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Myotonin-protein kinase Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
Y-27632 DihydrochlorideIC508000.0 [1]
FasudilIC508000.0 [1]
N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(dimethylamino)-2-phenylacetamideIC508000.0 [1]
N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(cyclopropylamino)-2-phenylacetamideIC508000.0 [1]
N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-(methylamino)-2-phenylacetamideIC508000.0 [1]
2-Amino-N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamideIC508000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
TilfrinibIC5010000.0 [1]
5-[1-(Cyclopropylmethyl)-5-[(1R,5S)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]pyrazol-3-yl]-3-(trifluoromethyl)pyridin-2-amineIC501380.0 [1]
6-[4-[(5-Tert-butyl-1,2-oxazol-3-yl)carbamoylamino]phenyl]-N-[3-(dimethylamino)propyl]imidazo[2,1-b][1,3]thiazole-3-carboxamideIC5010000.0 [1]
2-Amino-7-methyl-4-[(4-methylphenyl)methylamino]-9H-pyrimido[4,5-b]indol-6-olIC50100000.0 [1]
2-[2,6-Bis[5-[5-(1,3-oxazol-5-yl)pyridin-2-yl]-1,3-oxazol-2-yl]pyridin-4-yl]oxy-N,N-dimethylethanamineIC501000.0 [1]
5-[6-(1,3-Oxazol-5-yl)pyridin-2-yl]-2-[6-[6-[5-[6-(1,3-oxazol-5-yl)pyridin-2-yl]-1,3-oxazol-2-yl]pyridin-2-yl]pyridin-2-yl]-1,3-oxazoleIC501000.0 [1]
5-[5-(1,3-Oxazol-5-yl)pyridin-2-yl]-2-[6-[5-[5-(1,3-oxazol-5-yl)pyridin-2-yl]-1,3-oxazol-2-yl]pyridin-2-yl]-1,3-oxazoleIC501000.0 [1]
N-(7-Chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)-2-phenylacetamideIC508000.0 [1]
2-(Benzylamino)-N-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)acetamideIC508000.0 [1]
1-[4-Chloro-3-(trifluoromethyl)phenyl]-3-[4-(1H-pyrazolo[3,4-d]pyrimidin-4-yloxy)phenyl]ureaIC5010000.0 [1]
1-[(3-Hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea;methanesulfonic acidIC5034.06 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Myotonin-protein kinase Inhibitors (IC50, Ki)." AAT Bioquest, Inc.10 May2024https://www.aatbio.com/data-sets/myotonin-protein-kinase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024May 10). Quest Database™ Myotonin-protein kinase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/myotonin-protein-kinase-inhibitors-ic50-ki.
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