Neuronal acetylcholine receptor protein alpha-7 subunit Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Nicotine	IC50	7600.0 [1], 21000.0 [2]
	Nicotine	Ki	6300.0 [1]
	Methyllycaconitine	IC50	8.32 [1], 1000.0 [2]
	Methyllycaconitine	Ki	1.0 [1], 1.62 [2], 6.31 [3], 7.3 [4]
	Epibatidine	IC50	31.0 [1]
	Epibatidine	Ki	2.7 [1], 10.0 [2], 10.2 [3], 25.0 [4]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Dimethyl-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	1479.11 [1], 1513.56 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Dimethyl-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	199.53 [1], 316.23 [2], 331.13 [3]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Di(cyclohex-2-en-1-yl)-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	2951.21 [1], 3019.95 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Di(cyclohex-2-en-1-yl)-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	630.96 [1], 794.33 [2], 851.14 [3]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(4-nitrophenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	363.08 [1], 371.54 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(4-nitrophenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	18.2 [1], 19.95 [2], 31.62 [3]
	(2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Dimethyl-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	IC50	1380.38 [1], 2089.3 [2]
	(2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Dimethyl-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	Ki	630.96 [1], 977.24 [2], 1000.0 [3]
	(S)-3-(Azetidin-2-ylmethoxy)pyridine	Ki	148.0 [1]
	Trimethyl-[[20-[(trimethylazaniumyl)methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl]azanium;diiodide	IC50	100000.0 [1]
	Trimethyl-[[20-[(trimethylazaniumyl)methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl]azanium;diiodide	Ki	1258.93 [1], 2511.89 [2], 4466.84 [3]
	Cytisine	Ki	1420.0 [1], 4200.0 [2], 5890.0 [3]
	Alcuronium	IC50	4073.8 [1]
	Alcuronium	Ki	1000.0 [1], 1995.26 [2]
	(5S)-Spiro[1,3-oxazolidine-5,3'-1-azabicyclo[2.2.2]octane]-2-one	Ki	92.0 [1], 340.0 [2], 420.0 [3]
	4-Bromophenyl 1,4-diazabicyclo(3.2.2)nonane-4-carboxylate	Ki	14.0 [1]
	Bradanicline	Ki	1.0 [1], 2.75 [2]
	4-Bromo-N-[(2S,3R)-2-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-yl]benzamide	Ki	6.0 [1], 6.2 [2], 13.18 [3]
	(1R,9R,18S,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-10,26-dioxa-8,15,24,31-tetrazaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	1584.89 [1]
	(1R,9R,18S,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-10,26-dioxa-8,15,24,31-tetrazaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	1000.0 [1], 1258.93 [2]
	(2E)-2-[(1R,9Z,11S,13S,17S,18R,20R,27S,29R,30R,31S)-19-Phenyl-21-oxa-8,14,19,26-tetrazadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	IC50	1513.56 [1]
	(2E)-2-[(1R,9Z,11S,13S,17S,18R,20R,27S,29R,30R,31S)-19-Phenyl-21-oxa-8,14,19,26-tetrazadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	Ki	1258.93 [1], 1584.89 [2]
	[20-[[Dimethyl-[(4-nitrophenyl)methyl]azaniumyl]methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl-dimethyl-[(4-nitrophenyl)methyl]azanium	IC50	100000.0 [1]
	[20-[[Dimethyl-[(4-nitrophenyl)methyl]azaniumyl]methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl-dimethyl-[(4-nitrophenyl)methyl]azanium	Ki	1995.26 [1], 3981.07 [2]
	[20-[[Dimethyl(prop-2-enyl)azaniumyl]methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl-dimethyl-prop-2-enylazanium	IC50	100000.0 [1]
	[20-[[Dimethyl(prop-2-enyl)azaniumyl]methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]methyl-dimethyl-prop-2-enylazanium	Ki	3162.28 [1], 3981.07 [2]
	(1R,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-15-prop-2-enyl-10,26-dioxa-8,24,31-triaza-15-azoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	338.84 [1]
