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Microsomal triglyceride transfer protein large subunit Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
LomitapideIC500.8 [1], 8.0 [2]
DirlotapideIC500.01 [1], 2.7 [2], 2.9 [3]
Unii-0Z473OO6GBIC500.03 [1], 1.0 [2]
3-Methyl-N-[(2S)-2-(pyridin-2-ylmethylamino)-2,3-dihydro-1H-inden-5-yl]-2-[4-(trifluoromethyl)phenyl]benzamideIC50100.0 [1], 2350.0 [2]
Methyl N-[(2S)-5-[[3-methyl-2-[4-(trifluoromethyl)phenyl]benzoyl]amino]-2,3-dihydro-1H-inden-2-yl]carbamateIC504.3 [1], 70.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMicrosomal triglyceride transfer protein large subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc.17 Dec2025https://www.aatbio.com/data-sets/microsomal-triglyceride-transfer-protein-large-subunit-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 17). Quest DatabaseMicrosomal triglyceride transfer protein large subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/microsomal-triglyceride-transfer-protein-large-subunit-inhibitors-ic50-ki.
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