 | N-[4-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide | IC50 | 204.0 [1], 1700.0 [2], 2010.0 [3], 4400.0 [4] |
| N-[4-(1,1,1,3,3,3-Hexafluoro-2-hydroxypropan-2-yl)phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide | Ki | 51.0 [1] |
 | CID 51035449 | IC50 | 110.0 [1], 320.0 [2], 3540.0 [3] |
| CID 51035449 | Ki | 105.0 [1] |
 | N-[5-(2-Chlorobenzoyl)-4-(3-chlorophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 15.85 [1], 22.0 [2], 180.0 [3] |
| N-[5-(2-Chlorobenzoyl)-4-(3-chlorophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | Ki | 39.81 [1] |
 | N-(5-Benzoyl-4-phenyl-1,3-thiazol-2-yl)-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 10.0 [1], 31.62 [2], 39.81 [3] |
 | N-[4-(2,5-Dichlorophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 1000.0 [1] |
| N-[4-(2,5-Dichlorophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | Ki | 398.11 [1] |
 | N-[5-(2-Chlorobenzoyl)-4-(3-chlorophenyl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 2.0 [1], 6.0 [2], 10.0 [3], 23.0 [4] |
| N-[5-(2-Chlorobenzoyl)-4-(3-chlorophenyl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | Ki | 25.12 [1] |
 | Chembl4175305 | IC50 | 0.6 [1], 14.0 [2], 17.0 [3], 23.0 [4], 255.0 [5] |
 | Digoxin | IC50 | 1980.0 [1], 2000.0 [2], 4000.0 [3], 4100.0 [4] |
 | Ursolic acid | IC50 | 130.0 [1], 680.0 [2], 1060.0 [3], 9410.0 [4] |
 | CID 118622692 | IC50 | 1.9 [1], 3.1 [2], 6.1 [3], 14.0 [4] |
 | 5-[(1R)-1-[(3,5-Difluoro-4-trimethylsilylphenyl)carbamoyl]-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl]-5-oxopentanoic acid | IC50 | 3.0 [1], 23.0 [2] |
 | N-[(1R)-2-(3,5-Difluoro-4-trimethylsilylanilino)-1-(4-methoxyphenyl)-2-oxoethyl]-N-methyl-3-oxo-1,2-oxazole-5-carboxamide | IC50 | 4.3 [1], 13.0 [2], 18.0 [3] |
 | 3-[(5R)-5-[(7-Fluoro-1,1-dimethyl-2,3-dihydroinden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-5H-1,6-naphthyridine-6-carbonyl]cyclobutane-1-carboxylic acid | IC50 | 2.0 [1], 2.6 [2], 31.0 [3], 34.0 [4] |
 | 4-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]pyridine-2-carboxamide | IC50 | 5.0 [1], 130.0 [2] |
| 4-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]pyridine-2-carboxamide | Ki | 20.0 [1] |
 | 3-[2-[(5R)-5-[(7-Fluoro-1,1-dimethyl-2,3-dihydroinden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-5H-1,6-naphthyridin-6-yl]-2-oxoethyl]cyclobutane-1-carboxylic acid | IC50 | 3.0 [1], 3.3 [2], 27.0 [3], 29.0 [4] |
 | 4-Cyano-N-[3-[1-(cyclohexanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]pyridine-2-carboxamide | IC50 | 5.0 [1], 42.0 [2], 120.0 [3] |
| 4-Cyano-N-[3-[1-(cyclohexanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]pyridine-2-carboxamide | Ki | 20.0 [1] |
 | 3-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1H-indol-5-yl]benzamide | IC50 | 54.0 [1], 2700.0 [2], 2900.0 [3] |
| 3-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1H-indol-5-yl]benzamide | Ki | 1200.0 [1] |
 | CID 44241473 | IC50 | 2000.0 [1] |
| CID 44241473 | Ki | 111.0 [1] |
 | 1-Ethyl-N-isonicotinoyl-N-(4-methoxyphenyl)-2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide | IC50 | 80.0 [1], 90.0 [2], 5880.0 [3] |
