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Opioid receptors; mu/kappa/delta Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
▲
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Standard Values (in nM)
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▼
MorphineIC5010.0 [1], 28.0 [2], 65.0 [3], 250.0 [4]
NaloxoneIC501.6 [1], 5.5 [2], 43.0 [3]
NaltrexoneIC503.8 [1], 5.7 [2]
BremazocineIC500.5 [1], 1.5 [2]
6beta-NaltrexolIC508.3 [1], 13.0 [2]
Methyl 2-[[(4R,4aS,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]oxymethyl]prop-2-enoateIC5011.0 [1], 11.1 [2], 12.0 [3]
Naloxone hydrochlorideIC504.3 [1], 5.5 [2]
Naltrexone hydrochlorideIC500.55 [1], 0.59 [2]
MeperidineIC50500.0 [1], 40000.0 [2]
EtorphineIC500.3 [1], 1.7 [2]
DpdpeIC50140.0 [1], 1000.0 [2]
(2S)-N-[(2S)-6-Amino-1-[[(2S)-1-[[(2S)-1,6-diamino-1-oxohexan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-1-oxohexan-2-yl]-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carboxamideIC500.24 [1], 1.7 [2]
(7R)-3-(Cyclopropylmethyl)-7-phenylmethoxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diolIC503.4 [1]
(1S,13R)-1,13-Dimethyl-10-(2,2,2-trifluoroethyl)-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-ol;methanesulfonic acidIC501700.0 [1], 2500.0 [2]
(1S,13R)-10-(2-Fluoroethyl)-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-ol;methanesulfonic acidIC5050.0 [1], 100.0 [2]
Ethyl 1-(2,2-difluoroethyl)-4-phenylpiperidine-4-carboxylate;hydrochlorideIC5085000.0 [1], 110000.0 [2]
Ethyl 1-(2-fluoroethyl)-4-phenylpiperidine-4-carboxylate;hydrochlorideIC5020000.0 [1], 64000.0 [2]
Ethyl 1-ethyl-4-phenylpiperidine-4-carboxylate;hydrochlorideIC505000.0 [1], 120000.0 [2]
Ethyl 4-phenyl-1-(2,2,2-trifluoroethyl)piperidine-4-carboxylate;hydrochlorideIC5010000.0 [1], 60000.0 [2]
(1S,13R)-10-Ethyl-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-ol;methanesulfonic acidIC50180.0 [1], 200.0 [2]
(1S,13R)-10-(2,2-Difluoroethyl)-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-ol;methanesulfonic acidIC501000.0 [1], 1150.0 [2]
(4R,4As,7R,7aR,12bS)-7-amino-3-prop-2-enyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diol;hydrochlorideIC5053.0 [1], 86.0 [2]
(4R,4As,7R,7aR,12bS)-7-amino-3-(cyclopropylmethyl)-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diol;hydrochlorideIC500.7 [1], 0.91 [2]
(4R,4As,7S,7aR,12bS)-7-amino-3-(cyclopropylmethyl)-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diol;hydrochlorideIC502.9 [1], 9.0 [2]
1-[4-[2-[(1R,9R,10R)-4-Hydroxy-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-17-yl]ethyl]phenyl]pyrrole-2,5-dioneIC505.3 [1], 57.0 [2]
(4R,4As,7S,7aR,12bS)-7-amino-3-prop-2-enyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diolIC50110.0 [1], 140.0 [2]
Morphine sulfateIC5024.0 [1]
DamgoIC5014.0 [1]
trans-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]-benzeneacetamideIC502.61 [1]
NalorphineIC5028.0 [1]
NorbinaltorphimineIC5011.0 [1]
NaltrindoleIC5047.0 [1]
OxymorphoneIC5090.0 [1]
DiprenorphineIC501.3 [1]
EthylketocyclazocineIC505.9 [1]
n-Methyl-2-phenyl-n-[(5r,7s,8s)-7-(pyrrolidin-1-yl)-1-oxaspiro[4.5]dec-8-yl]acetamideIC50139.0 [1]
