Name: Neuronal acetylcholine receptor; alpha2/beta2 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Neuronal acetylcholine receptor; alpha2/beta2 Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	Nicotine	Ki	5.5 ^[1], 12.0 ^[2]
	7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino(2,3-h)(3)benzazepine	Ki	0.48 ^[1]
	Sazetidine A	Ki	0.09 ^[1]
	2-Methyl-4-[5-((S)-1-methyl-pyrrolidin-2-ylmethoxy)-pyridin-3-yl]-but-3-yn-2-ol	Ki	61000.0 ^[1]
	(3S)-3-[[(2S)-1-[(2S)-4-Amino-2-[[(2S)-4-amino-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S)-1-[(2S)-1-[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2R)-2-[(2-aminoacetyl)amino]-3-sulfanylpropanoyl]amino]-3-sulfanylpropanoyl]amino]-3-hydroxypropanoyl]amino]-4-methylpentanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]amino]-3-sulfanylpropanoyl]amino]propanoyl]amino]propanoyl]amino]-4-oxobutanoyl]amino]-4-oxobutanoyl]pyrrolidine-2-carbonyl]amino]-4-[[(2S)-1-[[(2R)-1-amino-1-oxo-3-sulfanylpropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-4-oxobutanoic acid	IC50	9.6 ^[1]
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References

This online resource may be cited as follows

MLA	"Quest Database™ Neuronal acetylcholine receptor; alpha2/beta2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 Mar. 2026, https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-alpha2-beta2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2026, March 10). Quest Database™ Neuronal acetylcholine receptor; alpha2/beta2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-alpha2-beta2-inhibitors-ic50-ki.
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