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ORAI1/STIM1 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
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▼
5-(5-Chloro-2-methyl-1,3-benzoxazol-6-yl)-N-(2-chlorophenyl)thiophene-2-carboxamideIC50600.0 [1]
2-Fluoro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]thiophen-2-yl]benzamideIC50600.0 [1]
2,6-Difluoro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]thiophen-2-yl]benzamideIC50600.0 [1]
3,5-Difluoro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]thiophen-2-yl]pyridine-4-carboxamideIC50600.0 [1]
N-[5-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)thiophen-2-yl]-2-fluorobenzamideIC501200.0 [1]
N-[5-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)thiophen-2-yl]-2,6-difluorobenzamideIC501200.0 [1]
5-(1,5-Dimethylindazol-6-yl)-N-(2-fluorophenyl)thiophene-2-carboxamideIC50600.0 [1]
N-(2-Chlorophenyl)-5-(2,5-dimethylindazol-6-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-(2,5-dimethylindazol-6-yl)thiophene-2-carboxamideIC50600.0 [1]
2-Chloro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
2,6-Difluoro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
4-Chloro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
2-Fluoro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
3-Fluoro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-2-yl]pyridine-4-carboxamideIC50600.0 [1]
3,5-Difluoro-N-[5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-2-yl]pyridine-4-carboxamideIC501200.0 [1]
2-Chloro-N-[5-[2-ethyl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
2-Chloro-N-[5-[2-propan-2-yl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-2-yl]benzamideIC501200.0 [1]
2-Fluoro-N-[5-(2-methyl-5-phenylpyrazol-3-yl)-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
2-Fluoro-N-[5-[5-(2-fluorophenyl)-2-methylpyrazol-3-yl]-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
2,6-Difluoro-N-[5-(6-methyl-1,3-benzothiazol-5-yl)-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
2-Chloro-N-[5-(5-chloro-2-methyl-1,3-benzoxazol-6-yl)-1,3-thiazol-2-yl]benzamideIC50600.0 [1]
2-Chloro-N-[5-(1-methylindol-2-yl)-1,3-thiazol-2-yl]benzamideIC501200.0 [1]
2-Chloro-N-[5-[2-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)pyrazol-3-yl]-1,3-thiazol-2-yl]benzamideIC501200.0 [1]
N-[5-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)-1,3-thiazol-2-yl]-3,5-difluoropyridine-4-carboxamideIC501200.0 [1]
N-[5-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)-1,3-thiazol-2-yl]-3-fluoropyridine-4-carboxamideIC50600.0 [1]
N-[5-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)-1,3-thiazol-2-yl]-2,6-difluorobenzamideIC501200.0 [1]
N-[5-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)-1,3-thiazol-2-yl]-2-fluorobenzamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-(6-methyl-1,3-benzothiazol-5-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(2-Chlorophenyl)-5-(6-methyl-1,3-benzothiazol-5-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(2-Fluorophenyl)-5-(6-methyl-1,3-benzothiazol-5-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-[5-(2-fluorophenyl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
5-(5-Chloro-1,3-benzothiazol-6-yl)-N-(2-chlorophenyl)thiophene-2-carboxamideIC50600.0 [1]
5-(5-Chloro-1,3-benzothiazol-6-yl)-N-(2,6-difluorophenyl)thiophene-2-carboxamideIC50600.0 [1]
N-(2-Fluorophenyl)-5-[2-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-[2-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-(3,5-dimethyl-1,2-benzoxazol-6-yl)thiophene-2-carboxamideIC50600.0 [1]