DermorphinIC501.41 [1]
(1R,9S,13S)-1,13-Dimethyl-10-[[(2S)-oxolan-2-yl]methyl]-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-4-olIC501000.0 [1]
NaluzotanKi2000.0 [1]
Dynorphin A (1-11) amideIC507.5 [1]
Dynorphin A (swine)IC502.5 [1]
CID 11496610Ki550.0 [1]
10-(Cyclopropylmethyl)-4-ethoxy-1,13-dimethyl-10-azatricyclo[7.3.1.02,7]trideca-2(7),3,5-trien-8-oneIC500.6 [1]
(2S)-6-Amino-2-[[(2R)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]hexanoic acidIC500.22 [1]
(4R,12Bs)-3-(cyclopropylmethyl)-4a,9-dihydroxy-3'-methylidenespiro[2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-7,5'-oxolane]-2'-oneIC506.0 [1]
6-Benzyloxymethyl-5-[4-(4-chloro-benzylamino)-phenyl]-pyrimidine-2,4-diamineIC5033000.0 [1]
6a-NaltrexolIC508.3 [1]
3-(2-Cyclopropylmethyl-octahydro-isoquinolin-4a-yl)-phenolIC50150.0 [1]
(2S)-6-Amino-2-[[(2R)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-(benzylamino)-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]hexanoic acidIC50990.0 [1]
1,2-Dimethyl-4-phenyl-4-(propionyloxy)piperidineIC502000.0 [1]
1-[2-[1'-(2,2-Dimethylpropyl)spiro[2H-indole-3,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]ureaIC502700.0 [1]
Methyl 2-[[(4R,4aS,7aR,12bS)-4a-hydroxy-3-methyl-7-oxo-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinolin-9-yl]oxymethyl]prop-2-enoateIC50110.0 [1]
(3S,6S,9S,12S,15R,20R,23S)-15-[[(2S)-2-[[2-[[2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-6-[(2S)-butan-2-yl]-3,9,12-tris[3-(diaminomethylideneamino)propyl]-2,5,8,11,14,22-hexaoxo-17,18-dithia-1,4,7,10,13,21-hexazabicyclo[21.3.0]hexacosane-20-carboxamideIC501080.0 [1]
4-(4-Bromophenyl)-4-(dimethylamino)-1-(2-phenylethyl)cyclohexan-1-ol;hydrochlorideIC500.8 [1]
Methyl 2-[[(4R,4aS,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a,7-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-9-yl]oxymethyl]prop-2-enoateIC5027.0 [1]
Methyl 2-[[(1R,2S,6R,14R,15R,19R)-19-[(2R)-2-hydroxypentan-2-yl]-15-methoxy-5-methyl-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11,16-tetraen-11-yl]oxymethyl]prop-2-enoateIC502.4 [1]
Methyl 2-[[(1S,2S,7S,8S,12R,20R,24R,32R)-11,33-bis(cyclopropylmethyl)-2,7-dihydroxy-27-(2-methoxycarbonylprop-2-enoxy)-19,25-dioxa-11,22,33-triazaundecacyclo[24.9.1.18,14.01,24.02,32.04,23.05,21.07,12.08,20.030,36.018,37]heptatriaconta-4(23),5(21),14(37),15,17,26,28,30(36)-octaen-17-yl]oxymethyl]prop-2-enoateIC5022.0 [1]
Methyl 2-[[(4R,4aS,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a-hydroxy-9-(2-methoxycarbonylprop-2-enoxy)-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]oxymethyl]prop-2-enoateIC5014.0 [1]
Methyl 2-[[(4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a-hydroxy-7-oxo-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinolin-9-yl]oxymethyl]prop-2-enoateIC5010.3 [1]
Methyl 3-[[(4R,4aS,7aR,12bS)-3-(cyclopropylmethyl)-4a-hydroxy-7-oxo-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinolin-9-yl]oxy]-2-methylpropanoateIC503000.0 [1]
Methyl 2-[[(1S,2S,6R,14R,15R,16R)-5-(cyclopropylmethyl)-16-(2-hydroxypropan-2-yl)-15-methoxy-13-oxa-5-azahexacyclo[13.2.2.12,8.01,6.02,14.012,20]icosa-8(20),9,11-trien-11-yl]oxymethyl]prop-2-enoateIC502.2 [1]
