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Microtubule-associated protein 2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
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▼
EbselenIC502430.0 [1]
Ebselen diselenideIC50230.0 [1]
5-Bromo-1H-indazoleIC5037000.0 [1]
5-Chloro-6-methyl-N-(2-phenylethyl)-2-pyridin-2-ylpyrimidin-4-amineIC509000.0 [1]
N'-(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-N-[5-(trifluoromethyl)pyridin-2-yl]ethane-1,2-diamineIC50100000.0 [1]
2-{4-[5-Chloro-6-Methyl-2-(Pyridin-2-Yl)pyrimidin-4-Yl]piperazin-1-Yl}ethanolIC50100000.0 [1]
5-Chloro-N-[1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl]-6-methyl-2-pyridin-2-ylpyrimidin-4-amineIC50100000.0 [1]
2-Methyl-1,2-benzoselenazol-3-oneIC5010400.0 [1]
6-Bromo-1H-indazoleIC501100.0 [1]
1,2-Benzoselenazol-3-oneIC504970.0 [1]
N'-(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-N-[6-(trifluoromethyl)pyridin-2-yl]ethane-1,2-diamineIC50100000.0 [1]
N-Benzyl-5-chloro-6-methyl-2-pyridin-3-ylpyrimidin-4-amineIC50100000.0 [1]
4-Benzylsulfanyl-5-chloro-6-methyl-2-pyridin-2-ylpyrimidineIC50100000.0 [1]
N-Benzyl-5-chloro-N,6-dimethyl-2-pyridin-2-ylpyrimidin-4-amineIC5013000.0 [1]
6-Methyl-N-(2-phenylethyl)-2-pyridin-2-ylpyrimidin-4-amineIC50100000.0 [1]
2-(2-Phenylethyl)-1,2-benzoselenazol-3-oneIC507570.0 [1]
6-(1-Methylpyrazol-4-yl)-1H-indazoleIC50100000.0 [1]
7-[5-(4-Methylpiperazin-1-yl)pyridin-3-yl]-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,5]naphthyridin-4-oneIC5024000.0 [1]
7-(4-Fluorophenyl)-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,5]naphthyridin-4-oneIC50234000.0 [1]
7-(2-Methylphenyl)-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,5]naphthyridin-4-oneIC503000.0 [1]
5-(2,2,2-Trifluoroethyl)-7-[2-(trifluoromethyl)phenyl]-1H-pyrazolo[4,3-c][1,5]naphthyridin-4-oneIC5020000.0 [1]
2-[4-Oxo-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,5]naphthyridin-7-yl]benzamideIC501020000.0 [1]
N-Methyl-2-[4-oxo-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,5]naphthyridin-7-yl]benzenesulfonamideIC504000.0 [1]
N-[2-[4-Oxo-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,5]naphthyridin-7-yl]phenyl]methanesulfonamideIC508000.0 [1]
7-[6-(4-Methylpiperazin-1-yl)pyridin-3-yl]-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,5]naphthyridin-4-oneIC505000.0 [1]
7-(2-Morpholin-4-ylphenyl)-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,5]naphthyridin-4-oneIC50187000.0 [1]
7-[2-[(Cyclopropylamino)methyl]phenyl]-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,6]naphthyridin-4-oneIC5021000.0 [1]
7-(3-Chloropyridin-2-yl)-5-(2,2,2-trifluoroethyl)-1H-pyrazolo[4,3-c][1,6]naphthyridin-4-oneIC5013000.0 [1]
6-Fluoro-4-phenyl-1H-indazoleIC50960.0 [1]
6-Methyl-4-phenyl-1H-indazoleIC50220.0 [1]
6-Methoxy-4-phenyl-1H-indazoleIC50730.0 [1]
4-Phenyl-1H-indazole-6-carbonitrileIC5062.0 [1]
4-Phenyl-6-(trifluoromethoxy)-1H-indazoleIC5091.0 [1]
6-Methylsulfonyl-4-phenyl-1H-indazoleIC50360.0 [1]
