Name: Neuropeptide FF receptor 1 Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Neuropeptide FF receptor 1 Inhibitors (IC50, Ki)

Structure	Compound Name	Standard Type	Standard Values (in nM)
	(2R)-5-(Diaminomethylideneamino)-2-[(2,2-diphenylacetyl)amino]-N-[(4-hydroxyphenyl)methyl]pentanamide	Ki	12.0 ^[1], 18.0 ^[2]
	(2S)-2-[[(2S)-1-[(2S)-5-Amino-2-[[(2S)-2-[[(2R)-2-[[(2R)-2-amino-3-(4-hydroxyphenyl)propanoyl]-methylamino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]-5-oxopentanoyl]pyrrolidine-2-carbonyl]amino]-N-[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]pentanediamide	Ki	3.85 ^[1], 4.0 ^[2]
	Kisspeptin-10	IC50	4.7 ^[1]
	1-Adamantanecarbonyl-RF-NH2	Ki	22.0 ^[1]
	N-[(2S)-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-Amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-2-oxoethyl]amino]-1-oxo-3-phenylpropan-2-yl]-4-fluorobenzamide	IC50	160.0 ^[1]
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References

This online resource may be cited as follows

MLA	"Quest Database™ Neuropeptide FF receptor 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 16 Mar. 2026, https://www.aatbio.com/data-sets/neuropeptide-ff-receptor-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2026, March 16). Quest Database™ Neuropeptide FF receptor 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/neuropeptide-ff-receptor-1-inhibitors-ic50-ki.
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