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Motilin receptor Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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(6R,9R,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneIC5074.0 [1]
(6R,9R,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi137.0 [1]
ErythromycinIC5043.65 [1], 70.79 [2]
ErythromycinKi37000.0 [1]
Erythromycin A enol etherIC503.39 [1], 223.87 [2]
(2S)-5-Amino-2-[[2-[[(2S)-6-amino-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-5-amino-2-[[(2R)-2-[[(2S)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S)-2-[[2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-amino-3-phenylpropanoyl]amino]-3-methylbutanoyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-3-hydroxybutanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]-4-carboxybutanoyl]amino]-4-methylpentanoyl]amino]-5-oxopentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-4-methylsulfanylbutanoyl]amino]-5-oxopentanoyl]amino]-4-carboxybutanoyl]amino]hexanoyl]amino]-4-carboxybutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-4-oxobutanoyl]amino]hexanoyl]amino]acetyl]amino]-5-oxopentanoic acidKi0.36 [1], 3.1 [2]
(6R,9R,12S,16E)-12-(4-Aminobutyl)-6-[(4-hydroxyphenyl)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi664.0 [1]
2-[(6R,9R,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-7,10,13-trioxo-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraen-12-yl]acetic acidKi2553.0 [1]
(6R,9R,12S)-6-[(4-Methoxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneIC5023.0 [1]
(6R,9R,12S)-6-[(4-Methoxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi8.0 [1]
(6R,9R,12S)-9-Propan-2-yl-12-(pyrrolidin-1-ylmethyl)-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneIC502.0 [1]
(6R,9R,12S)-9-Propan-2-yl-12-(pyrrolidin-1-ylmethyl)-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi4.6 [1]
(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-9-propan-2-yl-12-(pyrazol-1-ylmethyl)-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneIC5056.0 [1]
(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-9-propan-2-yl-12-(pyrazol-1-ylmethyl)-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi18.0 [1]
(6R,9R,12S)-12-(Aminomethyl)-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneIC508.0 [1]
(6R,9R,12S)-12-(Aminomethyl)-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi15.0 [1]
(6R,9R,12S)-6-[(4-Chlorophenyl)methyl]-12-(methylaminomethyl)-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneIC5033.0 [1]
(6R,9R,12S)-6-[(4-Chlorophenyl)methyl]-12-(methylaminomethyl)-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi31.0 [1]
(6R,9R,12S)-12-(Methylaminomethyl)-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneIC503.0 [1]
(6R,9R,12S)-12-(Methylaminomethyl)-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi6.0 [1]
(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-12-[(dimethylamino)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneIC5095.0 [1]
(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-12-[(dimethylamino)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi27.0 [1]
2-[[(6R,9R,12S)-7,10,13-Trioxo-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-trien-12-yl]methyl]guanidineIC5028.0 [1]
2-[[(6R,9R,12S)-7,10,13-Trioxo-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-trien-12-yl]methyl]guanidineKi6.0 [1]
(2R,3R,4R,11R,12S)-11-[(3R)-4-(Dimethylamino)-3-hydroxy-6-methyloxan-2-yl]oxy-5-ethyl-3-hydroxy-9-[(2R,4R,5S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-2,4,8,10,12,14-hexamethyl-6,15,16-trioxatricyclo[10.2.1.11,4]hexadecan-7-oneIC50154.88 [1], 169.82 [2]
