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Multidrug resistance-associated protein 1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
VerlukastIC50400.0 [1], 3300.0 [2], 5220.0 [3]
VerlukastKi600.0 [1], 134700.0 [2], 139600.0 [3]
Cyclosporin AIC502700.0 [1], 2810.0 [2], 2970.0 [3], 3530.0 [4], 4780.0 [5]
Cyclosporin AKi5000.0 [1]
VerapamilIC503500.0 [1], 6800.0 [2], 9660.0 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMultidrug resistance-associated protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.2 Feb2026https://www.aatbio.com/data-sets/multidrug-resistance-associated-protein-1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026February 2). Quest DatabaseMultidrug resistance-associated protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/multidrug-resistance-associated-protein-1-inhibitors-ic50-ki.
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