Methyl 2-[[(1S,2S,13R,21R)-22-(cyclopropylmethyl)-2-hydroxy-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5,7,9,15,17,19(25)-heptaen-16-yl]oxymethyl]prop-2-enoateIC5080.0 [1]
1-[4-[4-[2-Tert-butyl-6-(trifluoromethyl)pyrimidin-4-yl]piperazin-1-yl]butyl]-3,4-dihydro-1-benzazepine-2,5-dioneIC5010000.0 [1]
2-[[(2S)-2-[[(2R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-4-methylsulfinylbutanoyl]amino]-3-phenylpropanoyl]amino]acetic acidIC5016.7 [1]
(2R)-2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]-N-[(2S)-1-[(2-amino-2-oxoethyl)amino]-1-oxo-3-phenylpropan-2-yl]-4-methylsulfinylbutanamideIC5013.6 [1]
4-[[(4R,4As,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-4-oxobutanoic acidIC50144.0 [1]
(Z)-4-[[(4R,4As,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-4-oxobut-2-enoic acidIC5039.0 [1]
(E)-4-[[(4R,4As,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-4-oxobut-2-enoic acidIC50130.0 [1]
2-[2-[[(4R,4As,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethoxy]acetic acidIC5027.0 [1]
4-[[(4R,4As,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-3-amino-4-oxobutanoic acidIC5031.0 [1]
(3S,6R,9S,12S,15R,20R,23S)-15-[[(2S)-2-[[2-[[2-[[(2S)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-3,9,12-tris[3-(diaminomethylideneamino)propyl]-6-methyl-2,5,8,11,14,22-hexaoxo-17,18-dithia-1,4,7,10,13,21-hexazabicyclo[21.3.0]hexacosane-20-carboxamideIC504406.0 [1]
(4R,4As,7R,7aR,12bS)-3-(cyclopropylmethyl)-7-[[(2R)-oxiran-2-yl]methoxy]-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diolIC5011.0 [1]
(4R,4As,7R,7aR,12bS)-3-(cyclopropylmethyl)-7-[[(2S)-oxiran-2-yl]methoxy]-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diolIC5012.0 [1]
[(4R,4As,7R,7aR,12bS)-3-(cyclopropylmethyl)-9-hydroxy-7-[[(2R)-4-methylidene-5-oxooxolan-2-yl]methoxy]-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-4a-yl] acetateIC5015.0 [1]
[(4R,4As,7R,7aR,12bS)-3-(cyclopropylmethyl)-9-hydroxy-7-[[(2S)-4-methylidene-5-oxooxolan-2-yl]methoxy]-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-4a-yl] acetateIC5014.0 [1]
(5R)-5-[[(4R,4As,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]oxymethyl]-3-methylideneoxolan-2-oneIC5019.0 [1]
(5S)-5-[[(4R,4As,7R,7aR,12bS)-3-(cyclopropylmethyl)-4a,9-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]oxymethyl]-3-methylideneoxolan-2-oneIC5018.0 [1]
N-[1-(6,7-Dihydro-5H-cyclopenta[f][1,3]benzodioxol-7-yl)piperidin-4-yl]-6-fluoro-4-oxochromene-2-carboxamideIC5010000.0 [1]
(3S,6R,11R,14S,17S,20S)-17-(4-Aminobutyl)-6-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-2,5,13,16,19-pentaoxo-8,9-dithia-1,4,12,15,18-pentazabicyclo[18.3.0]tricosane-11-carboxamideIC501.3 [1]
(3S,6S,11R,14S,17S,20S)-17-(4-Aminobutyl)-6-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-2,5,13,16,19-pentaoxo-8,9-dithia-1,4,12,15,18-pentazabicyclo[18.3.0]tricosane-11-carboxamideIC502.27 [1]
(3S,6S,11S,14S,17S,20S)-17-(4-Aminobutyl)-6-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-amino-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-2,5,13,16,19-pentaoxo-8,9-dithia-1,4,12,15,18-pentazabicyclo[18.3.0]tricosane-11-carboxamideIC501.75 [1]