(2R,3R,4S,11R,12S)-5-Ethyl-11-[(3R)-4-[ethyl(methyl)amino]-3-hydroxy-6-methyloxan-2-yl]oxy-3-hydroxy-9-[(2R,4R,5S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-4-methoxy-2,4,8,10,12,14-hexamethyl-6,15-dioxabicyclo[10.2.1]pentadec-1(14)-en-7-oneIC504.68 [1], 8.32 [2]
(2R,3R,4S,11R,12S)-5-Ethyl-3-hydroxy-9-[(2R,4R,5S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-11-[(3R)-3-hydroxy-6-methyl-4-[methyl(propan-2-yl)amino]oxan-2-yl]oxy-4-methoxy-2,4,8,10,12,14-hexamethyl-6,15-dioxabicyclo[10.2.1]pentadec-1(14)-en-7-oneIC506.92 [1], 15.14 [2]
(2R,3R,4S,11R,12S)-5-Ethyl-11-[(3R)-4-[ethyl(methyl)amino]-3-hydroxy-6-methyloxan-2-yl]oxy-3,4-dihydroxy-9-[(4R,5S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-2,4,8,12,14-pentamethyl-6,15-dioxabicyclo[10.2.1]pentadec-1(14)-en-7-oneIC503.16 [1], 302.0 [2]
(2R,3R,4S,11R,12S)-11-[(3R)-4-(Dimethylamino)-3-hydroxy-6-methyloxan-2-yl]oxy-5-ethyl-3-hydroxy-9-[(2R,4R,5S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-4-methoxy-2,4,8,10,12,14-hexamethyl-6,15-dioxabicyclo[10.2.1]pentadec-1(14)-en-7-oneIC507.59 [1], 39.81 [2]
CipargaminIC5010000.0 [1]
(2S,4R,5R,8R,9S,10S,11R,12S)-5-Ethyl-9-[(2R,4R,5S,6S)-5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl]oxy-11-[(2S,3R,4S,6R)-3-hydroxy-6-methyl-4-[methyl(propan-2-yl)amino]oxan-2-yl]oxy-4-methoxy-2,4,8,10,12,14-hexamethyl-6,15-dioxabicyclo[10.2.1]pentadec-1(14)-ene-3,7-dioneIC503.98 [1]
(2R,3S,4R,5R,8R,9S,10S,11R,12R)-5-Ethyl-11-[(2S,3R,4S,6R)-4-[ethyl(methyl)amino]-3-hydroxy-6-methyloxan-2-yl]oxy-3-hydroxy-9-[(2S,4S,6R)-4-methoxy-4,6-dimethyloxan-2-yl]oxy-2,4,8,10,12,14-hexamethyl-6,15-dioxabicyclo[10.2.1]pentadec-1(14)-en-7-oneKi3.4 [1]
[3-[4-[[(3S,5R)-3,5-Dimethylpiperazin-1-yl]methyl]phenyl]pyridin-2-yl]-[4-(4-fluoroanilino)piperidin-1-yl]methanoneIC503.98 [1]
N-[(2S)-1-[[(2S)-1-Amino-1-oxo-4-phenylbutan-2-yl]amino]-1-oxo-4-phenylbutan-2-yl]-2-(1,3-benzodioxol-5-ylmethyl)-1,3-dioxospiro[7,8-dihydro-6H-[1,2,4]triazolo[1,2-a]pyridazine-5,4'-piperidine]-8-carboxamideKi0.7 [1]
(6R,9R,12S)-12-(Aminomethyl)-6-[(4-chlorophenyl)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi60.0 [1]
(6R,9R,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-12-(2-methylpropyl)-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi62.0 [1]
N-[(2S)-1-[[(2S)-1-Amino-1-oxo-4-phenylbutan-2-yl]amino]-1-oxo-4-phenylbutan-2-yl]-2-(1,3-benzodioxol-5-ylmethyl)-1,3-dioxospiro[8H-[1,2,4]triazolo[1,2-a]pyridazine-5,4'-piperidine]-8-carboxamideKi2.0 [1]
(6R,9R,12S)-6-(1H-Indol-3-ylmethyl)-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi255.0 [1]
(6R,9R,12S,16E)-6-Benzyl-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi78.0 [1]
2-[[(6R,9R,12S)-6-[(4-Chlorophenyl)methyl]-7,10,13-trioxo-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-trien-12-yl]methyl]guanidineKi6.0 [1]
N-[(2R)-1-Amino-1-oxo-4-phenylbutan-2-yl]-2-(1,3-benzodioxol-5-ylmethyl)-1,3-dioxospiro[8H-[1,2,4]triazolo[1,2-a]pyridazine-5,4'-piperidine]-8-carboxamideKi10000.0 [1]
(6R,9R,12S)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi55.0 [1]
(6R,9R,12S)-6-[(4-Hydroxyphenyl)methyl]-11-methyl-12-(2-methylpropyl)-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi222.0 [1]
(6R,9R,12S)-12-(Aminomethyl)-6-[(3-chlorophenyl)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi64.0 [1]
N-[(2S)-1-Amino-1-oxo-4-phenylbutan-2-yl]-2-(1,3-benzodioxol-5-ylmethyl)-1,3-dioxospiro[8H-[1,2,4]triazolo[1,2-a]pyridazine-5,4'-piperidine]-8-carboxamideKi10000.0 [1]
(6R,9R,12S)-6-[(4-Chlorophenyl)methyl]-12-[(dimethylamino)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi16.0 [1]
(6R,9R,12S)-6-(Naphthalen-1-ylmethyl)-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi8.3 [1]
