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Opioid receptors; mu/kappa/delta Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
MorphineIC5010.0 [1], 28.0 [2], 65.0 [3], 250.0 [4]
NaloxoneIC501.6 [1], 5.5 [2], 43.0 [3]
NaltrexoneIC503.8 [1], 5.7 [2]
BremazocineIC500.5 [1], 1.5 [2]
6beta-NaltrexolIC508.3 [1], 13.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseOpioid receptors; mu/kappa/delta Inhibitors (IC50, Ki)." AAT Bioquest, Inc.31 Dec2025https://www.aatbio.com/data-sets/opioid-receptors-mu-kappa-delta-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 31). Quest DatabaseOpioid receptors; mu/kappa/delta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/opioid-receptors-mu-kappa-delta-inhibitors-ic50-ki.
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