Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| 2-Methyl-6-(phenylethynyl)pyridine | IC50 | 22.0 [1] | |
| 2-Methyl-4-(pyridin-3-ylethynyl)thiazole | IC50 | 5.0 [1], 47.3 [2], 462.0 [3] | |
| 2-Methyl-4-(pyridin-3-ylethynyl)thiazole | Ki | 32.7 [1] | |
| Fenobam | IC50 | 36.3 [1], 43.0 [2], 330.0 [3] | |
| Fenobam | Ki | 6.76 [1], 31.62 [2], 162.2 [3] | |
MLA | "Quest Database™ Metabotropic glutamate receptor 5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 31 Dec. 2025, https://www.aatbio.com/data-sets/metabotropic-glutamate-receptor-5-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 31). Quest Database™ Metabotropic glutamate receptor 5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/metabotropic-glutamate-receptor-5-inhibitors-ic50-ki. | |
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