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Menin/Histone-lysine N-methyltransferase MLL Inhibitors (IC50, Ki)
Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
 | 4-(2-Benzyl-2,7-diazaspiro[3.4]octan-7-yl)-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidine | IC50 | 56.0 [1], 144.0 [2] |
 | 4-[2-(2-Methyl-4,5,6,7-tetrahydroindazol-4-yl)-2,7-diazaspiro[3.4]octan-7-yl]-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidine | IC50 | 120.0 [1], 385.0 [2] |
 | 4-(2-Benzyl-2,7-diazaspiro[4.5]decan-7-yl)-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidine | IC50 | 140.0 [1], 227.0 [2] |
 | [(6S)-5-Azaspiro[2.4]heptan-6-yl]-[7-[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]-2,7-diazaspiro[3.4]octan-2-yl]methanone | IC50 | 92.0 [1], 102.0 [2] |
 | 4-[2-[(1R)-1-(Azetidin-3-yl)-2-methylpropyl]-2,7-diazaspiro[3.4]octan-7-yl]-6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidine | IC50 | 8.0 [1], 21.0 [2] |
References
This online resource may be cited as follows
MLA | "Quest Database™ Menin/Histone-lysine N-methyltransferase MLL Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2025, https://www.aatbio.com/data-sets/menin-histone-lysine-n-methyltransferase-mll-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, November 21). Quest Database™ Menin/Histone-lysine N-methyltransferase MLL Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/menin-histone-lysine-n-methyltransferase-mll-inhibitors-ic50-ki. | |
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