(3S)-1-[4-Methyl-5-[6-(trifluoromethyl)-1H-indazol-4-yl]pyrimidin-2-yl]pyrrolidin-3-olIC506.0 [1]
6-(1-Methylpyrazol-4-yl)-4-phenyl-1H-indazoleIC5024000.0 [1]
4-Phenyl-6-propan-2-yl-1H-indazoleIC50550.0 [1]
(3S)-1-[6-Methyl-5-[6-(trifluoromethyl)-1H-indazol-4-yl]pyridin-2-yl]pyrrolidin-3-olIC505.0 [1]
6-Chloro-4-phenyl-1H-indazoleIC5079.0 [1]
(3R)-1-[6-Methyl-5-[6-(trifluoromethyl)-1H-indazol-4-yl]pyridin-2-yl]pyrrolidin-3-olIC505.0 [1]
6-Chloro-4-pyridin-3-yl-1H-pyrazolo[4,3-b]indoleIC505.01 [1]
3-Chloro-5-(7-fluoro-1H-pyrazolo[4,3-b]indol-4-yl)pyridin-2-amineIC507.94 [1]
2-Benzyl-1,2-benzoselenazol-3-oneIC50320.0 [1]
N-(5-Chloro-2-methoxyphenyl)-2-[[2-[(5-chloro-2-methoxyphenyl)carbamoyl]phenyl]diselanyl]benzamideIC504470.0 [1]
2-(5-Chloro-2-methoxyphenyl)-1,2-benzoselenazol-3-oneIC502350.0 [1]
2-(2-Methoxy-5-methylphenyl)-1,2-benzoselenazol-3-oneIC50920.0 [1]
N-(2-Chloro-4-methylphenyl)-2-[[2-[(2-chloro-4-methylphenyl)carbamoyl]phenyl]diselanyl]benzamideIC50119200.0 [1]
2-(4-Methoxy-2-methylphenyl)-1,2-benzoselenazol-3-oneIC501350.0 [1]
2-(5-Tert-butyl-2-methoxyphenyl)-1,2-benzoselenazol-3-oneIC502670.0 [1]
2-(4-Butoxyphenyl)-1,2-benzoselenazol-3-oneIC506270.0 [1]
2-[(4-Tert-butylphenyl)methyl]-1,2-benzoselenazol-3-oneIC508850.0 [1]
1,4-Dihydropyrazolo[4,3-b]indoleIC501000.0 [1]
2-(3-Fluorophenyl)-1,2-benzoselenazol-3-oneIC50935.0 [1]
N-(2-Hydroxyphenyl)-2-[[2-[(2-hydroxyphenyl)carbamoyl]phenyl]diselanyl]benzamideIC505440.0 [1]
N-(4-Methoxyphenyl)-2-[[2-[(4-methoxyphenyl)carbamoyl]phenyl]diselanyl]benzamideIC5013900.0 [1]
N-(2-Methoxyphenyl)-2-[[2-[(2-methoxyphenyl)carbamoyl]phenyl]diselanyl]benzamideIC506790.0 [1]
Benzamide, 2,2'-diselenobis[N-(phenylmethyl)-IC503430.0 [1]
7-Fluoro-1,4-dihydropyrazolo[4,3-b]indoleIC5079.43 [1]
4-[[(2R)-1-([1,2,4]Triazolo[1,5-a]pyrimidin-7-yl)pyrrolidin-2-yl]methoxy]isoquinolineIC5038.0 [1]
4-[(2R)-2-[(3-Fluorophenoxy)methyl]pyrrolidin-1-yl]-7H-pyrrolo[2,3-d]pyrimidineIC5050000.0 [1]
2-[(2-Carbamoylphenyl)diselanyl]benzamideIC509130.0 [1]
6-[(2R)-2-[(3-Fluorophenoxy)methyl]pyrrolidin-1-yl]-7H-purineIC502000.0 [1]
6-[(2R)-2-[(2,3-Difluorophenoxy)methyl]pyrrolidin-1-yl]-7H-purineIC501600.0 [1]
4-[[(2R)-1-(7H-Purin-6-yl)pyrrolidin-2-yl]methoxy]benzonitrileIC501300.0 [1]
6-[(2R)-2-[(4-Fluorophenoxy)methyl]pyrrolidin-1-yl]-7H-purineIC503800.0 [1]
6-[(2R)-2-[(2-Methylphenoxy)methyl]pyrrolidin-1-yl]-7H-purineIC50700.0 [1]
6-[(2R)-2-[(2-Chlorophenoxy)methyl]pyrrolidin-1-yl]-7H-purineIC501000.0 [1]
6-(Trifluoromethyl)-1H-IndazoleIC5050.12 [1]
6-Bromo-1H-indazol-3-olIC502800.0 [1]
5-Chloro-N,6-dimethyl-2-pyridin-2-ylpyrimidin-4-amineIC5014000.0 [1]
1,2-Benzisoselenazol-3(2H)-one, 2-(4-methylphenyl)-IC5024300.0 [1]
1,2-Benzisoselenazol-3(2H)-one, 2-(4-fluorophenyl)-IC5010900.0 [1]
1,2-Benzisoselenazol-3(2H)-one, 2-(4-methoxyphenyl)-IC502070.0 [1]
1,2-Benzisoselenazol-3(2H)-one, 2-(2-hydroxyphenyl)-IC5010200.0 [1]
7-[(2R)-2-[(2-Chlorophenoxy)methyl]pyrrolidin-1-yl]-1H-imidazo[4,5-b]pyridineIC502200.0 [1]
4-[(2R)-2-[(2-Chlorophenoxy)methyl]pyrrolidin-1-yl]-1H-pyrazolo[3,4-d]pyrimidineIC508600.0 [1]
