N-type calcium channel alpha-1b/alpha2delta-1/beta-1b Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	1-[4-(Diphenylmethyl)-1-piperazinyl]-3,3-diphenyl-1-propanone	IC50	110.0 [1]
	N,4-Dibenzhydrylpiperazine-1-carboxamide	IC50	150.0 [1]
	1-(4-Benzhydrylpiperazin-1-yl)-2-(N-phenylanilino)ethanone	IC50	6610.0 [1]
	2-(4-(Diphenylmethyl)piperazinyl)-N,N-diphenylethanamide	IC50	260.0 [1]
	1-[4-[(2-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	90.0 [1]
	1-[4-[(2,6-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	210.0 [1]
	1-[4-[(2,4-Dimethylphenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	230.0 [1]
	1-[4-[(3-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	40.0 [1]
	3,3-Diphenyl-1-[4-[phenyl-[2-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]propan-1-one	IC50	300.0 [1]
	3,3-Diphenyl-1-[4-[phenyl-(3,4,5-trimethoxyphenyl)methyl]piperazin-1-yl]propan-1-one	IC50	510.0 [1]
	1-[4-[(3,4-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	1000.0 [1]
	1-[4-[(4-Fluorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	380.0 [1]
	1-{4-[(4-Chloro-phenyl)-phenyl-methyl]-piperazin-1-yl}-3,3-diphenyl-propan-1-one	IC50	110.0 [1]
	1-[4-[Bis(4-methoxyphenyl)methyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	240.0 [1]
	1-[4-[(2,3-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	220.0 [1]
	1-[4-[(4-Methylphenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	310.0 [1]
	1-[4-(1-Methyl-piperidin-4-ylmethyl)piperazin-1-yl]-3,3-diphenyl-propan-1-one	IC50	2400.0 [1]
	1-[4-[(3,5-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	170.0 [1]
	1-[4-[(4-Methoxyphenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	250.0 [1]
	1-[4-[(2,4-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	1000.0 [1]
	N-Benzhydryl-4-[(2,3-dichlorophenyl)-phenylmethyl]piperazine-1-carboxamide	IC50	200.0 [1]
	N-Benzhydryl-4-[(4-chlorophenyl)-phenylmethyl]piperazine-1-carboxamide	IC50	280.0 [1]
	1-[4-[(2,4-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-2-(N-phenylanilino)ethanone	IC50	460.0 [1]
	2-[4-[(2,4-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-N,N-diphenylacetamide	IC50	510.0 [1]
	2-[4-[(2,4-Dimethylphenyl)-phenylmethyl]piperazin-1-yl]-N,N-diphenylacetamide	IC50	1250.0 [1]
	2-[4-[(4-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-N,N-diphenylacetamide	IC50	110.0 [1]
	2-[4-[(3-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-N,N-diphenylacetamide	IC50	320.0 [1]
	2-[4-[(2,3-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-N,N-diphenylacetamide	IC50	240.0 [1]
	N-Benzhydryl-4-[(2,4-dimethylphenyl)-phenylmethyl]piperazine-1-carboxamide	IC50	2710.0 [1]
	1-[4-[(2,3-Dichlorophenyl)-phenylmethyl]piperazin-1-yl]-2-(N-phenylanilino)ethanone	IC50	140.0 [1]
	1-[4-[(2-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-2-(N-phenylanilino)ethanone	IC50	320.0 [1]
	2-[4-[(2-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-N,N-diphenylacetamide	IC50	50.0 [1]
	N-Benzhydryl-4-[(2-chlorophenyl)-phenylmethyl]piperazine-1-carboxamide	IC50	180.0 [1]
	1-{4-[(4-Chloro-phenyl)-phenyl-methyl]-piperazin-1-yl}-2-diphenylaminoethanone	IC50	500.0 [1]
	1-[4-[(3-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-2-(N-phenylanilino)ethanone	IC50	280.0 [1]
	N-Benzhydryl-4-[(2,4-dichlorophenyl)-phenylmethyl]piperazine-1-carboxamide	IC50	1480.0 [1]
	N-Benzhydryl-4-[(3-chlorophenyl)-phenylmethyl]piperazine-1-carboxamide	IC50	340.0 [1]
	1-[4-[(2,4-Dimethylphenyl)-phenylmethyl]piperazin-1-yl]-2-(N-phenylanilino)ethanone	IC50	260.0 [1]
	3,3-Diphenyl-1-[4-[phenyl-[4-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]propan-1-one	IC50	70.0 [1]
	1-[4-[(R)-(4-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	50.0 [1]
	1-[4-[(S)-(4-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	140.0 [1]
	3,3-Diphenyl-1-[4-[phenyl(piperidin-4-yl)methyl]piperazin-1-yl]propan-1-one	IC50	60.0 [1]
	1-[4-[(1-Methylpiperidin-4-yl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	690.0 [1]
	1-[4-[(1-Methylpiperidin-3-yl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	270.0 [1]
	1-[4-[(4-Chlorophenyl)-(1-methylpiperidin-4-yl)methyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	40.0 [1]
	1-[4-[(4-Fluorophenyl)-(1-methylpiperidin-4-yl)methyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	100.0 [1]
	3,3-Diphenyl-1-[4-(piperidin-4-ylmethyl)piperazin-1-yl]propan-1-one	IC50	2500.0 [1]
	3,3-Diphenyl-1-[4-(piperidin-2-ylmethyl)piperazin-1-yl]propan-1-one	IC50	2700.0 [1]
	1-[4-[(3,5-Dimethoxyphenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one	IC50	210.0 [1]
	3,3-Diphenyl-1-[4-[phenyl-[3-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]propan-1-one	IC50	110.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 50 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ N-type calcium channel alpha-1b/alpha2delta-1/beta-1b Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/n-type-calcium-channel-alpha-1b-alpha2delta-1-beta-1b-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ N-type calcium channel alpha-1b/alpha2delta-1/beta-1b Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/n-type-calcium-channel-alpha-1b-alpha2delta-1-beta-1b-inhibitors-ic50-ki.
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