1]
	N-(3-Chlorophenethyl)-4-isopropoxy-N-(pyrrolidin-3-yl)benzamide	IC50	9600.0 [1]
	N-(2-Methoxyphenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamide	IC50	540.0 [1]
	N-(2-Methoxyphenethyl)-4-(benzyloxy)-N-(pyrrolidin-3-yl)benzamide	IC50	310.0 [1]
	N-(2-Chlorophenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamide	IC50	840.0 [1]
	N-(2-Chlorophenethyl)-4-(benzyloxy)-N-(pyrrolidin-3-yl)benzamide	IC50	590.0 [1]
	N-(2-Chlorobenzyl)-4-isopropoxy-N-(pyrrolidin-3-yl)benzamide	IC50	5000.0 [1]
	N-(2,6-Dichlorophenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamide	IC50	430.0 [1]
	N-(4-Chlorophenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamide	IC50	3700.0 [1]
	N-(3-Chlorophenethyl)-4-(benzyloxy)-N-(pyrrolidin-3-yl)benzamide	IC50	510.0 [1]
	4-Diethylaminomethyl-N-pyrrolidin-3-yl-N-(2-o-tolyl-ethyl)-benzamide	IC50	1600.0 [1]
	N-(2-Ethoxyphenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamide	IC50	16000.0 [1]
	N-(2-Chlorophenethyl)-4-isopropoxy-N-(1-methylpyrrolidin-3-yl)benzamide	IC50	30000.0 [1]
	N-(2-Chlorophenethyl)-4-isopropoxy-N-(tetrahydrothiophen-3-yl)benzamide	IC50	30000.0 [1]
	N-(2-Chlorophenethyl)-N-(1-formylpyrrolidin-3-yl)-4-isopropoxybenzamide	IC50	30000.0 [1]
	N-(2-Chlorophenethyl)-4-isopropoxy-N-(piperidin-3-yl)benzamide	IC50	30000.0 [1]
	N-(2-Chlorophenethyl)-N-(azetidin-3-yl)-4-isopropoxybenzamide	IC50	30000.0 [1]
	N-(2-Chlorophenethyl)-4-(piperidin-1-ylmethyl)-N-(tetrahydrofuran-3-yl)benzamide	IC50	30000.0 [1]
	N-[2-(2-Methoxyphenyl)ethyl]-4-[[3-(2-methylphenyl)piperidin-1-yl]methyl]-N-pyrrolidin-3-ylbenzamide	IC50	37.0 [1]
	4-(6-Azabicyclo[3.2.1]octan-6-ylmethyl)-N-[2-(2-methoxyphenyl)ethyl]-N-pyrrolidin-3-ylbenzamide	IC50	29.0 [1]
	4-(2-Azabicyclo[2.2.1]heptan-2-ylmethyl)-N-[2-(2-methoxyphenyl)ethyl]-N-pyrrolidin-3-ylbenzamide	IC50	95.0 [1]
	4-[[[(1S,2S)-2-Hydroxycyclohexyl]amino]methyl]-N-[2-(2-methoxyphenyl)ethyl]-N-pyrrolidin-3-ylbenzamide	IC50	100.0 [1]
	N-(2-Methoxyphenethyl)-4-(piperidin-1-ylmethyl)-N-(pyrrolidin-3-yl)benzamide	IC50	250.0 [1]
	4-[[(2S)-2-(Methoxymethyl)pyrrolidin-1-yl]methyl]-N-[2-(2-methoxyphenyl)ethyl]-N-pyrrolidin-3-ylbenzamide	IC50	140.0 [1]
	1-[[4-[2-(2-Methoxyphenyl)ethyl-pyrrolidin-3-ylcarbamoyl]phenyl]methyl]piperidine-3-carboxamide	IC50	160.0 [1]
	(S)-N-(2-Methoxyphenethyl)-4-((diethylamino)methyl)-N-(pyrrolidin-3-yl)benzamide	IC50	970.0 [1]
	Benzyl (2S)-3-methyl-2-[[2-[2-[[2-[2-[[(2S)-3-methyl-1-oxo-1-phenylmethoxybutan-2-yl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]butanoate	Ki	125000.0 [1]
	Benzyl (2S)-2-[[2-[2-[[2-[2-oxo-2-[[(2S)-1-oxo-3-phenyl-1-phenylmethoxypropan-2-yl]amino]ethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-phenylpropanoate	Ki	11800.0 [1]
	(2S)-2-[[2-[2-[[2-[2-[[(1S)-1-Carboxy-2-methylpropyl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-methylbutanoic acid	Ki	75000.0 [1]
	(2S)-2-[[2-[2-[[2-[2-[[(1S)-1-Carboxy-2-phenylethyl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-phenylpropanoic acid	Ki	225000.0 [1]
	2-[[2-[2-[[2-[2-(Carboxymethylamino)-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]acetic acid	Ki	265000.0 [1]
	(2S)-2-[[(2S)-2-[[2-[2-[[2-[2-[[(2S)-1-[[(1S)-1-Carboxy-2-phenylethyl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethoxy]phenyl]diazenyl]phenoxy]acetyl]amino]-3-phenylpropanoyl]amino]-3-phenylpropanoic acid	Ki	140000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 35 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Membrane-bound transcription factor site-1 protease Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/membrane-bound-transcription-factor-site-1-protease-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Membrane-bound transcription factor site-1 protease Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/membrane-bound-transcription-factor-site-1-protease-inhibitors-ic50-ki.
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