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Mitogen-activated protein kinase kinase kinase 5 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
StaurosporineIC500.69 [1], 37.0 [2], 1000.0 [3]
SelonsertibIC505.0 [1], 5.01 [2], 6.0 [3]
HymenialdisineIC50150.0 [1], 7000.0 [2]
Ethyl 8,15-dioxo-14-azatetracyclo[7.7.1.02,7.013,17]heptadeca-1(16),2,4,6,9(17),10,12-heptaene-16-carboxylateIC503000.0 [1]
Ethyl 8,15-dioxo-14-azatetracyclo[7.7.1.02,7.013,17]heptadeca-1(16),2,4,6,9(17),10,12-heptaene-16-carboxylateKi500.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMitogen-activated protein kinase kinase kinase 5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.21 Jan2026https://www.aatbio.com/data-sets/mitogen-activated-protein-kinase-kinase-kinase-5-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026January 21). Quest DatabaseMitogen-activated protein kinase kinase kinase 5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/mitogen-activated-protein-kinase-kinase-kinase-5-inhibitors-ic50-ki.
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