Multidrug and toxin extrusion protein 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Ondansetron	IC50	10.0 [1], 30.0 [2], 150.0 [3], 160.0 [4]
	Imatinib	IC50	40.0 [1], 50.0 [2], 350.0 [3]
	Irinotecan	IC50	2100.0 [1], 4300.0 [2], 7900.0 [3]
	Ritonavir	IC50	80.0 [1], 2100.0 [2], 4400.0 [3]
	Mitoxantrone	IC50	190.0 [1], 400.0 [2], 530.0 [3]
	Indinavir	IC50	1700.0 [1], 1900.0 [2], 7800.0 [3]
	Pantoprazole	IC50	2800.0 [1], 43200.0 [2]
	Pentamidine	IC50	410.0 [1], 2000.0 [2], 2700.0 [3]
	Nifekalant	IC50	650.0 [1], 1100.0 [2], 6500.0 [3]
	Cimetidine	IC50	1200.0 [1], 5700.0 [2]
	Dexamethasone	IC50	500000.0 [1]
	Indomethacin	IC50	500000.0 [1]
	Lidocaine	IC50	500000.0 [1]
	Metformin	IC50	250000.0 [1]
	Clonidine	IC50	33300.0 [1]
	Furosemide	IC50	500000.0 [1]
	Nicotinic acid	IC50	500000.0 [1]
	Erythromycin	IC50	500000.0 [1]
	Diclofenac	IC50	500000.0 [1]
	Risperidone	IC50	1600.0 [1]
	Losartan	IC50	250000.0 [1]
	Ethinyl estradiol	IC50	21100.0 [1]
	Spironolactone	IC50	18600.0 [1]
	Imipramine	IC50	10000.0 [1]
	Dipyridamole	IC50	26000.0 [1]
	Prazosin	IC50	1600.0 [1]
	Azacitidine	IC50	500000.0 [1]
	Enalapril	IC50	500000.0 [1]
	Chlorhexidine	IC50	700.0 [1]
	Quinidine	IC50	11200.0 [1]
	Levofloxacin	IC50	17900.0 [1]
	Ranitidine Base	IC50	8300.0 [1]
	Tubocurarine	IC50	9400.0 [1]
	Carvedilol	IC50	92400.0 [1]
	Aripiprazole	IC50	130000.0 [1]
	Topotecan	IC50	1300.0 [1]
	Amantadine	IC50	37800.0 [1]
	Sumatriptan	IC50	6700.0 [1]
	Dabigatran	IC50	8100.0 [1]
	Vecuronium	IC50	1900.0 [1]
	Telmisartan	IC50	17900.0 [1]
	Buspirone	IC50	1700.0 [1]
	Phenacetin	IC50	500000.0 [1]
	Irbesartan	IC50	500000.0 [1]
	Domperidone	IC50	2300.0 [1]
	Thiabendazole	IC50	500000.0 [1]
	Cetirizine	IC50	500000.0 [1]
	Pimozide	IC50	500000.0 [1]
	Tacrine	IC50	1100.0 [1]
	Dihydroergotamine	IC50	2800.0 [1]
	Disopyramide	IC50	66000.0 [1]
	Pepcid	IC50	760.0 [1]
	Maraviroc	IC50	17300.0 [1]
	Granisetron	IC50	5000.0 [1]
	Astemizole	IC50	26400.0 [1]
	Zafirlukast	IC50	1300.0 [1]
	Gabexate	IC50	500.0 [1]
	Ciclopirox	IC50	500000.0 [1]
	Methylergonovine	IC50	250000.0 [1]
	Orphenadrine	IC50	65000.0 [1]
	Rimantadine	IC50	7300.0 [1]
	Noscapine	IC50	34500.0 [1]
	Sulfacetamide	IC50	500000.0 [1]
	Camostat	IC50	2900.0 [1]
	Epinastine	IC50	1100.0 [1]
	Bithionol	IC50	5200.0 [1]
	(3R,8S,9S,10R,13S,14S,17R)-3,17-Dihydroxy-17-(2-hydroxyacetyl)-10,13-dimethyl-2,3,6,7,8,9,12,14,15,16-decahydro-1H-cyclopenta[a]phenanthren-11-one	IC50	21400.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 67 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Multidrug and toxin extrusion protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/multidrug-and-toxin-extrusion-protein-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Multidrug and toxin extrusion protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/multidrug-and-toxin-extrusion-protein-1-inhibitors-ic50-ki.
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