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Multidrug and toxin extrusion protein 2 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
OndansetronIC50160.0 [1], 300.0 [2], 6900.0 [3]
ImatinibIC50350.0 [1], 2900.0 [2]
IrinotecanIC507900.0 [1], 78600.0 [2]
RitonavirIC504400.0 [1], 23700.0 [2]
MitoxantroneIC50530.0 [1], 830.0 [2]
IndinavirIC507800.0 [1], 500000.0 [2]
PantoprazoleIC5043200.0 [1], 500000.0 [2]
PentamidineIC502700.0 [1], 10400.0 [2]
NifekalantIC502700.0 [1], 6500.0 [2]
RisperidoneIC50291000.0 [1]
Ethinyl estradiolIC5020200.0 [1]
ImipramineIC50100000.0 [1]
DipyridamoleIC5074000.0 [1]
PrazosinIC5038400.0 [1]
CimetidineIC5039000.0 [1]
ChlorhexidineIC50500.0 [1]
TubocurarineIC5055500.0 [1]
AripiprazoleIC50500000.0 [1]
TopotecanIC508600.0 [1]
DabigatranIC5025300.0 [1]
VecuroniumIC5025200.0 [1]
BuspironeIC5046000.0 [1]
DomperidoneIC5014800.0 [1]
PimozideIC50500000.0 [1]
TacrineIC50100000.0 [1]
DihydroergotamineIC5012600.0 [1]
DisopyramideIC50100000.0 [1]
PepcidIC5036200.0 [1]
MaravirocIC50297000.0 [1]
GranisetronIC50311000.0 [1]
ZafirlukastIC507600.0 [1]
GabexateIC5010800.0 [1]
OrphenadrineIC50100000.0 [1]
RimantadineIC50288000.0 [1]
CamostatIC5012700.0 [1]
EpinastineIC5029800.0 [1]
BithionolIC506600.0 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Multidrug and toxin extrusion protein 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.9 May2024https://www.aatbio.com/data-sets/multidrug-and-toxin-extrusion-protein-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 9). Quest Database™ Multidrug and toxin extrusion protein 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/multidrug-and-toxin-extrusion-protein-2-inhibitors-ic50-ki.
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