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Methionine aminopeptidase 2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
O-(Chloroacetylcarbamoyl)fumagillolIC501.0 [1], 1050.0 [2], 1320.0 [3]
O-(Chloroacetylcarbamoyl)fumagillolKi1.0 [1]
4-(p-Tolyl)-1H-1,2,3-triazoleIC5010.0 [1]
4-(p-Tolyl)-1H-1,2,3-triazoleKi4.2 [1], 15.0 [2], 4400.0 [3]
2-[(Phenylsulfonyl)amino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC509.0 [1], 10.0 [2], 3300.0 [3], 4200.0 [4]
FumagillinIC500.63 [1], 1.0 [2], 1.2 [3], 30.0 [4]
8-HydroxyquinolineIC501270.0 [1], 2030.0 [2], 5600.0 [3]
4-(4-Chlorophenyl)-1H-1,2,3-triazoleKi6.0 [1], 11000.0 [2]
5-Methyl-2-[(phenylsulfonyl)amino]benzoic acidIC501000.0 [1], 1400.0 [2], 100000.0 [3]
2-[[2-(3-Piperidin-1-ylpropylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5019.95 [1], 20.0 [2], 1200.0 [3]
2-[[2-(3-Pyrrolidin-1-ylpropylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5016.98 [1], 17.0 [2], 490.0 [3]
2-[[2-(Piperidin-3-ylmethylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5034.67 [1], 35.0 [2], 1600.0 [3]
2-[[2-[2-(1-Methylpyrrolidin-2-yl)ethylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5016.98 [1], 17.0 [2], 560.0 [3]
2-[[2-[3-(Diethylamino)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5025.0 [1], 181.97 [2], 950.0 [3]
2-[[2-(2-Pyrrolidin-1-ylethylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5069.0 [1], 69.18 [2], 1500.0 [3]
2-[[4-Chloro-2-[3-(diethylamino)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC50109.65 [1], 110.0 [2], 1400.0 [3]
2-[[2-[2-[1-(Cyclohexylmethyl)pyrrolidin-2-yl]ethylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC50150.0 [1], 151.36 [2], 23000.0 [3]
2-[[2-(Pyridin-4-ylmethylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5034.67 [1], 35.0 [2], 11000.0 [3]
2-[[2-[[1-(1-Methylpiperidin-4-yl)piperidin-4-yl]methylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5054.95 [1], 55.0 [2], 2500.0 [3]
2-[[2-(2-Pyridin-4-ylethylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5015.85 [1], 16.0 [2], 5700.0 [3]
2-[[2-[[3-(Dimethylamino)-2,2-dimethylpropyl]amino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5018.0 [1], 18.2 [2], 780.0 [3]
2-[[2-[3-(Diethylamino)propylamino]-4-methylphenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC50150.0 [1], 151.36 [2], 3200.0 [3]
2-[(2-Aminophenyl)sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5012.88 [1], 13.0 [2], 7300.0 [3]
2-[[2-[2-(Dimethylamino)ethylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5047.86 [1], 48.0 [2], 560.0 [3]
2-[[2-(2-Pyrrolidin-2-ylethylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5021.88 [1], 22.0 [2], 550.0 [3]
2-[[2-(2-Pyridin-2-ylethylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5052.48 [1], 53.0 [2], 12000.0 [3]
2-[[2-[(1-Methylpiperidin-4-yl)methylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5015.0 [1], 15.14 [2], 1200.0 [3]
2-[[2-[3-(Dimethylamino)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5014.0 [1], 14.13 [2], 470.0 [3]
2-[[2-[4-(Dimethylamino)butylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5012.0 [1], 12.02 [2], 630.0 [3]
2-[[5-Chloro-2-[3-(diethylamino)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5056.0 [1], 56.23 [2], 1700.0 [3]
2-[[2-[2-(1-Cyclohexylpyrrolidin-2-yl)ethylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5069.0 [1], 69.18 [2], 9100.0 [3]
2-[[2-(3-Morpholin-4-ylpropylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5021.88 [1], 22.0 [2], 5900.0 [3]
2-[[2-[2-(Diethylamino)ethylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5030.9 [1], 31.0 [2], 480.0 [3]