(2S)-6-Amino-2-[[(2R)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-[bis(prop-2-enyl)amino]-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]hexanoic acidIC50687.0 [1]
[(4S)-1,2-Dimethyl-4-phenylpiperidin-4-yl] propanoateIC5011000.0 [1]
beta-FuoxymorphineIC5022.0 [1]
2-[[(2R)-2-[[2-[[(2S)-2-[[(2R)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]-methylamino]-3-phenylpropanoyl]amino]acetic acidIC5028.0 [1]
(2R)-2-[[(2R)-2-[[2-[[(2S)-2-[[(2R)-2-Amino-3-(4-hydroxyphenyl)propanoyl]amino]propanoyl]amino]acetyl]amino]-4-methylsulfanylbutanoyl]amino]-4-methylpentanoic acidIC5021.0 [1]
N-[(4As,7R,7aR)-3-(cyclopropylmethyl)-4a,9-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]-2-[bis(2-chloroethyl)amino]acetamideIC503.8 [1]
10-(Cyclopropylmethyl)-4-ethoxy-1,12-dimethyl-10-azatricyclo[7.2.1.02,7]dodeca-2(7),3,5-trien-8-oneIC500.07 [1]
1-(2-Adamantyl)-2-[[3-(cyclopropylmethyl)-4a,9-dihydroxy-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]oxy]ethanoneIC5013.0 [1]
(2S)-6-Amino-2-[[(2R)-1-[(2S)-5-(diaminomethylideneamino)-2-[[(2S,3S)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-3-(4-hydroxyphenyl)-2-(prop-2-enylamino)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]pentanoyl]amino]pentanoyl]amino]-3-methylpentanoyl]amino]pentanoyl]pyrrolidine-2-carbonyl]amino]hexanoic acidIC5018.3 [1]
(2S)-6-Amino-2-[[(2R)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-(cyclopropylmethylamino)-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-methylpentanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]amino]hexanoic acidIC502.16 [1]
3-[(8Ar)-2-(cyclopropylmethyl)-1,3,4,5,8,8a-hexahydroisoquinolin-4a-yl]phenolIC5090.0 [1]
3-[(8Ar)-2-(cyclobutylmethyl)-1,3,4,5,8,8a-hexahydroisoquinolin-4a-yl]phenolIC5060.0 [1]
3-[(8Ar)-2-methyl-1,3,4,5,8,8a-hexahydroisoquinolin-4a-yl]phenolIC50130.0 [1]
(8Ar)-2-(cyclopropylmethyl)-4a-(3-hydroxyphenyl)-3,4,5,7,8,8a-hexahydro-1H-isoquinolin-6-oneIC50120.0 [1]
3-[(8Ar)-6-methylidene-2-prop-2-enyl-3,4,5,7,8,8a-hexahydro-1H-isoquinolin-4a-yl]phenolIC50140.0 [1]
3-[(8Ar)-2-(cyclopropylmethyl)-6-methylidene-3,4,5,7,8,8a-hexahydro-1H-isoquinolin-4a-yl]phenolIC5015.0 [1]
3-[(8Ar)-2-methyl-6-methylidene-3,4,5,7,8,8a-hexahydro-1H-isoquinolin-4a-yl]phenolIC5060.0 [1]
(4As,7R,7aR)-3-(cyclopropylmethyl)-7-[(4-isothiocyanatophenyl)methoxy]-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diolIC5022.0 [1]
(4As,7R,7aR)-3-(cyclopropylmethyl)-7-[[3-(isothiocyanatomethyl)phenyl]methoxy]-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinoline-4a,9-diolIC5024.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Opioid receptors; mu/kappa/delta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 8 May. 2024, https://www.aatbio.com/data-sets/opioid-receptors-mu-kappa-delta-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 8). Quest Database™ Opioid receptors; mu/kappa/delta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/opioid-receptors-mu-kappa-delta-inhibitors-ic50-ki.
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