 | CID 71470549 | IC50 | 1000.0 [1], 1500.0 [2] |
| CID 71470549 | Ki | 1000.0 [1] |
 | N-(3-Chloro-4-cyanophenyl)-N'-(9-ethylcarbazol-3-yl)-3-methylpentanediamide | IC50 | 2.1 [1], 11.0 [2], 50.6 [3] |
 | 4'-[[(2-Methylpropyl)(benzylsulfonyl)amino]methyl]-1,1'-biphenyl-4-carboxamide | IC50 | 31.0 [1], 33.0 [2] |
 | N-(4-(1-Ethyl-2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamido)phenyl)acetamide | IC50 | 90.0 [1], 320.0 [2], 89760.0 [3] |
 | N-[3-Chloro-4-[2-(trifluoromethyl)phenyl]phenyl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 6.31 [1], 7.94 [2], 15.85 [3] |
 | [4-Chloro-2-methoxy-3-[(4-pyrazol-1-ylphenyl)methyl]quinolin-6-yl]-(4-chlorophenyl)-(3-methylimidazol-4-yl)methanol | IC50 | 73.0 [1], 85.0 [2], 670.0 [3] |
 | [4-Chloro-2-methoxy-3-[(4-pyrazol-1-ylphenyl)methyl]quinolin-6-yl]-(3-methylimidazol-4-yl)-[6-(trifluoromethyl)pyridin-3-yl]methanol | IC50 | 57.0 [1], 89.0 [2], 170.0 [3] |
 | 4-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-ethylindol-5-yl]pyridine-2-carboxamide | IC50 | 295.0 [1], 10000.0 [2] |
| 4-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-ethylindol-5-yl]pyridine-2-carboxamide | Ki | 19000.0 [1] |
 | N-(4-Methoxyphenyl)-4-{[(2-oxo-1,2-dihydrobenzo[cd]indol-6-yl)sulfonyl]amino}benzamide | IC50 | 180.0 [1], 380.0 [2], 8350.0 [3] |
 | N-[4-(5-Cyano-2-methoxyphenyl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 20.0 [1], 30.0 [2], 3300.0 [3] |
 | Methyl 4-[[3-[5-[[2-(4-ethylsulfonylphenyl)acetyl]amino]thiophen-3-yl]pyridin-2-yl]oxymethyl]benzoate | IC50 | 14.0 [1], 21.0 [2], 35.0 [3] |
 | 2-Acetamido-N-[4-(5-cyano-3-fluoro-2-methoxyphenyl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 9.0 [1], 57.0 [2], 63.0 [3] |
 | 2-Oxo-N-(4-phenoxyphenyl)-1,2-dihydrobenzo[cd]indole-6-sulfonamide | IC50 | 140.0 [1], 150.0 [2], 3090.0 [3] |
 | N-[4-(4-Morpholinyl)phenyl]-2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide | IC50 | 300.0 [1], 410.0 [2], 48420.0 [3] |
 | 2-Amino-N-[4-(5-cyano-3-fluoro-2-methoxyphenyl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 75.0 [1], 452.0 [2], 1690.0 [3] |
 | 2-Acetamido-N-[4-(5-cyano-2-methoxypyridin-3-yl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 14.0 [1], 67.0 [2], 990.0 [3] |
 | N-[4-(5-Cyano-2-methoxypyridin-3-yl)thiophen-2-yl]-2-[4-(methylsulfamoyl)phenyl]acetamide | IC50 | 40.0 [1], 70.0 [2], 3300.0 [3] |
 | 2-Acetamido-N-[4-[2-(4-cyanophenoxy)pyridin-3-yl]thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 55.0 [1], 66.0 [2], 640.0 [3] |
 | N-[4-[2-[(4-Cyanophenyl)methoxy]pyridin-3-yl]thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 10.0 [1], 30.0 [2], 100.0 [3] |
 | N-[4-[5-Cyano-2-(2,2,2-trifluoroethoxy)pyridin-3-yl]thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 2.0 [1], 30.0 [2], 65.0 [3] |
 | (2S)-2-Acetamido-2-(4-ethylsulfonylphenyl)-N-[4-[2-[[4-(trifluoromethoxy)phenyl]methoxy]pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 23.0 [1], 270.0 [2], 3530.0 [3] |
