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Nuclear factor NF-kappa-B complex Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
Pyrrolidine dithiocarbamic acidIC5034500.0 [1], 37200.0 [2]
(1E,4Z,6E)-5-Hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneIC508000.0 [1], 20900.0 [2]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-chloro-4-(trifluoromethyl)pyrimidine-5-carboxamideIC5050.0 [1]
6-Hydroxy-7-methoxy-N-phenyl-3,4-dihydro-2H-chromene-2-carboxamideIC5037200.0 [1], 40100.0 [2]
2-Phenyl-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC50100.0 [1]
Ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)-2-(trifluoromethyl)pyrimidine-5-carboxylateIC501000.0 [1]
2-(2-Thienyl)-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC5020.0 [1]
CID 10407641IC5050.0 [1]
CID 10499355IC504000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2,4-bis(trifluoromethyl)pyrimidine-5-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-cyano-4-(trifluoromethyl)pyrimidine-5-carboxamideIC5010000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-6-chloro-4-(trifluoromethyl)pyridazine-3-carboxamideIC5010000.0 [1]
CID 10666814IC501700.0 [1]
N-(3,5-Bis-trifluoromethyl-phenyl)-4-chloro-2-trifluoromethyl-benzamideIC5030000.0 [1]
N-[3,5-Bis(trifluoromethyl)phenyl]-2-fluoro-4-(trifluoromethyl)pyrimidine-5-carboxamideIC50400.0 [1]
CID 10741998IC50400.0 [1]
CID 10763720IC50600.0 [1]
ResveratrolIC502500.0 [1]
BortezomibIC509.7 [1]
PhloretinIC5041000.0 [1]
SanguinarineIC502000.0 [1]
(E)-3-TosylacrylonitrileIC502000.0 [1]
Tosylphenylalanyl chloromethyl ketoneIC503800.0 [1]
ParthenolideIC503400.0 [1]
IsoliquiritigeninIC5032000.0 [1]
beta-LapachoneIC504000.0 [1]
IxazomibIC506.2 [1]
ButeinIC5038000.0 [1]
TetrahydrocurcuminIC5050000.0 [1]
GoniothalaminIC507000.0 [1]
Lantadene AIC501060.0 [1]
4-HydroxychalconeIC5024000.0 [1]
(1E,4E)-1,5-Bis(4-hydroxy-3-methoxyphenyl)penta-1,4-dien-3-oneIC501800.0 [1]
HydrazinocurcuminIC5029800.0 [1]
1-(5-Methoxy-2-(thiophen-2-yl)quinazolin-4-ylamino)-3-methyl-1H-pyrrole-2,5-dioneIC508.0 [1]
4-MethoxychalconeIC5029000.0 [1]
HeteroneminIC505000.0 [1]
(1'S,3'R,5'S,7'R,10'R,12'R,14'R,15'S,18'R,19'R,22'S,23'R)-10',22'-Dihydroxy-14'-(hydroxymethyl)-7',18'-dimethyl-19'-(5-oxo-2H-furan-3-yl)spiro[1,3-thiazolidine-2,9'-4,6,11-trioxahexacyclo[12.11.0.03,12.05,10.015,23.018,22]pentacosane]-4-oneIC5030.0 [1]
Altersolanol AIC50800.0 [1]
Lantadene BIC501560.0 [1]
(4R,4As,6aR,6aS,6bR,8aR,10S,12aR,14bS)-10-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-4-[(Z)-2-methylbut-2-enoyl]oxy-1,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydropicene-4a-carboxylic acidIC50980.0 [1]
2',4-Dihydroxy-4',6'-dimethoxychalconeIC508000.0 [1]
HomobuteinIC5038000.0 [1]
(4R,4As,6aR,6aS,6bR,8aR,12aR,14bS)-4-hydroxy-2,2,6a,6b,9,9,12a-heptamethyl-10-oxo-3,4,5,6,6a,7,8,8a,11,12,13,14b-dodecahydro-1H-picene-4a-carboxylic acidIC506420.0 [1]
1-(6-Methoxy-2-thiophen-2-yl-quinazolin-4-ylamino)-3-methyl-pyrrole-2,5-dioneIC503.0 [1]
3-(4-Chloro-phenyl)-2-(4-methyl-2-methylamino-thiazol-5-yl)-3H-quinazolin-4-oneIC501200.0 [1]
2-[2-(4-Chloroanilino)-4-methyl-1,3-thiazol-5-yl]-3-(4-chlorophenyl)quinazolin-4-oneIC501200.0 [1]
Reduced Lantadene BIC501020.0 [1]
Ethyl 2-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]-4-(5-methylthiophen-2-yl)pyrimidine-5-carboxylateIC5045.0 [1]
Ethyl 4-ethyl-2-[methyl-(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC5035.0 [1]
MyricatomentogeninIC509400.0 [1]
2-(4-Methyl-2-phenylamino-thiazol-5-yl)-3-o-tolyl-3H-quinazolin-4-oneIC505500.0 [1]
4-[(E)-2-[3-(4-Hydroxy-3-methoxyphenyl)-1H-pyrazol-5-yl]ethenyl]-2-methoxyphenolIC5030000.0 [1]
Lantadene DIC5010000.0 [1]
3-(4-Acetylphenyl)-2-(5-morpholin-4-yl-4-pyridin-4-ylthiophen-2-yl)quinazolin-4-oneIC5010000.0 [1]
(4R,4As,6aR,6aS,6bR,8aR,12aR,14bS)-4-butanoyloxy-2,2,6a,6b,9,9,12a-heptamethyl-10-oxo-3,4,5,6,6a,7,8,8a,11,12,13,14b-dodecahydro-1H-picene-4a-carboxylic acidIC5010000.0 [1]
2-(4-Methyl-2-methylamino-thiazol-5-yl)-3-o-tolyl-3H-quinazolin-4-oneIC505500.0 [1]
Ethyl 2-(4-fluorophenyl)-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)pyrimidine-5-carboxylateIC50700.0 [1]
Ethyl 2-(3-methoxyphenyl)-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)pyrimidine-5-carboxylateIC505000.0 [1]
Ethyl 2-(4-methoxyphenyl)-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)pyrimidine-5-carboxylateIC50900.0 [1]
Ethyl 2-(furan-2-carbonyl)-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)pyrimidine-5-carboxylateIC50700.0 [1]
