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Opioid receptors; mu & delta Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
MorphineIC50309.0 [1]
NaltrexoneKi0.02 [1]
DamgoIC5076.1 [1]
DpdpeIC502.5 [1]
NaltrindoleKi31.5 [1]
DsletIC500.4 [1]
(2S)-1-[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]-N-[(2S)-1-[[(2R)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]pyrrolidine-2-carboxamideIC503333.0 [1]
(2S)-2-Amino-3-(4-hydroxyphenyl)-N-[(2R)-1-[[2-(4-methylpentan-2-ylamino)-2-oxoethyl]amino]-1-oxopropan-2-yl]propanamideIC501050.0 [1]
(2S)-2-Amino-3-(4-hydroxyphenyl)-N-[(2S)-1-[[2-(4-methylpentan-2-ylamino)-2-oxoethyl]amino]-1-oxopropan-2-yl]propanamideIC5050000.0 [1]
(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R,3R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxybutanoic acidIC500.15 [1]
(1S,2R,13R)-13,22-Dimethyl-2-[(E)-3-phenylprop-2-enyl]-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5,7,9,15,17,19(25)-heptaen-16-olKi3.5 [1]
2-Amino-3-(4-hydroxy-phenyl)-N-(1-{[(3-methyl-butylcarbamoyl)-methyl]-carbamoyl}-ethyl)-propionamideIC503410.0 [1]
2-[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]-3,4-dihydro-1H-isoquinoline-3-carboxylic acidIC5036.9 [1]
2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-2-methyl-N-[2-(4-methylpentan-2-ylamino)-2-oxoethyl]propanamideIC504720.0 [1]
(2S)-2-Amino-N-[(2R)-3-hydroxy-1-[[2-(4-methylpentan-2-ylamino)-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamideIC50990.0 [1]
(2S)-2-Amino-3-(4-hydroxyphenyl)-N-[(2R)-1-[[2-(4-methylpentan-2-ylamino)-2-oxoethyl]amino]-3-[(2-methylpropan-2-yl)oxy]-1-oxopropan-2-yl]propanamideIC50105.0 [1]
(2S)-2-Amino-N-[(2R)-1-[[2-[ethyl(4-methylpentan-2-yl)amino]-2-oxoethyl]amino]-1-oxopropan-2-yl]-3-(4-hydroxyphenyl)propanamideIC501800.0 [1]
(2R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-N-[2-(3-methylbutylamino)-2-oxoethyl]-4-methylsulfanylbutanamideIC50733.0 [1]
(2S)-2-[[2-[[(2R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]-methylamino]-N-(2-hydroxyethyl)-4-methylpentanamideIC503180.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxypropanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-4-methylpentanoic acidIC502.45 [1]
(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R,3R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-phenylpropanoyl]-methylamino]-4-methylpentanoyl]amino]-3-hydroxybutanoic acidIC501.33 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R,3R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoic acidIC500.25 [1]
(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2R,3R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-4-methylpentanoic acidIC500.41 [1]
(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[2-[[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]carbamoylamino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxybutanoic acidIC5038.0 [1]
(2R)-2-[5-[[2-[[(3R)-2-[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]acetyl]amino]pentanoylamino]-6-[5-[[2-[[(2R)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]pyrrolidine-2-carbonyl]amino]-3-phenylpropanoyl]amino]-3-naphthalen-1-ylpropanoyl]amino]acetyl]amino]pentanoylamino]hexanoic acidIC50153.0 [1]
(1S,10S,14S,18E)-18-Benzylidene-3-hydroxy-4-methoxy-17-methyl-17-azapentacyclo[7.5.3.210,14.01,10.02,7]nonadeca-2(7),3,5-trien-13-oneKi0.08 [1]
(1S,2R,13R)-13,22-Dimethyl-2-(3-methylbut-2-enyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5,7,9,15,17,19(25)-heptaen-16-olKi4.9 [1]
(1S,2S,13R)-19-Methoxy-24-methyl-26-propan-2-ylidene-4,24-diazaheptacyclo[12.7.3.22,13.01,13.03,11.05,10.016,21]hexacosa-3(11),5,7,9,16(21),17,19-heptaen-20-olKi3.2 [1]
(1S,10S,14S,18E)-3-Hydroxy-4-methoxy-17-methyl-18-(1-phenylethylidene)-17-azapentacyclo[7.5.3.210,14.01,10.02,7]nonadeca-2(7),3,5-trien-13-oneKi0.8 [1]
(1S,2S,13R,26E)-26-Benzylidene-19-methoxy-24-methyl-4,24-diazaheptacyclo[12.7.3.22,13.01,13.03,11.05,10.016,21]hexacosa-3(11),5,7,9,16(21),17,19-heptaen-20-olKi0.4 [1]
(1S,2S,13R,26E)-19-Methoxy-24-methyl-26-(1-phenylethylidene)-4,24-diazaheptacyclo[12.7.3.22,13.01,13.03,11.05,10.016,21]hexacosa-3(11),5,7,9,16(21),17,19-heptaen-20-olKi0.6 [1]
(1S,2S,13R,26E)-26-Ethylidene-19-methoxy-24-methyl-4,24-diazaheptacyclo[12.7.3.22,13.01,13.03,11.05,10.016,21]hexacosa-3(11),5,7,9,16(21),17,19-heptaen-20-olKi1.5 [1]
(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[(2R,3R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxybutanoyl]-methylamino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxybutanoic acidIC507.3 [1]
(2S,3R)-2-[[(1S)-1-[[(2S)-2-[[2-[[(2R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxypropanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-3-methylbutyl]amino]-3-hydroxybutanoic acidIC503.45 [1]
(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-Amino-3-phenylpropanoyl]amino]acetyl]amino]acetyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-4-methylsulfanylbutanoic acidIC5013.0 [1]
(2S,4R)-1-[(2S)-2-[[(2S)-2-[[2-[[(2R,3S)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxybutanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]-4-hydroxypyrrolidine-2-carboxylic acidIC501.1 [1]
(2S,3R)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2S,3S)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-3-hydroxypentanoyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxybutanoic acidIC500.05 [1]
Items per page: 1 - 10 of 37
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References

This online tool may be cited as follows

MLA

"Quest Database™ Opioid receptors; mu & delta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/opioid-receptors-mu-delta-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Opioid receptors; mu & delta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/opioid-receptors-mu-delta-inhibitors-ic50-ki.
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