Peptidyl-prolyl cis-trans isomerase FKBP5 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Tacrolimus	Ki	79.0 [1], 80.0 [2]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	6300.0 [1], 8360.0 [2]
	SAFit1	Ki	4.0 [1]
	SAFit2	Ki	6.0 [1]
	Sirolimus	Ki	3.0 [1]
	(S)-3-(Pyridin-3-yl)propyl 1-(3,3-dimethyl-2-oxopentanoyl)pyrrolidine-2-carboxylate	IC50	100000.0 [1]
	Biricodar	IC50	8520.0 [1]
	Timcodar	IC50	100000.0 [1]
	(S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-carboxylic acid 3-pyridin-3-yl-propyl ester	IC50	150000.0 [1]
	2-[3-[(1R)-1-[(2S)-1-[(2S)-2-Cyclohexyl-2-phenylacetyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	Ki	600.0 [1]
	Methyl (2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate	IC50	100000.0 [1]
	(2S)-N-(1-Carbamoylcyclobutyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	4900.0 [1]
	(2S)-N-[1-[(2-Amino-2-oxoethyl)carbamoyl]cyclopentyl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	800.0 [1]
	(2S)-N-[(1R)-2-Amino-2-oxo-1-phenylethyl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	1500.0 [1]
	CID 117967787	Ki	140.0 [1]
	(2S)-N-[(2S,3S)-1-Amino-3-methyl-1-oxopentan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	7100.0 [1]
	(2R)-2-[[(2S)-1-[(2S)-2-Cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carbonyl]amino]pentanediamide	Ki	3400.0 [1]
	2-[3-[(1R)-1-[(2S)-1-[(2R)-2-Cyclohexylpent-4-enoyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	Ki	3400.0 [1]
	(2S)-N-[(2S)-1-Amino-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	3600.0 [1]
	(2S)-N-[(2S)-1-Amino-3-hydroxy-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	62900.0 [1]
	(2S)-N-[(2S)-1-Amino-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	17100.0 [1]
	2-[3-[(1R)-1-[[(2S)-1-[(2S)-2-Cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carbonyl]amino]-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	Ki	43.0 [1]
	(2S)-N-(4-Amino-2-methyl-4-oxobutan-2-yl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	3800.0 [1]
	(2S)-N-[(2R)-1-Amino-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	3800.0 [1]
	(2S)-N-[(2R)-1-Amino-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	10000.0 [1]
	(2S)-N-(1-Carbamoylcyclopropyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	19500.0 [1]
	(2S)-N-[(2S)-1-Amino-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	13400.0 [1]
	(2S)-N-[(2R)-1-Amino-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	4500.0 [1]
	(2S)-N-[(2S)-1-Amino-1-oxo-3-phenylpropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	6500.0 [1]
	(2S)-N-[(2S)-1-Amino-3-methyl-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	12600.0 [1]
	(2S)-N-[(2R)-1-Amino-1-oxo-3-phenylpropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	1400.0 [1]
	(2S)-N-[(2R)-1-Amino-4-hydroxy-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	4200.0 [1]
	(2S)-N-[(2S)-1-Amino-4-hydroxy-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	13000.0 [1]
	(2S)-N-[(2S)-1-Amino-4-methyl-1-oxopentan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	8700.0 [1]
	(2S)-N-[(2S)-1-Amino-4-cyclohexyl-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	12000.0 [1]
	(2S)-N-[(2S)-1-Amino-3-cyclohexyl-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	17800.0 [1]
	2-[3-[(1R)-1-[(2S)-1-[(2R)-2-Cyclohexylpropanoyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	Ki	1200.0 [1]
	(2S)-N-(1-Carbamoylcyclohexyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	1900.0 [1]
	(2S)-1-[(2S)-2-Cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]-N-ethylpiperidine-2-carboxamide	Ki	55000.0 [1]
	(2S)-N-[(2R,3R)-1-Amino-3-methyl-1-oxopentan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	3200.0 [1]
	(2S)-N-[(2S)-1-Amino-1-oxo-4-phenylbutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	9100.0 [1]
	(2S)-N-(2-Amino-2-oxoethyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	36700.0 [1]
	(2S)-N-[(1S)-2-Amino-2-oxo-1-phenylethyl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	3100.0 [1]
	(2S)-N-[(2R)-1-Amino-3-hydroxy-1-oxopropan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	2800.0 [1]
	(2S)-N-[(1S)-2-Amino-1-cyclohexyl-2-oxoethyl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	4300.0 [1]
	(2S)-2-[[(2S)-1-[(2S)-2-Cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carbonyl]amino]pentanediamide	Ki	345000.0 [1]
	(2S)-N-(1-Amino-2-methyl-1-oxopropan-2-yl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	2200.0 [1]
	(2S)-N-[(2R)-1-Amino-3-methyl-1-oxobutan-2-yl]-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	5000.0 [1]
	(2S)-N-(3-Amino-3-oxopropyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	7900.0 [1]
	(2S)-N-(4-Carbamoyloxan-4-yl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	1800.0 [1]
	2-[3-[(1R)-1-[(2S)-1-[(2S)-2-Cyclohexyl-2-(3,5-dimethoxyphenyl)acetyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	Ki	110.0 [1]
	2-[3-[(1R)-1-[(2S)-1-[(2S)-2-Cyclohexyl-2-(3-methoxyphenyl)acetyl]piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	Ki	160.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(2-Cyclohexylacetyl)piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	Ki	4200.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S)-2-cyclohexyl-3-(methoxymethoxy)propanoyl]piperidine-2-carboxylate	Ki	4100.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S)-2-cyclohexyl-3-hydroxypropanoyl]piperidine-2-carboxylate	Ki	2000.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S)-3-acetyloxy-2-cyclohexylpropanoyl]piperidine-2-carboxylate	Ki	2100.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S,3R)-2-cyclohexyl-3-(methoxymethoxy)butanoyl]piperidine-2-carboxylate	Ki	2000.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S)-2-cyclohexyl-3-oxobutanoyl]piperidine-2-carboxylate	Ki	2500.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(E,2S,3R)-2-cyclohexyl-3-hydroxyhex-4-enoyl]piperidine-2-carboxylate	Ki	1100.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2R,3R)-2-cyclohexyl-3-hydroxy-4-methylpentanoyl]piperidine-2-carboxylate	Ki	13000.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S,3R)-2-cyclohexyl-3-(methoxymethoxy)-5-methylhexanoyl]piperidine-2-carboxylate	Ki	17000.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2S,3R)-2-cyclohexyl-3-hydroxy-5-methylhexanoyl]piperidine-2-carboxylate	Ki	9000.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-[(2R,3S)-2-cyclohexyl-3-hydroxy-3-phenylpropanoyl]piperidine-2-carboxylate	Ki	100000.0 [1]