	(1R,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-15-prop-2-enyl-10,26-dioxa-8,24,31-triaza-15-azoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	50.12 [1], 63.1 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-15,31-bis(prop-2-enyl)-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	281.84 [1]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-24-Phenyl-15,31-bis(prop-2-enyl)-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	31.62 [1], 63.1 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(E)-but-2-enyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	1148.15 [1]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(E)-but-2-enyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	100.0 [1], 251.19 [2]
	2-[(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-31-(2-Acetyloxyethyl)-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaen-15-yl]ethyl acetate	IC50	1621.81 [1]
	2-[(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-31-(2-Acetyloxyethyl)-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaen-15-yl]ethyl acetate	Ki	251.19 [1], 316.23 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Dibenzyl-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	4466.84 [1]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Dibenzyl-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	199.53 [1], 251.19 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(3,4-dimethoxyphenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	1318.26 [1]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(3,4-dimethoxyphenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	63.1 [1], 125.89 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(4-bromophenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	IC50	10471.29 [1]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis[(4-bromophenyl)methyl]-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	251.19 [1], 630.96 [2]
	(2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Di(cyclohex-2-en-1-yl)-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	IC50	2344.23 [1]
	(2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Di(cyclohex-2-en-1-yl)-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	Ki	251.19 [1], 316.23 [2]
	(2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Bis[(3,4-dimethoxyphenyl)methyl]-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	IC50	2630.27 [1]
	(2E)-2-[(1S,9Z,11S,13S,17R,18R,20R,27S,29R,30R,31S)-14,26-Bis[(3,4-dimethoxyphenyl)methyl]-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	Ki	199.53 [1], 251.19 [2]
	(2E)-2-[(1S,9Z,11S,13S,18R,20R,27S,29R,30R,31S)-14,26-Bis[(4-nitrophenyl)methyl]-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	IC50	2454.71 [1]
	(2E)-2-[(1S,9Z,11S,13S,18R,20R,27S,29R,30R,31S)-14,26-Bis[(4-nitrophenyl)methyl]-19-phenyl-21-oxa-8,19-diaza-14,26-diazoniadecacyclo[24.5.2.211,14.01,27.02,7.08,31.010,18.013,17.020,30.024,29]pentatriaconta-2,4,6,9,23-pentaen-35-ylidene]ethanol	Ki	100.0 [1], 125.89 [2]
	(2E)-2-[(1S,9Z,11S,13S,25Z,27S,33S,35S,36S,38E)-38-(2-Hydroxyethylidene)-14,30-dimethyl-8,24-diaza-14,30-diazoniaundecacyclo[25.5.2.211,14.11,26.110,17.02,7.013,17.018,23.030,33.08,35.024,36]octatriaconta-2,4,6,9,18,20,22,25-octaen-28-ylidene]ethanol	IC50	9549.93 [1]
	(2E)-2-[(1S,9Z,11S,13S,25Z,27S,33S,35S,36S,38E)-38-(2-Hydroxyethylidene)-14,30-dimethyl-8,24-diaza-14,30-diazoniaundecacyclo[25.5.2.211,14.11,26.110,17.02,7.013,17.018,23.030,33.08,35.024,36]octatriaconta-2,4,6,9,18,20,22,25-octaen-28-ylidene]ethanol	Ki	1584.89 [1], 2511.89 [2]
	[1-[(3-Hydroxyphenyl)methyl]indol-3-yl]methyl-trimethylazanium	IC50	1000.0 [1]
	[1-[(3-Hydroxyphenyl)methyl]indol-3-yl]methyl-trimethylazanium	Ki	600.0 [1], 145000.0 [2]
	Acetylcholine	Ki	501.19 [1], 7943.28 [2]
	Naltrexone	IC50	25000.0 [1], 30000.0 [2]
	Bupropion	IC50	7900.0 [1], 50000.0 [2]
	Mecamylamine	IC50	1800.0 [1], 12300.0 [2]