 | 2-(4-Ethylsulfonylphenyl)-N-[4-[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 18.0 [1], 50.0 [2], 100.0 [3] |
 | N-[4-(5-Cyano-3-fluoro-2-methoxyphenyl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 20.0 [1], 30.0 [2], 700.0 [3] |
 | 2-Acetamido-N-[4-[5-cyano-2-(2,2,2-trifluoroethoxy)pyridin-3-yl]thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 7.0 [1], 49.0 [2], 72.0 [3] |
 | 2-(4-Ethylsulfonylphenyl)-N-[4-[2-[[4-(trifluoromethoxy)phenyl]methoxy]pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 7.0 [1], 25.0 [2], 30.0 [3] |
 | (2R)-2-Acetamido-2-(4-ethylsulfonylphenyl)-N-[4-[2-[[4-(trifluoromethoxy)phenyl]methoxy]pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 3.0 [1], 11.0 [2], 34.0 [3] |
 | N-[4-(5-Cyano-2-methoxypyridin-3-yl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 30.0 [1], 40.0 [2], 3300.0 [3] |
 | 2-(4-Ethylsulfonylphenyl)-N-[4-[2-[(E)-3-phenylprop-2-enoxy]pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 11.0 [1], 25.0 [2], 29.0 [3] |
 | 2-Acetamido-2-(4-ethylsulfonylphenyl)-N-[4-[2-[[4-(trifluoromethoxy)phenyl]methoxy]pyridin-3-yl]thiophen-2-yl]acetamide | IC50 | 6.0 [1], 32.0 [2], 75.0 [3] |
 | N-(6-Ethoxy-1,3-benzothiazol-2-yl)-1-ethyl-2-oxo-1,2-dihydrobenzo[cd]indole-6-sulfonamide | IC50 | 930.0 [1], 1350.0 [2], 6720.0 [3] |
 | 1-Ethyl-2-oxo-N-(4-phenyldiazenylphenyl)benzo[cd]indole-6-sulfonamide | IC50 | 200.0 [1], 6050.0 [2] |
 | 3-(1,3-Benzodioxol-5-yl)-1-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-3-(2-hydroxy-4,6-dimethoxyphenyl)propan-1-one | IC50 | 300.0 [1], 605.0 [2], 1100.0 [3] |
 | N-[4-(3-Chlorophenyl)thiophen-2-yl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 110.0 [1], 180.0 [2], 3000.0 [3] |
 | N-(4-Acetylphenyl)-1-ethyl-2-oxobenzo[cd]indole-6-sulfonamide | IC50 | 40.0 [1], 50.0 [2], 70140.0 [3] |
 | N-(3,4-Dimethoxyphenyl)-1-ethyl-2-oxobenzo[cd]indole-6-sulfonamide | IC50 | 20.0 [1], 50.0 [2], 20100.0 [3] |
 | 3-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]benzamide | IC50 | 5.5 [1], 170.0 [2] |
| 3-Cyano-N-[3-[1-(cyclopentanecarbonyl)piperidin-4-yl]-1-methylindol-5-yl]benzamide | Ki | 50.0 [1] |
 | N-(7,7-Dimethyl-9-oxo-6,8-dihydrodibenzofuran-3-yl)-2-oxo-1H-benzo[cd]indole-6-sulfonamide | IC50 | 7560.0 [1], 11840.0 [2], 20270.0 [3] |
 | 1-Ethyl-N-isoquinolin-8-yl-2-oxobenzo[cd]indole-6-sulfonamide | IC50 | 100.0 [1], 150.0 [2], 17520.0 [3] |
 | 1-Ethyl-N-(4-morpholin-4-ylphenyl)-2-oxobenzo[cd]indole-6-sulfonamide | IC50 | 340.0 [1], 550.0 [2], 12150.0 [3] |
 | Tert-butyl N-[3-[(1-ethyl-2-oxobenzo[cd]indol-6-yl)sulfonylamino]phenyl]carbamate | IC50 | 2510.0 [1], 3390.0 [2], 7040.0 [3] |
 | N-(2-Tert-butylphenyl)-1-ethyl-2-oxobenzo[cd]indole-6-sulfonamide | IC50 | 4900.0 [1], 9980.0 [2], 18980.0 [3] |
 | N-[(2,5-Dichlorophenyl)methyl]-1-ethyl-2-oxobenzo[cd]indole-6-sulfonamide | IC50 | 130.0 [1], 1080.0 [2], 31610.0 [3] |
 | 5-Butyl-2-[2,2,2-trifluoro-1-hydroxy-1-(trifluoromethyl)ethyl]phenanthridin-6-one | IC50 | 3900.0 [1], 4700.0 [2] |
 | N-[1-(4-Methoxyphenyl)-2-oxo-2-(4-propan-2-ylanilino)ethyl]-N-methyl-6-oxo-1H-pyridine-3-carboxamide | IC50 | 200.0 [1], 1600.0 [2] |
