 | Verapamil | IC50 | 6300.0 [1] |
| Verapamil | Ki | 1750.0 [1], 3000.0 [2], 15100.0 [3] |
 | Cyclosporin A | IC50 | 1400.0 [1] |
| Cyclosporin A | Ki | 20.0 [1], 1800.0 [2], 2180.0 [3] |
 | Hernandezine | IC50 | 204.61 [1] |
| Hernandezine | Ki | 20.0 [1] |
 | Tariquidar | IC50 | 210.0 [1] |
 | 2-(1H-Benzimidazol-2-ylmethylsulfanyl)-5-phenyl-1H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one | IC50 | 830.0 [1] |
 | Vinblastine | IC50 | 29000.0 [1] |
| Vinblastine | Ki | 2100.0 [1], 36500.0 [2], 140000.0 [3] |
 | Reserpine | IC50 | 3235.94 [1] |
| Reserpine | Ki | 100.0 [1], 970.0 [2], 2310.0 [3], 11500.0 [4], 12200.0 [5] |
 | Nicardipine | IC50 | 5128.61 [1] |
 | Quinidine | IC50 | 5600.0 [1] |
| Quinidine | Ki | 430.0 [1], 1500.0 [2], 2600.0 [3], 5000.0 [4], 8590.0 [5] |
 | Ketoconazole | IC50 | 5600.0 [1] |
| Ketoconazole | Ki | 1200.0 [1], 5270.0 [2], 24900.0 [3] |
 | N-(4-Tert-butylphenyl)-2-[[1-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]triazol-4-yl]methoxy]benzamide | IC50 | 10320.0 [1] |
 | 5-Hydroxy-3,9-bis(3-methylphenyl)pyrano[2,3-h]chromene-4,10-dione | IC50 | 59.6 [1] |
 | Quinine | IC50 | 112400.0 [1] |
| Quinine | Ki | 12000.0 [1] |
 | Progesterone | IC50 | 88100.0 [1] |
 | Clarithromycin | IC50 | 23800.0 [1] |
 | Emetine | IC50 | 35100.0 [1] |
 | Valspodar | IC50 | 22.2 [1], 110.0 [2], 291.0 [3], 501.19 [4], 1060.0 [5] |
| Valspodar | Ki | 134.0 [1], 1300.0 [2] |
 | 2-Benzamido-N-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]benzamide | IC50 | 512.86 [1] |
 | Diltiazem | IC50 | 49000.0 [1] |
 | Terfenadine | IC50 | 1400.0 [1] |
 | N-[2-[[4-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]phenyl]quinoline-3-carboxamide | IC50 | 354.81 [1] |
 | N-[2-[[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]phenyl]-3,4-dimethoxybenzamide | IC50 | 331.13 [1] |
 | 5-Hydroxy-3,9-bis(4-methoxyphenyl)pyrano[2,3-h]chromene-4,10-dione | IC50 | 499.76 [1] |
 | 3,9-Bis(3,4-dimethoxyphenyl)-5-hydroxypyrano[2,3-h]chromene-4,10-dione | IC50 | 84.95 [1] |
 | Paclitaxel | IC50 | 2596.0 [1], 2600.0 [2], 53900.0 [3], 54000.0 [4], 70200.0 [5] |
 | Etoposide | IC50 | 50000.0 [1] |
| Etoposide | Ki | 276000.0 [1], 768000.0 [2] |
 | Tamoxifen | IC50 | 6400.0 [1], 12100.0 [2], 29000.0 [3], 31400.0 [4] |
| Tamoxifen | Ki | 100.0 [1] |
 | Erythromycin | IC50 | 43000.0 [1], 50000.0 [2] |
| Erythromycin | Ki | 37790.0 [1], 1000000.0 [2] |
 | Simvastatin | IC50 | 9000.0 [1], 10000.0 [2], 26100.0 [3], 46000.0 [4], 56800.0 [5] |
 | Ritonavir | IC50 | 1500.0 [1], 3800.0 [2], 12000.0 [3], 15700.0 [4] |
 | Lovastatin | IC50 | 10000.0 [1], 26000.0 [2], 32700.0 [3], 67000.0 [4], 114400.0 [5] |
 | Sporanox | IC50 | 30.0 [1], 1700.0 [2], 2100.0 [3], 2400.0 [4] |
 | Miconazole | IC50 | 2000.0 [1], 3500.0 [2] |
