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Neuronal acetylcholine receptor; alpha3/beta4 Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
NicotineIC50430.0 [1], 1000.0 [2], 10000.0 [3]
NicotineKi530.0 [1]
CytisineKi840.0 [1]
BupropionIC501.8 [1], 1800.0 [2]
VareniclineIC50110.0 [1], 1000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseNeuronal acetylcholine receptor; alpha3/beta4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.13 Dec2025https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-alpha3-beta4-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 13). Quest DatabaseNeuronal acetylcholine receptor; alpha3/beta4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-alpha3-beta4-inhibitors-ic50-ki.
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