(6R,9R,12S)-6-(1-Benzothiophen-3-ylmethyl)-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi11.0 [1]
(6R,9R,12S,16E)-6-Methyl-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi10000.0 [1]
(6R,9R,12S,16E)-6,9-Di(propan-2-yl)-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi3566.0 [1]
(6R,9R,12S,16E)-6-(4-Aminobutyl)-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi10000.0 [1]
(6R,9S,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi10000.0 [1]
(6R,9R,12S,16E)-9-(Hydroxymethyl)-6-[(4-hydroxyphenyl)methyl]-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi10000.0 [1]
(6R,9R,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-12-methyl-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi1389.0 [1]
(6R,9R,12R,16E)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi335.0 [1]
(6R,9R,12S,16E)-12-Benzyl-6-[(4-hydroxyphenyl)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi185.0 [1]
(2E,7S,10R,13R)-13-[(4-Hydroxyphenyl)methyl]-10-propan-2-yl-7-propyl-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),2,18,20-tetraene-6,9,12-trioneKi10000.0 [1]
(6S,9R,12R)-12-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-6-propyl-4,7,10,13-tetrazabicyclo[15.4.0]henicosa-1(21),17,19-triene-5,8,11-trioneKi10000.0 [1]
(5R,8R,11S)-5-[(4-Hydroxyphenyl)methyl]-8-propan-2-yl-11-propyl-4,7,10,13-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-6,9,12-trioneKi6064.0 [1]
(5R,8R,11S)-5-[(4-Hydroxyphenyl)methyl]-8-propan-2-yl-11-propyl-4,7,10,13-tetrazabicyclo[15.4.0]henicosa-1(21),17,19-triene-6,9,12-trioneKi10000.0 [1]
(6S,9R,12R)-12-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-6-propyl-4,7,10,13-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-5,8,11-trioneKi6064.0 [1]
(3S,6R,9R,12E)-9-[(4-Hydroxyphenyl)methyl]-6-propan-2-yl-3-propyl-1,4,7,10-tetrazacyclopentadec-12-ene-2,5,8-trioneKi701.0 [1]
(6R,9R,12S)-6-Benzyl-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi57.0 [1]
(6R,9R,12S)-6-Phenyl-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi10000.0 [1]
(6R,9R,12S)-6-(Naphthalen-2-ylmethyl)-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi79.0 [1]
(6R,9R,12S)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2,8-dioxa-5,11,14-triazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi192.0 [1]
(6R,9R,12S)-6-[(4-Hydroxyphenyl)methyl]-8-methyl-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi10000.0 [1]
(6R,9R,12S)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-10,13-dioneKi3237.0 [1]
(6R,10R,13S)-6-[(4-Hydroxyphenyl)methyl]-10-propan-2-yl-13-propyl-2-oxa-5,8,9,12,15-pentazabicyclo[17.4.0]tricosa-1(23),19,21-triene-7,11,14-trioneKi2373.0 [1]
(6S,9R,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi10000.0 [1]
3-[(6R,9R,12S,16E)-7,10,13-Trioxo-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraen-6-yl]propanoic acidKi10000.0 [1]
(6R,9R,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-9-methyl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi196.0 [1]
3-[(6R,9R,12S,16E)-6-[(4-Hydroxyphenyl)methyl]-7,10,13-trioxo-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraen-9-yl]propanoic acidKi4898.0 [1]
(6R,9R,12S,16E)-9-Benzyl-6-[(4-hydroxyphenyl)methyl]-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi1524.0 [1]
(6R,9R,12S,16E)-12-(Hydroxymethyl)-6-[(4-hydroxyphenyl)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trioneKi650.0 [1]
(7S,10R,13R)-13-[(4-Hydroxyphenyl)methyl]-10-propan-2-yl-7-propyl-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-6,9,12-trioneKi10000.0 [1]
(5R,8R,11S,15E)-5-[(4-Hydroxyphenyl)methyl]-8-propan-2-yl-11-propyl-4,7,10,13-tetrazabicyclo[15.4.0]henicosa-1(21),15,17,19-tetraene-6,9,12-trioneKi9726.0 [1]
