Oligosaccharyl transferase 48 kDa subunit Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	82.0 [1]
	(3R,6S)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-Amino-3-(4-nitrophenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-6-[2-(decylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	61.0 [1]
	(3R,6S)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-Amino-3-(4-nitrophenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-6-[2-(naphthalen-2-ylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	40.0 [1]
	(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-amino-3-(4-nitrophenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	37.0 [1]
	(3R,6S)-N-[(2S,3R)-3-Hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-[2-(4-nitrophenyl)ethylamino]-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-6-[2-(naphthalen-2-ylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	10.0 [1]
	(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-3-hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-[2-(4-nitrophenyl)ethylamino]-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	20.0 [1]
	(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-3-hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-oxo-1-(4-phenylbutylamino)butan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	50.0 [1]
	(3R,6S)-N-[(2S,3R)-3-Hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-oxo-1-(2-phenylethylamino)butan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-6-[2-(naphthalen-2-ylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	18.0 [1]
	(3R,6S)-6-(2-Aminoethyl)-N-[(2S,3R)-3-hydroxy-1-[[(2S)-1-[[(2S,3R)-3-hydroxy-1-oxo-1-(2-phenylethylamino)butan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxobutan-2-yl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	44.0 [1]
	(3R,6S)-N-[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-Amino-3-(4-nitrophenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]-6-[2-(naphthalen-1-ylamino)ethyl]-5,8-dioxo-1-thia-4,7-diazacyclotridecane-3-carboxamide	Ki	98.0 [1]
	(2S)-N-[2-[[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-Amino-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-2-oxoethyl]-2-(benzylamino)-5-[(4-nitrophenyl)methylamino]pentanamide	Ki	154.0 [1]
	(2S)-N-[2-[[(2S,3R)-1-[[(2S)-1-[[(2S,3S)-1-Amino-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-2-oxoethyl]-2,5-bis(benzylamino)pentanamide	Ki	5000.0 [1]
	(2S)-N-[2-[[(2S,3R)-1-[[(2S)-1-[[(2S,3R)-1-Amino-3-hydroxy-1-oxobutan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-2-oxoethyl]-2-(benzylamino)-5-[(4-methoxyphenyl)methylamino]pentanamide	Ki	305.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 13 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Oligosaccharyl transferase 48 kDa subunit Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/oligosaccharyl-transferase-48-kda-subunit-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 8). Quest Database™ Oligosaccharyl transferase 48 kDa subunit Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/oligosaccharyl-transferase-48-kda-subunit-inhibitors-ic50-ki.
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