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Mineralocorticoid receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
DexamethasoneIC5033.0 [1]
DexamethasoneKi0.36 [1], 7.2 [2]
MifepristoneIC501000.0 [1], 1155.0 [2], 6000.0 [3]
MifepristoneKi640.0 [1], 851.0 [2], 10000.0 [3]
EplerenoneIC50135.0 [1], 240.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMineralocorticoid receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.14 Jan2026https://www.aatbio.com/data-sets/mineralocorticoid-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026January 14). Quest DatabaseMineralocorticoid receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/mineralocorticoid-receptor-inhibitors-ic50-ki.
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