5-(5-Chloro-1,3-benzothiazol-6-yl)-N-(2-fluorophenyl)thiophene-2-carboxamideIC50600.0 [1]
5-(3,5-Dimethyl-1,2-benzoxazol-6-yl)-N-(2-fluorophenyl)thiophene-2-carboxamideIC50600.0 [1]
5-(2,5-Dimethylindazol-6-yl)-N-(2-fluorophenyl)thiophene-2-carboxamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-[5-(furan-2-yl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
5-(5-Chloro-2-methyl-1,3-benzoxazol-6-yl)-N-(2-fluorophenyl)thiophene-2-carboxamideIC50600.0 [1]
5-(5-Chloro-2-methyl-1,3-benzoxazol-6-yl)-N-(2,6-difluorophenyl)thiophene-2-carboxamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-(2-methyl-5-phenylpyrazol-3-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-[2-methyl-5-(1,3-thiazol-2-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(3-Fluoropyridin-2-yl)-5-[5-(furan-2-yl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(2,6-Difluorophenyl)-5-(2-methyl-5-thiophen-2-ylpyrazol-3-yl)thiophene-2-carboxamideIC501200.0 [1]
5-[5-(2-Fluorophenyl)-2-methylpyrazol-3-yl]-N-(3-fluoropyridin-2-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(2-Chlorophenyl)-5-(2-methyl-5-thiophen-2-ylpyrazol-3-yl)thiophene-2-carboxamideIC501200.0 [1]
N-(2-Fluorophenyl)-5-[5-(furan-2-yl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(2-Fluorophenyl)-5-[2-methyl-5-(1,3-thiazol-2-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(2-Chlorophenyl)-5-[5-(furan-2-yl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(3-Fluoropyridin-2-yl)-5-[2-methyl-5-(1,3-thiazol-2-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(2-Chlorophenyl)-5-[2-methyl-5-(1,3-thiazol-2-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(2-Fluorophenyl)-5-(2-methyl-5-phenylpyrazol-3-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(2-Chlorophenyl)-5-(2-methyl-5-phenylpyrazol-3-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(3-Fluoropyridin-2-yl)-5-(2-methyl-5-phenylpyrazol-3-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(2-Chlorophenyl)-5-[5-(2-fluorophenyl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
4-Amino-N-(2-fluorophenyl)-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]thiophene-2-carboxamideIC501200.0 [1]
4-Amino-N-(2-chlorophenyl)-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]thiophene-2-carboxamideIC501200.0 [1]
4-Amino-N-(2,6-difluorophenyl)-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]thiophene-2-carboxamideIC501200.0 [1]
2-Chloro-N-[2-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1,3-thiazol-5-yl]benzamideIC501200.0 [1]
N-(3,5-Difluoropyridin-4-yl)-5-[5-(2-fluorophenyl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(5-Chloro-3-fluoropyridin-2-yl)-5-[5-(2-fluorophenyl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
5-[5-(2-Fluorophenyl)-2-methylpyrazol-3-yl]-N-(3-fluoropyridin-4-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(3,5-Difluoropyridin-4-yl)-5-(2-methyl-5-phenylpyrazol-3-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(3-Fluoropyridin-4-yl)-5-(2-methyl-5-phenylpyrazol-3-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(5-Chloro-3-fluoropyridin-2-yl)-5-(2-methyl-5-phenylpyrazol-3-yl)thiophene-2-carboxamideIC50600.0 [1]
N-(3-Fluoropyridin-4-yl)-5-[2-methyl-5-(1,3-thiazol-2-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(3,5-Difluoropyridin-4-yl)-5-[2-methyl-5-(1,3-thiazol-2-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(5-Chloro-3-fluoropyridin-2-yl)-5-[2-methyl-5-(1,3-thiazol-2-yl)pyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(3,5-Difluoropyridin-4-yl)-5-[5-(furan-2-yl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(3-Fluoropyridin-4-yl)-5-[5-(furan-2-yl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-(5-Chloro-3-fluoropyridin-2-yl)-5-[5-(furan-2-yl)-2-methylpyrazol-3-yl]thiophene-2-carboxamideIC50600.0 [1]
