Opioid receptors; mu & kappa Inhibitors (IC50, Ki)

Name: Opioid receptors; mu & kappa Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Naloxone	IC50	9.0 ^[1], 127.0 ^[2]
	Naltrexone	IC50	2.6 ^[1], 12.0 ^[2]
	trans-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]-benzeneacetamide	IC50	5.0 ^[1], 3100.0 ^[2]
	Levallorphan	IC50	0.67 ^[1], 2.6 ^[2]
	Cyprodime	IC50	170.0 ^[1], 628.0 ^[2]
	N-[(4R,4As,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]acetamide	IC50	66.8 ^[1]
	N,N'-Bis[(4R,4aS,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]butanediamide	IC50	30.2 ^[1]
	N,N'-Bis[2-[[2-[[2-[[(4R,4aS,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]amino]-2-oxoethyl]butanediamide	IC50	25.1 ^[1]
	N,N'-Bis[2-[[2-[[(4R,4aS,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]butanediamide	IC50	3.9 ^[1]
	N,N'-Bis[2-[[(4R,4aS,7S,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]butanediamide	IC50	22.0 ^[1]
	N,N'-Bis[(4R,4aR,7R,7aS,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]butanediamide	IC50	15.7 ^[1]
	N,N'-Bis[2-[[(4R,4aR,7R,7aS,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]butanediamide	IC50	19.2 ^[1]
	N,N'-Bis[2-[[2-[[(4R,4aR,7R,7aS,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]butanediamide	IC50	6.3 ^[1]
	N-[(4R,4As,7R,7aR,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]acetamide	IC50	45.9 ^[1]
	N,N'-Bis[2-[[2-[[2-[[(4R,4aR,7R,7aS,12bS)-4a,9-dihydroxy-3-methyl-1,2,4,5,6,7,7a,13-octahydro-4,12-methanobenzofuro[3,2-e]isoquinolin-7-yl]amino]-2-oxoethyl]amino]-2-oxoethyl]amino]-2-oxoethyl]butanediamide	IC50	12.6 ^[1]

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References

This online tool may be cited as follows

MLA	"Quest Database™ Opioid receptors; mu & kappa Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/opioid-receptors-mu-kappa-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Opioid receptors; mu & kappa Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/opioid-receptors-mu-kappa-inhibitors-ic50-ki.
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Opioid receptors; mu & kappa Inhibitors (IC50, Ki)

References

This online tool may be cited as follows

MLA

APA