Ethyl 2-(1-benzothiophen-2-yl)-4-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC504000.0 [1]
Ethyl 2-(5-chlorothiophen-2-yl)-4-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC50300.0 [1]
Ethyl 2-(3,5-dimethylpyrazol-1-yl)-4-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC5010000.0 [1]
2-(4-Pyridinyl)-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC506000.0 [1]
Ethyl 2-(cyclohexenylmethyl)-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)pyrimidine-5-carboxylateIC502000.0 [1]
2-Cyclopropyl-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC501000.0 [1]
Ethyl 4-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxylateIC508000.0 [1]
Ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)-2-(quinolin-3-yl)pyrimidine-5-carboxylateIC506000.0 [1]
Ethyl 2-(2,6-dichloropyridin-4-yl)-4-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC502000.0 [1]
Ethyl 2-(3,5-dichlorophenyl)-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)pyrimidine-5-carboxylateIC50300.0 [1]
1-[2-(2-Thienyl)-5-(4-methyl-2-oxazolyl)pyrimidine-4-ylamino]-3-methyl-3-pyrroline-2,5-dioneIC50200.0 [1]
4-(3-Methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)-2-(thiophen-2-yl)pyrimidine-5-carbonitrileIC505000.0 [1]
Ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)-2-(3-nitrophenyl)pyrimidine-5-carboxylateIC507000.0 [1]
Ethyl 2-(3-bromophenyl)-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)pyrimidine-5-carboxylateIC50700.0 [1]
1-[2-(2-Thienyl)5-(2-methyl-2H-tetrazole-5-yl)pyrimidine-4-ylamino]-3-methyl-3-pyrroline-2,5-dioneIC50200.0 [1]
Ethyl 4-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]-2-(5-methylthiophen-2-yl)pyrimidine-5-carboxylateIC50200.0 [1]
2-(3-Thienyl)-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC50100.0 [1]
1-[2-(2-Thienyl)5-(3-methyl-5-isoxazolyl)pyrimidine-4-ylamino]-3-methyl-3-pyrroline-2,5-dioneIC50300.0 [1]
2-(Trifluoromethyl)-4-(2,5-dioxo-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC5010000.0 [1]
1-[2-(2-Thienyl)-5-(2-oxazoline-2-yl)pyrimidine-4-ylamino]-3-methyl-3-pyrroline-2,5-dioneIC50200.0 [1]
Ethyl 4-(2,5-dioxo-3-phenyl-2H-pyrrol-1(5H)-ylamino)-2-(trifluoromethyl)pyrimidine-5-carboxylateIC5020000.0 [1]
Ethyl 4-(3,4-dimethyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)-2-(trifluoromethyl)pyrimidine-5-carboxylateIC5010000.0 [1]
3-Methyl-1-[[5-(5-methyl-1,3,4-oxadiazol-2-yl)-2-thiophen-2-ylpyrimidin-4-yl]amino]pyrrole-2,5-dioneIC50300.0 [1]
2-Phenoxy-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC5015000.0 [1]
2-Benzyl-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC507000.0 [1]
2-Ethyl-4-[methyl(2,5-dioxo-3-methyl-3-pyrroline-1-yl)amino]pyrimidine-5-carboxylic acid ethyl esterIC5010000.0 [1]
Ethyl 2-(4-fluorophenyl)-4-[methyl-(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC503000.0 [1]
2-(Phenylthio)-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC501000.0 [1]
Ethyl 2-(4-chlorophenyl)-4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)pyrimidine-5-carboxylateIC50300.0 [1]
2-(Methylthio)-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC50200.0 [1]
Ethyl 4-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]-2-[4-(trifluoromethyl)phenyl]pyrimidine-5-carboxylateIC50400.0 [1]
2-Methyl-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC5016000.0 [1]
2-Ethyl-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC5010000.0 [1]
Ethyl 4-[methyl-(3-methyl-2,5-dioxopyrrol-1-yl)amino]-2-thiophen-2-ylpyrimidine-5-carboxylateIC501000.0 [1]
Ethyl 4-[acetyl-(3-methyl-2,5-dioxopyrrol-1-yl)amino]-2-phenylpyrimidine-5-carboxylateIC504000.0 [1]
Ethyl 4-(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-ylamino)-2-(phenylsulfonyl)pyrimidine-5-carboxylateIC5010000.0 [1]
Ethyl 4-(methyl(3-methyl-2,5-dioxo-2H-pyrrol-1(5H)-yl)amino)-2-phenylpyrimidine-5-carboxylateIC502000.0 [1]
2-Tert-Butyl-4-(2,5-dioxo-3-methyl-3-pyrroline-1-ylamino)pyrimidine-5-carboxylic acid ethyl esterIC501000.0 [1]
Ethyl 4-ethyl-2-[(3-methyl-2,5-dioxopyrrol-1-yl)amino]pyrimidine-5-carboxylateIC50400.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Nuclear factor NF-kappa-B complex Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/nuclear-factor-nf-kappa-b-complex-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Nuclear factor NF-kappa-B complex Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/nuclear-factor-nf-kappa-b-complex-inhibitors-ic50-ki.
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