N-[(2,6-Difluorophenyl)methyl]-5-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)pyridin-2-amineIC50600.0 [1]
N-[(2-Fluoro-6-methylphenyl)methyl]-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]pyridin-2-amineIC50600.0 [1]
N-[(2-Fluorophenyl)methyl]-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]pyrimidin-2-amineIC50600.0 [1]
5-(6-Chloro-2,2-difluoro-1,3-benzodioxol-5-yl)-N-[(2-chlorophenyl)methyl]pyridin-2-amineIC501200.0 [1]
N-[(2,6-Difluorophenyl)methyl]-5-(6-methoxy-4-methylpyridin-3-yl)pyrimidin-2-amineIC50600.0 [1]
N-[(2,6-Difluoro-4-methoxyphenyl)methyl]-5-(2,2-difluoro-6-methyl-1,3-benzodioxol-5-yl)pyrimidin-2-amineIC50600.0 [1]
N-[(3,5-Difluoropyridin-4-yl)methyl]-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]pyridin-2-amineIC50600.0 [1]
5-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)-N-[(2,6-difluorophenyl)methyl]pyridin-2-amineIC50600.0 [1]
5-(6-Chloro-2,2-difluoro-1,3-benzodioxol-5-yl)-N-[(2,6-difluorophenyl)methyl]pyridin-2-amineIC50600.0 [1]
6-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)-N-[(2,6-difluorophenyl)methyl]pyridin-3-amineIC50600.0 [1]
5-(6-Chloro-2,3-dihydro-1,4-benzodioxin-7-yl)-N-[(2,6-difluorophenyl)methyl]pyridin-2-amineIC501200.0 [1]
N-[(2,6-Difluoro-4-methoxyphenyl)methyl]-5-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-2-amineIC50600.0 [1]
N-[(2,6-Difluorophenyl)methyl]-5-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-2-amineIC50600.0 [1]
5-(6-Chloro-2,2-difluoro-1,3-benzodioxol-5-yl)-N-[(2-chloro-3-fluorophenyl)methyl]pyridin-2-amineIC501200.0 [1]
N-[(2,4-Difluorophenyl)methyl]-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]pyridin-2-amineIC50600.0 [1]
N-[(2,6-Difluorophenyl)methyl]-5-[2-(trifluoromethyl)phenoxy]pyrimidin-2-amineIC50600.0 [1]
N-[(3,5-Difluoropyridin-4-yl)methyl]-5-[5-methyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-2-amineIC50600.0 [1]
N-[(2,6-Difluorophenyl)methyl]-5-[2-methyl-4-(trifluoromethyl)imidazol-1-yl]pyridin-2-amineIC50600.0 [1]
N-[(2-Fluorophenyl)methyl]-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]pyridin-2-amineIC50600.0 [1]
N-[(2,6-Difluorophenyl)methyl]-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]pyridin-2-amineIC50600.0 [1]
N-[(2,6-Difluorophenyl)methyl]-5-(6-methyl-2,3-dihydro-1H-inden-5-yl)pyridin-2-amineIC50600.0 [1]
2-[(2-Chloro-6-fluorophenyl)methoxy]-5-(2,2-difluoro-6-methyl-1,3-benzodioxol-5-yl)pyrimidineIC501200.0 [1]
5-(6-Chloro-2,2-difluoro-1,3-benzodioxol-5-yl)-N-[(2-chloro-4-fluorophenyl)methyl]pyridin-2-amineIC501200.0 [1]
5-(6-Chloro-2,2-difluoro-1,3-benzodioxol-5-yl)-N-[(3-fluorophenyl)methyl]pyridin-2-amineIC50600.0 [1]
5-(6-Chloro-2,2-difluoro-1,3-benzodioxol-5-yl)-N-[(2-methoxyphenyl)methyl]pyridin-2-amineIC501200.0 [1]
5-(2,2-Difluoro-6-methyl-1,3-benzodioxol-5-yl)-N-[(2-methylphenyl)methyl]pyridin-2-amineIC50600.0 [1]
N-[(2-Chlorophenyl)methyl]-5-(2,2-difluoro-6-methyl-1,3-benzodioxol-5-yl)pyridin-2-amineIC501200.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ ORAI1/STIM1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/orai1-stim1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ ORAI1/STIM1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/orai1-stim1-inhibitors-ic50-ki.
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