2-[[2-[3-(4-Piperidin-1-ylpiperidin-1-yl)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5057.54 [1], 58.0 [2], 1400.0 [3]
2-[[2-[2-[Di(propan-2-yl)amino]ethylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5030.9 [1], 31.0 [2], 410.0 [3]
2-[[2-[2-(1-Propan-2-ylpyrrolidin-2-yl)ethylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5061.66 [1], 62.0 [2], 680.0 [3]
2-[[2-[3-[Methyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC50109.65 [1], 110.0 [2], 37000.0 [3]
2-[[2-[3-(2-Hydroxyethylamino)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5015.0 [1], 15.14 [2], 490.0 [3]
2-[[2-[3-(Diethylamino)propylamino]-5-methylphenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5066.0 [1], 66.07 [2], 2300.0 [3]
2-[[2-(3-Aminopropylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5012.88 [1], 13.0 [2], 360.0 [3]
2-[[2-[3-(2-Oxopyrrolidin-1-yl)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5039.81 [1], 40.0 [2], 11000.0 [3]
2-[[2-(Piperidin-4-ylmethylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5016.98 [1], 17.0 [2], 1200.0 [3]
2-[[2-[3-[Bis(2-hydroxyethyl)amino]propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5025.7 [1], 26.0 [2], 490.0 [3]
2-[[2-[2-[1-(1-Methylpiperidin-4-yl)pyrrolidin-2-yl]ethylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5070.0 [1], 70.79 [2], 420.0 [3]
2-[[2-(Pyrrolidin-3-ylmethylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5033.88 [1], 34.0 [2], 790.0 [3]
2-[[2-[(1-Propan-2-ylpiperidin-4-yl)methylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5045.71 [1], 46.0 [2], 3600.0 [3]
2-[[2-[3-[(2-Methylpropan-2-yl)oxycarbonylamino]propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5077.0 [1], 77.62 [2], 26000.0 [3]
2-[[2-[3-(Diethylamino)propylamino]-6-fluorophenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5019.0 [1], 19.05 [2], 410.0 [3]
2-[[2-(3-Imidazol-1-ylpropylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5010.0 [1], 3300.0 [2]
2-[[2-[3-(4-Methylpiperazin-1-yl)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5025.7 [1], 26.0 [2], 2100.0 [3]
4-(4-Bromophenyl)-1H-1,2,3-triazoleKi3.0 [1], 11000.0 [2]
5-(3,4-Dibromophenyl)-1H-1,2,3-triazoleKi1.0 [1], 16000.0 [2]
5-Methyl-2-(1H-1,2,3-triazol-5-yl)pyridineKi3.0 [1], 15000.0 [2]
Pyridine, 4-methyl-2-(1H-1,2,3-triazol-5-yl)-Ki8.0 [1], 14000.0 [2]
8-HydroxyquinaldineIC502030.0 [1], 15000.0 [2]
5-Chloro-8-hydroxyquinolineIC5055.0 [1], 1270.0 [2]
Bengamide AIC50400.0 [1], 11000.0 [2]
2-[(2,1,3-Benzothiadiazol-4-ylsulfonyl)amino]-5-bromobenzoic acidIC503900.0 [1], 100000.0 [2]
Tert-Butyl {2-[(1,3-Thiazol-2-Ylamino)carbonyl]pyridin-3-Yl}carbamateIC50300000.0 [1]
4-(3-Methylphenyl)-1H-1,2,3-triazoleIC5018.0 [1]
4-(3-Methylphenyl)-1H-1,2,3-triazoleKi18.0 [1]
5-Bromo-2-{[(4-chlorophenyl)sulfonyl]amino}benzoic acidIC509100.0 [1], 100000.0 [2]
2-[[3-Chloro-2-[3-(diethylamino)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5015.14 [1], 190.0 [2]
2-[[2-[3-(Ethylamino)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5012.02 [1], 400.0 [2]
N-(2-Isopropylphenyl)-3-[(2-Thienylmethyl)thio]-1h-1,2,4-Triazol-5-AmineKi2.0 [1], 1500.0 [2]
3-(Furan-2-ylmethylsulfanyl)-N-(2-propan-2-ylphenyl)-1H-1,2,4-triazol-5-amineKi3.0 [1], 1500.0 [2]
3-(Furan-3-ylmethylsulfanyl)-N-(2-propan-2-ylphenyl)-1H-1,2,4-triazol-5-amineKi24.0 [1], 1800.0 [2]
3-Anilino-5-benzylthio-1,2,4-triazoleKi0.5 [1], 180.0 [2]
5-Ethyl-2-[(4-fluorophenyl)sulfonylamino]benzoic acidIC5055.0 [1], 4200.0 [2]
N-Phenyl-3-(thiophen-2-ylmethylsulfanyl)-1H-1,2,4-triazol-5-amineKi0.75 [1], 630.0 [2]
Benzoic acid, 5-ethyl-2-[(phenylsulfonyl)amino]-IC5090.0 [1], 100000.0 [2]