	(2S)-N-(4-Amino-4-oxobutyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	5700.0 [1]
	(2S)-N-(5-Amino-5-oxopentyl)-1-[(2S)-2-cyclohexyl-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxamide	Ki	3900.0 [1]
	(1S,5S,6R)-10-(3,5-Dichlorophenyl)sulfonyl-5-(methoxymethyl)-3-(pyridin-2-ylmethyl)-3,10-diazabicyclo[4.3.1]decan-2-one	Ki	24.5 [1]
	[(1R)-1-(3-Aminophenyl)-3-(3,4-dimethoxyphenyl)propyl] (2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate	IC50	3800.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1S,2R)-2-ethyl-1-hydroxycyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	5800.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1R,2S)-2-ethyl-1-hydroxycyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	3900.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1S,2S)-1-hydroxy-2-(hydroxymethyl)cyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	8500.0 [1]
	2-(3,4-Dimethoxyphenoxy)ethyl (2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate	IC50	100000.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate	IC50	4150.0 [1]
	[(1R)-3-(3,4-Dimethoxyphenyl)-1-[3-(2-morpholin-4-ylethoxy)phenyl]propyl] (2S)-1-(3,3-dimethyl-2-oxopentanoyl)pyrrolidine-2-carboxylate	IC50	15340.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-oxo-2-(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	19300.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1S,2R)-1-hydroxy-2-methylcyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	4270.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1R,2S)-1-hydroxy-2-methylcyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	4540.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1S,2S)-1-hydroxy-2-methylcyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	4180.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[2-[(1R,2R)-1-hydroxy-2-methylcyclohexyl]-2-oxoacetyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	4960.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(4-pyrimidin-2-ylphenyl)sulfonylpiperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	62800.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3-Chlorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	30700.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(1,3-Benzothiazol-6-ylsulfonyl)piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	11600.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(furan-3-ylsulfonyl)piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	100000.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(1-Benzothiophen-2-ylsulfonyl)piperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	67100.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3-Cyanophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	28500.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(3-nitrophenyl)sulfonylpiperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	47200.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3-Aminophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	45400.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(3-fluorophenyl)sulfonylpiperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	54050.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3-Bromophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	15780.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3,5-Dichlorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	22600.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3,4-Dichlorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	100000.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-(3,4-dimethoxyphenyl)sulfonylpiperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	100000.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3-Chloro-4-methoxyphenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	29600.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3,5-Difluorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	88200.0 [1]
	2-[3-[(1R)-1-[(2S)-1-[3,5-Bis(trifluoromethyl)phenyl]sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	100000.0 [1]
	2-[3-[(1R)-1-[(2S)-1-[3-Bromo-5-(trifluoromethyl)phenyl]sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	100000.0 [1]
	2-[3-[(1R)-1-[(2S)-1-[3,5-Bis(methoxycarbonyl)phenyl]sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	100000.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3,5-Dichloro-4-hydroxyphenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	6200.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(3,5-Dichloro-4-methoxyphenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	16400.0 [1]
	2-[3-[(1R)-1-[(2S)-1-(4-Acetamido-3,5-dichlorophenyl)sulfonylpiperidine-2-carbonyl]oxy-3-(3,4-dimethoxyphenyl)propyl]phenoxy]acetic acid	IC50	16100.0 [1]
	2-[3-[(1R)-3-(3,4-Dimethoxyphenyl)-1-[(2S)-1-[(7-nitro-2,3-dihydro-1-benzofuran-5-yl)sulfonyl]piperidine-2-carbonyl]oxypropyl]phenoxy]acetic acid	IC50	27200.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Peptidyl-prolyl cis-trans isomerase FKBP5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/peptidyl-prolyl-cis-trans-isomerase-fkbp5-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 10). Quest Database™ Peptidyl-prolyl cis-trans isomerase FKBP5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/peptidyl-prolyl-cis-trans-isomerase-fkbp5-inhibitors-ic50-ki.
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