	Tropisetron	Ki	6.9 [1]
	Nornicotine	Ki	730.0 [1], 138000.0 [2]
	Benzamide, N-(3R)-1-azabicyclo[2.2.2]oct-3-yl-4-chloro-	Ki	24.55 [1], 26.0 [2]
	Pozanicline	Ki	10000.0 [1]
	Stilonium iodide	IC50	41.0 [1]
	Stilonium iodide	Ki	104.0 [1]
	5-{6-[(3R)-1-Azabicyclo[2.2.2]oct-3-yloxy]pyridazin-3-yl}-1H-indole	Ki	0.2 [1], 7.0 [2]
	Encenicline	Ki	4.3 [1], 9.98 [2]
	Spiro[1-azabicyclo[2.2.2]octane-3,2'(3'H)-furo[2,3-b]pyridine], (2'R)-	Ki	3.0 [1]
	Psab-ofp	Ki	2.0 [1], 3.1 [2]
	3-(5-Chloro-2-furoyl)-3,7-diazabicyclo[3.3.0]octane	Ki	6700.0 [1]
	(4-Bromo-phenyl)-carbamic acid 1-aza-bicyclo[2.2.2]oct-3-yl ester	Ki	40.0 [1], 167.0 [2]
	N-(1-Azabicyclo[2.2.2]octan-3-yl)-1-benzothiophene-2-carboxamide	Ki	14.6 [1]
	Cyclopropyl(3,7-diazabicyclo[3.3.1]nonan-3-yl)methanone	Ki	20.0 [1]
	2,3,3a,4,6,6a-Hexahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl(cyclopropyl)methanone	Ki	840.0 [1]
	1-[20-[(Dimethylamino)methyl]-3,13-diazapentacyclo[11.7.0.03,11.04,9.014,19]icosa-1(20),4,6,8,10,14,16,18-octaen-10-yl]-N,N-dimethylmethanamine	Ki	5011.87 [1], 19952.62 [2]
	N-[(2S,3R)-2-(Pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-yl]benzamide	Ki	61.66 [1], 97.0 [2]
	(4-Chlorophenyl)(4-isopropyl-1,4-diazocan-1-yl)methanone	IC50	7000.0 [1]
	4-Chloro-N-(1,2,3,5,6,7-hexahydropyrrolizin-8-ylmethyl)benzamide	IC50	7200.0 [1]
	[(3S,9Ar)-3-methyl-1,3,4,6,7,8,9,9a-octahydropyrido[1,2-a]pyrazin-2-yl]-(2,3-dihydro-1,4-benzodioxin-6-yl)methanone	IC50	6100.0 [1]
	(4-Bromophenyl) (9aS)-1,3,4,5,7,8,9,9a-octahydropyrrolo[1,2-a][1,4]diazepine-2-carboxylate	IC50	5600.0 [1]
	4-[4-[(E)-2-(3,5-Dimethoxyphenyl)ethenyl]phenoxy]butyl-triethylazanium;iodide	IC50	24.3 [1]
	4-[4-[(E)-2-(3,5-Dimethoxyphenyl)ethenyl]phenoxy]butyl-triethylazanium;iodide	Ki	305.0 [1]
	4-[4-[(E)-2-(3,5-Dimethoxyphenyl)ethenyl]phenoxy]butyl-triphenylphosphanium;iodide	IC50	10000.0 [1]
	4-[4-[(E)-2-(3,5-Dimethoxyphenyl)ethenyl]phenoxy]butyl-triphenylphosphanium;iodide	Ki	1826.0 [1]
	Triethyl-[6-[4-[(E)-2-phenylethenyl]phenoxy]hexyl]azanium;iodide	IC50	12.3 [1]
	Triethyl-[6-[4-[(E)-2-phenylethenyl]phenoxy]hexyl]azanium;iodide	Ki	465.0 [1]
	Triethyl-[4-[4-[(E)-2-phenylethenyl]phenoxy]butyl]azanium;iodide	IC50	6.5 [1]
	Triethyl-[4-[4-[(E)-2-phenylethenyl]phenoxy]butyl]azanium;iodide	Ki	186.0 [1]
	Triethyl-[8-[4-[(E)-2-phenylethenyl]phenoxy]octyl]azanium;iodide	IC50	92.0 [1]
	Triethyl-[8-[4-[(E)-2-phenylethenyl]phenoxy]octyl]azanium;iodide	Ki	164.0 [1]
	2-[4-[(E)-2-(3,5-Dimethoxyphenyl)ethenyl]phenoxy]ethyl-triethylazanium;iodide	IC50	47.0 [1]
	2-[4-[(E)-2-(3,5-Dimethoxyphenyl)ethenyl]phenoxy]ethyl-triethylazanium;iodide	Ki	189.0 [1]
	[(1r,5s)-8-Phenethyl-8-Azabicyclo[3.2.1]octan-3-Yl] Benzoate	Ki	5011.87 [1], 7943.28 [2]
	[(1S,5R)-8-[2-(3,5-Dihydroxyphenyl)-2-hydroxyethyl]-8-azabicyclo[3.2.1]octan-3-yl] benzoate	Ki	12589.25 [1], 15848.93 [2]
	N-[(3R)-1-Azabicyclo[2.2.2]octan-3-yl]-5-bromoindolizine-2-carboxamide	Ki	14.9 [1], 93.6 [2]
	(1S,9R,18R,19S,21R,22R,23R,25R,32S,34R,35R,36S)-15,31-Bis(naphthalen-2-ylmethyl)-24-phenyl-10,26-dioxa-8,24-diaza-15,31-diazoniaundecacyclo[29.5.2.01,32.02,7.08,36.09,22.013,21.015,19.018,23.025,35.029,34]octatriaconta-2,4,6,12,28-pentaene	Ki	316.23 [1], 630.96 [2]
	[1-[(4-Hydroxyphenyl)methyl]indol-3-yl]methyl-trimethylazanium	IC50	2200.0 [1]
	[1-[(4-Hydroxyphenyl)methyl]indol-3-yl]methyl-trimethylazanium	Ki	2900.0 [1]
	Carbastat	Ki	66000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Neuronal acetylcholine receptor protein alpha-7 subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-protein-alpha-7-subunit-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Neuronal acetylcholine receptor protein alpha-7 subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/neuronal-acetylcholine-receptor-protein-alpha-7-subunit-inhibitors-ic50-ki.
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