(4R,7R,10S)-4-[(4-Hydroxyphenyl)methyl]-7-propan-2-yl-10-propyl-3,6,9,12-tetrazabicyclo[15.4.0]henicosa-1(21),17,19-triene-5,8,11-trioneKi10000.0 [1]
(6R,9R,12S)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[15.4.0]henicosa-1(21),17,19-triene-7,10,13-trioneKi982.0 [1]
(3S,6R,9R)-9-[(4-Hydroxyphenyl)methyl]-6-propan-2-yl-3-propyl-1,4,7,10-tetrazacyclooctadecane-2,5,8-trioneKi1197.0 [1]
(6R,9R,12S)-6-(Cyclohexylmethyl)-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi3247.0 [1]
(6R,9R,12S)-6-(2-Phenylethyl)-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi1486.0 [1]
(6R,9R,12S)-6-[(4-Hydroxyphenyl)methyl]-9-propan-2-yl-12-propyl-2,11-dioxa-5,8,14-triazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi1876.0 [1]
(6R,9R,12S)-6-[(4-Hydroxyphenyl)methyl]-5-methyl-9-propan-2-yl-12-propyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi2777.0 [1]
N-[[(1R,3S)-3-[Benzyl(2,2-dimethylpropanoyl)amino]cyclohexyl]methyl]-4-fluoro-N-[3-(2-pyrrolidin-1-ylethoxy)phenyl]benzamideIC502480.0 [1]
N-[[3-[(3-Chlorophenyl)methyl-(2,2,2-trichloroacetyl)amino]cyclohexyl]methyl]-4-fluoro-N-[3-(2-piperidin-1-ylethoxy)phenyl]benzamideIC50228.0 [1]
N-[[3-[Benzyl(2,2-dimethylpropanoyl)amino]cyclohexyl]methyl]-4-fluoro-N-[3-(2-pyrrolidin-1-ylethoxy)phenyl]benzamideIC50990.0 [1]
2-[2-[(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-7,10,13-trioxo-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-trien-12-yl]ethyl]guanidineKi33.0 [1]
(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-12-(imidazol-1-ylmethyl)-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi62.0 [1]
3-[(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-7,10,13-trioxo-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-trien-12-yl]propanimidamideKi27.0 [1]
(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-12-[(4,5-dihydro-1H-imidazol-2-ylamino)methyl]-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi51.0 [1]
(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-9-propan-2-yl-12-[(1,4,5,6-tetrahydropyrimidin-2-ylamino)methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi87.0 [1]
2-[[(6R,9R,12S)-6-[(3-Chlorophenyl)methyl]-7,10,13-trioxo-9-propan-2-yl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-trien-12-yl]methyl]-1-cyanoguanidineKi100.0 [1]
(6R,9R,12S)-9-Propan-2-yl-12-[(pyrimidin-2-ylamino)methyl]-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi20.0 [1]
(6R,9R,12S)-12-[(5-Methyltriazol-1-yl)methyl]-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi17.0 [1]
(6R,9R,12S)-12-[(5-Methyltetrazol-1-yl)methyl]-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi21.0 [1]
(6R,9R,12S)-12-[(4,5-Dimethyltriazol-1-yl)methyl]-9-propan-2-yl-6-[[3-(trifluoromethyl)phenyl]methyl]-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),18,20-triene-7,10,13-trioneKi23.0 [1]
Methyl (2R)-2-[[2-(1,3-benzodioxol-5-ylmethyl)-1,3-dioxospiro[8H-[1,2,4]triazolo[1,2-a]pyridazine-5,4'-piperidine]-8-carbonyl]amino]-4-phenylbutanoateKi10000.0 [1]
N-[(2R)-1-[[(2R)-1-Amino-1-oxo-4-phenylbutan-2-yl]amino]-1-oxo-4-phenylbutan-2-yl]-2-(1,3-benzodioxol-5-ylmethyl)-1,3-dioxospiro[7,8-dihydro-6H-[1,2,4]triazolo[1,2-a]pyridazine-5,4'-piperidine]-8-carboxamideKi2.7 [1]
N-[[3-[(3-Chlorophenyl)methyl-(2,2,2-trichloroacetyl)amino]cyclohexyl]methyl]-4-fluoro-N-[3-(2-pyrrolidin-1-ylethoxy)phenyl]benzamideIC50267.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Motilin receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/motilin-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Motilin receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/motilin-receptor-inhibitors-ic50-ki.
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