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Nerve growth factor receptor Trk-A Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
StaurosporineIC500.5 [1], 1.29 [2], 1.7 [3], 3.1 [4], 8.3 [5]
N-(5-Cyclopropyl-2-phenylpyrazol-3-yl)-2-[4-[3-methoxy-4-(4-methylimidazol-1-yl)phenyl]triazol-1-yl]acetamideIC5047.0 [1], 85.4 [2], 119.3 [3], 287.2 [4], 662.0 [5]
Antibiotic K 252aIC502.4 [1], 13.0 [2]
Methyl (15S,16S,18R)-16-hydroxy-15-methyl-3-oxo-28-oxa-4,14,19-triazaoctacyclo[12.11.2.115,18.02,6.07,27.08,13.019,26.020,25]octacosa-1,6,8,10,12,20,22,24,26-nonaene-16-carboxylateIC501.2 [1], 5.0 [2]
AZ-23IC503.2 [1], 8.9 [2], 9.9 [3]

References
This online resource may be cited as follows
MLA
"Quest DatabaseNerve growth factor receptor Trk-A Inhibitors (IC50, Ki)." AAT Bioquest, Inc.8 Jun2026https://www.aatbio.com/data-sets/nerve-growth-factor-receptor-trk-a-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2026June 8). Quest DatabaseNerve growth factor receptor Trk-A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/nerve-growth-factor-receptor-trk-a-inhibitors-ic50-ki.
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