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Neuronal acetylcholine receptor; alpha2/beta4 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
NicotineKi70.0 [1], 103.0 [2], 110.0 [3]
7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino(2,3-h)(3)benzazepineKi94.0 [1]
MecamylamineIC5016000.0 [1]
EpibatidineKi0.09 [1]
MethyllycaconitineIC501000.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabaseNeuronal acetylcholine receptor; alpha2/beta4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-alpha2-beta4-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabaseNeuronal acetylcholine receptor; alpha2/beta4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-alpha2-beta4-inhibitors-ic50-ki.
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