| Miconazole | Ki | 26360.0 [1], 55500.0 [2] |
 | Clotrimazole | IC50 | 1300.0 [1], 6700.0 [2] |
| Clotrimazole | Ki | 29920.0 [1], 44000.0 [2] |
 | Saquinavir | IC50 | 1600.0 [1], 6500.0 [2], 12000.0 [3], 100000.0 [4] |
 | Mibefradil | IC50 | 1200.0 [1], 1500.0 [2], 1600.0 [3], 1800.0 [4] |
 | Troleandomycin | IC50 | 68300.0 [1], 78200.0 [2], 86300.0 [3] |
| Troleandomycin | Ki | 87640.0 [1], 483300.0 [2] |
 | Elacridar | IC50 | 72.44 [1], 193.0 [2], 2000.0 [3] |
 | Zosuquidar | IC50 | 20.0 [1], 24.0 [2], 58.88 [3], 80.0 [4], 180.0 [5] |
 | Imatinib | IC50 | 7244.36 [1], 12589.25 [2], 15135612484.36 [3] |
 | Dexverapamil | IC50 | 2370.0 [1], 2580.0 [2], 5520.0 [3] |
| Dexverapamil | Ki | 1600.0 [1] |
 | Amiodarone | IC50 | 22500.0 [1], 45600.0 [2] |
| Amiodarone | Ki | 3200.0 [1], 5780.0 [2] |
 | Trifluoperazine | IC50 | 6300.0 [1], 7200.0 [2], 10900.0 [3] |
| Trifluoperazine | Ki | 6500.0 [1] |
 | Nelfinavir | IC50 | 350.0 [1], 1400.0 [2], 3400.0 [3] |
 | N-[2-[[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]carbamoyl]phenyl]quinoline-3-carboxamide | IC50 | 87.1 [1], 165.96 [2], 239.88 [3] |
 | 2-Amino-N-(4-(2-(3,4-dihydroisoquinolin-2(1H)-yl)ethyl)phenyl)benzamide | IC50 | 9332.54 [1], 9549.93 [2], 9900.0 [3] |
 | N-(4-(2-(3,4-Dihydroisoquinolin-2(1H)-yl)ethyl)phenyl)-2-nitrobenzamide | IC50 | 12302.69 [1], 13489.63 [2], 14000.0 [3] |
 | N-(4-(2-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)phenyl)-2-nitrobenzamide | IC50 | 4786.3 [1], 5400.0 [2], 5495.41 [3] |
 | 2-Amino-N-(4-(2-(6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)phenyl)benzamide | IC50 | 8500.0 [1], 9120.11 [2], 11220.18 [3] |
 | 4-Amino-N-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]benzamide | IC50 | 4073.8 [1], 4400.0 [2], 7079.46 [3] |
 | N-(4-(2-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)ethyl)phenyl)-4-nitrobenzamide | IC50 | 1096.48 [1], 1380.38 [2], 1400.0 [3] |
 | [4-[Methyl-[4-[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]oxycyclohexyl]amino]cyclohexyl] 3,4,5-trimethoxybenzoate | IC50 | 12.0 [1], 30.0 [2], 92.0 [3], 320.0 [4] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]quinoline-3-carboxamide | IC50 | 144.54 [1], 570.0 [2], 645.65 [3] |
 | 4-Amino-N-[4-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]benzamide | IC50 | 4168.69 [1], 12000.0 [2], 13489.63 [3] |
 | N-[4-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]-4-nitrobenzamide | IC50 | 4466.84 [1], 5011.87 [2], 5600.0 [3] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]quinoline-6-carboxamide | IC50 | 650.0 [1], 724.44 [2], 741.31 [3] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]pyridine-3-carboxamide | IC50 | 3162.28 [1], 4168.69 [2], 4800.0 [3] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]quinoxaline-2-carboxamide | IC50 | 208.93 [1], 470.0 [2], 489.78 [3] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]naphthalene-2-carboxamide | IC50 | 630.0 [1], 776.25 [2] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]naphthalene-1-carboxamide | IC50 | 1400.0 [1], 1412.54 [2], 1862.09 [3] |
