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Muscarinic acetylcholine receptor M4 Inhibitors (IC50, Ki)
StructureCompound NameStandard TypeStandard Values (in nM)
CarbacholIC500.4 [1], 50.12 [2], 1000.0 [3], 7200.0 [4]
CarbacholKi24.0 [1], 398.11 [2], 2600.0 [3]
4-Damp methiodideIC501.9 [1]
4-Damp methiodideKi0.51 [1], 0.88 [2]
PirenzepineIC501.15 [1], 246.8 [2], 1047.13 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseMuscarinic acetylcholine receptor M4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Oct2025https://www.aatbio.com/data-sets/muscarinic-acetylcholine-receptor-m4-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025October 15). Quest DatabaseMuscarinic acetylcholine receptor M4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/muscarinic-acetylcholine-receptor-m4-inhibitors-ic50-ki.
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