1H-1,2,3-Triazole, 5-(2-benzofuranyl)-Ki13.0 [1]
2-[[2-(2-Piperidin-1-ylethylcarbamoyl)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5050.0 [1], 190.0 [2]
2-[[2-[(Z)-3-Pyrrolidin-1-ylprop-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5020.0 [1], 270.0 [2]
2-[[2-[3-(Diethylamino)propyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC509.0 [1], 440.0 [2]
2-[[2-(2-Piperidin-1-ylethylcarbamoylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5082.0 [1], 440.0 [2]
2-[[2-[2-(Dimethylamino)ethylsulfinyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5054.0 [1], 260.0 [2]
2-[[2-[4-(Diethylamino)butyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5019.0 [1], 1000.0 [2]
2-[[2-[5-(Diethylamino)pentyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5045.0 [1], 3400.0 [2]
2-[[2-[(1,2,2,6,6-Pentamethylpiperidin-4-yl)amino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5091.0 [1], 4600.0 [2]
2-[[2-[2-(Dimethylamino)ethylsulfanyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5052.0 [1], 900.0 [2]
2-[[2-[(E)-3-[2-Hydroxyethyl(methyl)amino]prop-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5015.0 [1], 120.0 [2]
2-[[2-[2-(Diethylamino)ethylsulfanyl]-4-fluorophenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5037.0 [1], 310.0 [2]
2-[[2-(4-Pyrrolidin-1-ylbutanoylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5042.0 [1], 210.0 [2]
2-[[2-[3-(Dibutylamino)propylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5052.0 [1], 1900.0 [2]
2-[[2-[2-(Dimethylamino)ethylsulfinyl]-4-fluorophenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5062.0 [1], 300.0 [2]
2-[[2-[(E)-3-(Dimethylamino)prop-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5027.0 [1], 410.0 [2]
2-[[2-[(E)-3-[Ethyl(methyl)amino]prop-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC509.0 [1], 180.0 [2]
2-[[2-[(Z)-3-(Diethylamino)but-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5019.0 [1], 280.0 [2]
2-[[2-(3-Piperidin-1-ylpropylcarbamoylamino)phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5042.0 [1], 410.0 [2]
2-[[2-[(E)-5-(Diethylamino)pent-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5020.0 [1], 1000.0 [2]
2-[[2-[(E)-3-[Methyl(propan-2-yl)amino]prop-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5012.0 [1], 170.0 [2]
2-[[4-Fluoro-2-[(Z)-3-pyrrolidin-1-ylbut-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5010.0 [1], 120.0 [2]
2-[[2-[5-(Diethylamino)pentan-2-ylcarbamoyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC50170.0 [1], 1000.0 [2]
2-[[2-[(Z)-3-Pyrrolidin-1-ylbut-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5030.0 [1], 560.0 [2]
2-[[2-[(Z)-4-(Diethylamino)but-1-enyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5016.0 [1], 470.0 [2]
2-[[2-[3-(Diethylamino)propylsulfanyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5043.0 [1], 1200.0 [2]
2-[[2-[2-(1-Methylpyrrolidin-2-yl)ethylcarbamoyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5037.0 [1], 170.0 [2]
2-[[2-[3-(Diethylamino)propylcarbamoyl]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5025.0 [1], 200.0 [2]
2-[[2-[2-(Diethylamino)ethoxycarbonylamino]phenyl]sulfonylamino]-5,6,7,8-tetrahydronaphthalene-1-carboxylic acidIC5051.0 [1], 490.0 [2]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Methionine aminopeptidase 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/methionine-aminopeptidase-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Methionine aminopeptidase 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/methionine-aminopeptidase-2-inhibitors-ic50-ki.
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