 | 4-Bromo-N-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]benzamide | IC50 | 2400.0 [1], 2454.71 [2], 3162.28 [3] |
 | 3-Bromo-N-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]benzamide | IC50 | 1800.0 [1], 2290.87 [2], 3235.94 [3] |
 | 2-Bromo-N-[4-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]benzamide | IC50 | 3300.0 [1], 3467.37 [2], 4265.8 [3] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]-4,5-dimethoxy-2-nitrobenzamide | IC50 | 4897.79 [1], 6165.95 [2], 13000.0 [3] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]quinoline-4-carboxamide | IC50 | 2238.72 [1], 2818.38 [2], 4700.0 [3] |
 | N-[4-[2-(3,4-Dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]quinoline-3-carboxamide | IC50 | 416.87 [1], 430.0 [2], 524.81 [3] |
 | N-[4-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]phenyl]-3,4-dimethoxybenzamide | IC50 | 4168.69 [1], 4200.0 [2], 5370.32 [3] |
 | [4-[Methyl-[4-[3-(3,4,5-trimethoxyphenyl)prop-2-ynoyloxy]cyclohexyl]amino]cyclohexyl] 3,4,5-trimethoxybenzoate | IC50 | 20.0 [1], 70.0 [2], 80.0 [3] |
 | [4-[Methyl-[4-[3-(3,4,5-trimethoxyphenyl)propanoyloxy]cyclohexyl]amino]cyclohexyl] 3,4,5-trimethoxybenzoate | IC50 | 350.0 [1], 610.0 [2], 630.0 [3], 1100.0 [4] |
 | [4-[[4-[2,2-Bis(4-methoxyphenyl)acetyl]oxycyclohexyl]-methylamino]cyclohexyl] 3-(3,4,5-trimethoxyphenyl)prop-2-ynoate | IC50 | 20.0 [1], 120.0 [2], 130.0 [3], 140.0 [4] |
 | [4-[Methyl-[4-[3-(3,4,5-trimethoxyphenyl)prop-2-ynoyloxy]cyclohexyl]amino]cyclohexyl] 9H-fluorene-9-carboxylate | IC50 | 50.0 [1], 120.0 [2], 290.0 [3], 500.0 [4] |
 | [4-[Methyl-[4-[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]oxycyclohexyl]amino]cyclohexyl] 4-cyano-4-(3,4-dimethoxyphenyl)-5-methylhexanoate | IC50 | 80.0 [1], 140.0 [2], 150.0 [3], 240.0 [4] |
 | [4-[Methyl-[4-[(E)-3-(3,4,5-trimethoxyphenyl)prop-2-enoyl]oxycyclohexyl]amino]cyclohexyl] 9H-fluorene-9-carboxylate | IC50 | 75.0 [1], 80.0 [2], 150.0 [3], 180.0 [4] |
 | Dimethyl-[10-[5-(piperidine-1-carbothioyl)thiophen-2-yl]-3-thia-17-azapentacyclo[11.7.1.02,11.04,9.017,21]henicosa-1(21),2(11),4,7,9,12-hexaen-6-ylidene]azanium | IC50 | 130.0 [1], 670.0 [2], 2100.0 [3], 12000.0 [4] |
 | Hydrocortisone | IC50 | 50000.0 [1] |
 | Morphine | IC50 | 50000.0 [1] |
 | Dexamethasone | IC50 | 50000.0 [1] |
 | Midazolam | IC50 | 50000.0 [1] |
 | Colchicine | IC50 | 50000.0 [1] |
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