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Muscarinic acetylcholine receptor M1 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
PirenzepineIC5019.0 [1]
PirenzepineKi15.0 [1], 23.5 [2]
CarbacholIC504090.0 [1], 10000.0 [2], 124830.0 [3], 150000.0 [4]
CarbacholKi170.0 [1], 3162.28 [2], 501187233627.27 [3]
XanomelineIC500.01 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMuscarinic acetylcholine receptor M1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.6 Dec2025https://www.aatbio.com/data-sets/muscarinic-acetylcholine-receptor-m1-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 6). Quest DatabaseMuscarinic acetylcholine receptor M1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/muscarinic-acetylcholine-receptor-m1-inhibitors-ic50-ki.
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