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Metabotropic glutamate receptor 5 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
2-Methyl-6-(phenylethynyl)pyridineIC5022.0 [1]
2-Methyl-4-(pyridin-3-ylethynyl)thiazoleIC505.0 [1], 47.3 [2], 462.0 [3]
2-Methyl-4-(pyridin-3-ylethynyl)thiazoleKi32.7 [1]
FenobamIC5036.3 [1], 43.0 [2], 330.0 [3]
FenobamKi6.76 [1], 31.62 [2], 162.2 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMetabotropic glutamate receptor 5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.31 Dec2025https://www.aatbio.com/data-sets/metabotropic-glutamate-receptor-5-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 31). Quest DatabaseMetabotropic glutamate receptor 5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/metabotropic-glutamate-receptor-5-inhibitors-ic50-ki.
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