 | CID 118977746 | IC50 | 4.1 [1], 9.5 [2] |
 | ROR gamma-t-IN-1 | IC50 | 3.98 [1], 34.0 [2] |
 | N-(2-Methylpropyl)-N-[[4-(4-methylsulfonylphenyl)phenyl]methyl]-1-phenylmethanesulfonamide | IC50 | 32.0 [1] |
 | N-[2-(4-Tert-butylanilino)-1-(4-methoxyphenyl)-2-oxoethyl]-N-methyl-6-oxo-1H-pyridine-3-carboxamide | IC50 | 100.0 [1], 270.0 [2] |
 | 4-Chloro-3-[4-[(1-methylindol-4-yl)sulfonyl-(2,2,2-trifluoroethyl)amino]phenyl]benzamide | IC50 | 710.0 [1] |
 | N-[4-[Hydroxy(dimethyl)silyl]phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide | IC50 | 11000.0 [1], 43000.0 [2] |
 | N-(2,4-Difluorophenyl)-2-[4-[[2-(4-ethylsulfonylphenyl)acetyl]amino]-2-fluorophenyl]-2-methylpropanamide | IC50 | 13.0 [1], 30.0 [2] |
 | 2-Chloro-6-fluoro-N-[1-(4-fluorophenyl)sulfonyl-3,4-dihydro-2H-quinolin-7-yl]benzamide | IC50 | 15000.0 [1] |
 | N-[[5-[4-(Methanesulfonamido)phenyl]thiophen-2-yl]methyl]-N-(2-methylpropyl)-1-phenylmethanesulfonamide | IC50 | 31.0 [1], 71.0 [2] |
 | 4-Chloro-3-[1-(2-chloro-6-fluorobenzoyl)-3,4-dihydro-2H-quinolin-6-yl]benzamide | IC50 | 220.0 [1] |
 | N-[4-(5-Carbamoyl-2-chlorophenyl)-2-(2,2,2-trifluoroethoxy)phenyl]-2-chloro-6-fluoro-N-(trideuteriomethyl)benzamide | IC50 | 29.0 [1] |
 | 4-Fluoro-N-[4-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)phenyl]-N-(2,2,2-trifluoroethyl)benzenesulfonamide | IC50 | 34.0 [1] |
 | (2,4-Dichloro-3-phenylquinolin-6-yl)(1-methyl-1H-imidazol-5-yl)(pyridin-4-yl)methanol | IC50 | 50.0 [1] |
 | N-[4-[[(4-Cyclopentyloxyphenyl)methyl-propylamino]methyl]phenyl]-2-(4-ethylsulfonylphenyl)acetamide | IC50 | 20.0 [1], 32.0 [2] |
 | N-(2-Methylpropyl)-N-({5-[4-(Methylsulfonyl)phenyl]thiophen-2-Yl}methyl)-1-Phenylmethanesulfonamide | IC50 | 130.0 [1] |
 | [2-Amino-4-[3-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl]-(2-chlorophenyl)methanone | IC50 | 40000.0 [1] |
 | 3-[1-(2-Chloro-6-fluorobenzoyl)-3,4-dihydro-2H-quinolin-6-yl]-5-fluorobenzamide | IC50 | 13000.0 [1] |
 | (4-Chlorophenyl)-(2,4-dichloro-3-phenylquinolin-6-yl)-(3-methylimidazol-4-yl)methanol | IC50 | 260.0 [1], 5500.0 [2] |
 | 1-Ethyl-N-(2-morpholin-4-ylethyl)-2-oxobenzo[cd]indole-6-sulfonamide | IC50 | 290.0 [1], 350.0 [2] |
 | N-(1-Acetylpiperidin-4-yl)-1-ethyl-2-oxobenzo[cd]indole-6-sulfonamide | IC50 | 90.0 [1], 270.0 [2] |
 | N-[(1-Acetylpiperidin-4-Yl)methyl]-1-Ethyl-2-Oxo-1,2-Dihydrobenzo[cd]indole-6-Sulfonamide | IC50 | 590.0 [1], 6030.0 [2] |
 | [4-Chloro-3-[(4-fluorophenyl)methyl]-2-methoxyquinolin-6-yl]-(4-chlorophenyl)-(3-methylimidazol-4-yl)methanol | IC50 | 420.0 [1], 6000.0 [2] |
 | [4-Chloro-3-[(4-fluorophenyl)methyl]-2-methoxyquinolin-6-yl]-(3-methylimidazol-4-yl)-[6-(trifluoromethyl)pyridin-3-yl]methanol | IC50 | 2740.0 [1], 6000.0 [2] |
 | N-(3-Chloro-4-cyanophenyl)-N'-(4-ethyl-3-oxo-1,4-benzoxazin-7-yl)-3-methylpentanediamide | IC50 | 110.0 [1], 1400.0 [2] |
 | N-(3-Chloro-4-cyanophenyl)-N'-(2,4-diethyl-3-oxo-1,4-benzoxazin-7-yl)-3-methylpentanediamide | IC50 | 7.5 [1], 100.0 [2] |
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