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Oxytocin receptor Inhibitors (IC50, Ki)
StructureCompound NameStandard TypeStandard Values (in nM)
OxytocinIC502.7 [1]
4-[(3,5-Dihydroxyphenyl)methyl]-N-[[2-methyl-4-(1-methyl-4,10-dihydropyrazolo[4,3-c][1,5]benzodiazepine-5-carbonyl)phenyl]methyl]piperazine-1-carboxamideIC5010000.0 [1]
AtosibanIC5059.0 [1], 372.0 [2]
AtosibanKi11.0 [1], 27.0 [2], 32.0 [3], 39.81 [4], 397.0 [5]
CligosibanIC5063.0 [1], 600.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabaseOxytocin receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc.11 Oct2025https://www.aatbio.com/data-sets/oxytocin-receptor-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025October 11). Quest DatabaseOxytocin receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/oxytocin-receptor-inhibitors-ic50-ki.
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