Name: Mitogen-activated protein kinase kinase kinase 12 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Mitogen-activated protein kinase kinase kinase 12 Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	Dlk-IN-1	IC50	129.0 ^[1], 195.0 ^[2]
	Dlk-IN-1	Ki	1.9 ^[1], 3.0 ^[2]
	5-[1-(Cyclopropylmethyl)-5-[(1R,5S)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine	IC50	144.0 ^[1]
	5-[1-(Cyclopropylmethyl)-5-[(1R,5S)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine	Ki	0.17 ^[1], 4.0 ^[2]
	5-[5-[(1S,5R)-3-(Oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(2,2,2-trifluoroethyl)pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amine	IC50	180.0 ^[1]
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References

This online resource may be cited as follows

MLA	"Quest Database™ Mitogen-activated protein kinase kinase kinase 12 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 Dec. 2025, https://www.aatbio.com/data-sets/mitogen-activated-protein-kinase-kinase-kinase-12-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, December 10). Quest Database™ Mitogen-activated protein kinase kinase kinase 12 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/mitogen-activated-protein-kinase-kinase-kinase-12-inhibitors-ic50-ki.
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