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Mu opioid receptor Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
NaltrexoneIC508.9 [1]
NaltrexoneKi0.2 [1], 0.7 [2], 3.6 [3]
DamgoIC501.5 [1], 2.5 [2], 3.18 [3], 5.0 [4]
DamgoKi36.7 [1]
MorphineIC500.57 [1], 2.5 [2], 4.3 [3], 6.3 [4]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMu opioid receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/mu-opioid-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseMu opioid receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/mu-opioid-receptor-inhibitors-ic50-ki.
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