6-[(2R)-2-(Naphthalen-1-yloxymethyl)pyrrolidin-1-yl]-7H-purineIC50450.0 [1]
7-[(2R)-2-[(2-Chlorophenoxy)methyl]pyrrolidin-1-yl]-[1,2,5]thiadiazolo[3,4-b]pyridineIC502800.0 [1]
4-[(2R)-2-[(2-Chlorophenoxy)methyl]pyrrolidin-1-yl]pyrido[2,3-d]pyrimidineIC5050000.0 [1]
5-[[(2R)-1-(7H-Purin-6-yl)pyrrolidin-2-yl]methoxy]isoquinolineIC50230.0 [1]
7-[(2R)-2-(Naphthalen-1-yloxymethyl)pyrrolidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidineIC50110.0 [1]
5-[(2R)-2-(Naphthalen-1-yloxymethyl)pyrrolidin-1-yl]imidazo[1,2-a]pyrimidineIC50560.0 [1]
5,6-Dimethyl-N-(2-phenylethyl)-2-pyridin-2-ylpyrimidin-4-amineIC50100000.0 [1]
5-Chloro-4-methyl-6-(2-phenylethylsulfanyl)-2-pyridin-2-ylpyrimidineIC50100000.0 [1]
7-[(2R)-2-(Naphthalen-1-yloxymethyl)pyrrolidin-1-yl]-[1,2,4]triazolo[1,5-a][1,3,5]triazineIC501800.0 [1]
6-[(2S)-2-[(2-Chlorophenoxy)methyl]pyrrolidin-1-yl]-7H-purineIC5050000.0 [1]
N-[(1R)-2-[(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]-1-phenylethyl]-3-piperazin-1-ylpropanamideIC5022000.0 [1]
N-[(1R)-2-[(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]-1-phenylethyl]-3-[4-(2-hydroxyethyl)piperazin-1-yl]propanamideIC50114000.0 [1]
N-[(1R)-2-[(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]-1-phenylethyl]-4-piperazin-1-ylbutanamideIC50300000.0 [1]
(1R)-N'-(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-1-phenyl-N-(4-piperazin-1-ylbutyl)ethane-1,2-diamineIC50188000.0 [1]
N-[(1R)-2-[(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]-1-phenylethyl]-2-piperazin-1-ylethanesulfonamideIC509400.0 [1]
5-Fluoro-6-methyl-N-(2-phenylethyl)-2-pyridin-2-ylpyrimidin-4-amineIC5062000.0 [1]
(1R)-N'-(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)-1-phenyl-N-(3-piperazin-1-ylpropyl)ethane-1,2-diamineIC50108000.0 [1]
2-[4-[4-[[(1R)-2-[(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]-1-phenylethyl]amino]butyl]piperazin-1-yl]ethanolIC50197000.0 [1]
N-[(1R)-2-[(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]-1-phenylethyl]-2-[4-(2-hydroxyethyl)piperazin-1-yl]ethanesulfonamideIC5095000.0 [1]
2-[4-[3-[[(1R)-2-[(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]-1-phenylethyl]amino]propyl]piperazin-1-yl]ethanolIC50101000.0 [1]
N-[(1R)-2-[(5-Chloro-6-methyl-2-pyridin-2-ylpyrimidin-4-yl)amino]-1-phenylethyl]-4-[4-(2-hydroxyethyl)piperazin-1-yl]butanamideIC50300000.0 [1]
7-[[2-[(Z)-3-(Diethylamino)prop-1-enyl]-4-fluorophenyl]sulfonylamino]-4H-pyrrolo[2,1-c][1,4]benzoxazine-6-carboxylic acidIC5050.0 [1]
CID 71735205IC5020.0 [1]
4-(3-Methylpyridin-4-yl)-6-(trifluoromethyl)-1H-indazoleIC5011.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Microtubule-associated protein 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/microtubule-associated-protein-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Microtubule-associated protein 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/microtubule-associated-protein-2-inhibitors-ic50-ki.
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