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Peroxisome proliferator-activated receptor delta Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
4-Chloro-N-[2-[[5-(trifluoromethyl)-2-pyridinyl]sulfonyl]ethyl]benzamideIC50199.53 [1], 5000.0 [2]
EndurobolKi0.05 [1]
RosiglitazoneIC505.0 [1], 10000.0 [2], 50000.0 [3]
RosiglitazoneKi33300.0 [1]
4-Methyl-2-[4-(trifluoromethyl)phenyl]-N-[2-[5-(trifluoromethyl)pyridin-2-yl]sulfonylethyl]-1,3-thiazole-5-carboxamideIC5010000.0 [1]
N-[2-[5-(Trifluoromethyl)pyridin-2-yl]sulfonylethyl]naphthalene-2-carboxamideIC50320.0 [1], 448.0 [2], 751.0 [3], 930.0 [4], 1931.0 [5]
N-[2-[5-(Trifluoromethyl)pyridin-2-yl]sulfonylethyl]quinoline-3-carboxamideIC50241.0 [1], 1431.0 [2], 2322.0 [3], 6815.0 [4], 17611.0 [5]
Methyl 3-[(4-anilino-2-methoxyphenyl)sulfamoyl]thiophene-2-carboxylateIC50155.0 [1], 158.49 [2], 316.23 [3]
F3MethylAAIC504.0 [1], 10.0 [2]
(R)-3-(4-(3-(2-Benzoyl-4-ethylphenoxy)butoxy)-2-methylphenyl)propanoic acidIC503.0 [1]
{5-Methyl-7-[4-(4-trifluoromethyl-benzyloxy)-benzylsulfanyl]-indan-4-yloxy}-acetic AcidIC50586.0 [1], 586.14 [2], 10000.0 [3]
2-(8-(4-(4-(Trifluoromethyl)benzyloxy)benzylthio)-6-methylchroman-5-yloxy)acetic acidIC50313.0 [1], 10000.0 [2]
LY-518674IC503800.0 [1], 3801.89 [2]
NaveglitazarIC501914.26 [1], 1916.0 [2]
5-[3-[3-(4-Phenoxy-2-propylphenoxy)propoxy]phenyl]-1,3-thiazolidine-2,4-dioneIC5010000.0 [1], 50000.0 [2]
Benzeneacetic acid, 3-chloro-4-((3-((3-phenyl-7-propyl-6-benzofuranyl)oxy)propyl)thio)-IC506.0 [1]
(2S)-2-Methyl-3-[4-[2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acidIC505253.0 [1]
CID 9889841IC504.0 [1]
2-Methyl-3-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenyl}-2-phenoxy-propionic acidIC507113.0 [1]
2-{5-[3-(6-Benzoyl-1-propylnaphthalen-2-yloxy)propoxy]indol-1-YL}ethanoic acidIC50222.84 [1], 223.0 [2]
4-Methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamideIC5025118.86 [1]
(2S)-2-Methyl-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acidIC505519.0 [1]
(2R)-7-(3-(2-Chloro-4-(4-fluorophenoxy)phenoxy)propoxy)-2-ethylchromane-2-carboxylic acidIC5015000.0 [1]
2-Methyl-2-{4-[2-(5-methyl-2-phenyl-oxazol-4-yl)-ethoxy]-phenoxy}-3-phenyl-propionic acidIC504448.0 [1]
(2R)-2-Methyl-3-[4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acidIC502685.0 [1], 2685.34 [2]
{3-Chloro-4-[3-(3-hydroxy-4-propionyl-2-propyl-phenoxy)-propylsulfanyl]-phenyl}-acetic acidIC5020.0 [1]
3-[4-[3-[(1R)-1-[(5-Chloro-1,3-dimethylindole-2-carbonyl)amino]ethyl]-5-fluorophenoxy]-2-ethylphenyl]propanoic acidIC505.0 [1]
2-[4-[3-[2-Chloro-4-(4-fluorophenoxy)phenoxy]propoxy]phenoxy]-2-methylpropanoic acidIC502390.0 [1]
{4-[3-(4-Acetyl-3-hydroxy-2-propyl-phenoxy)-propylsulfanyl]-3-chloro-phenyl}-acetic acidIC5020.0 [1]
{3-Chloro-4-[3-(3-ethyl-7-propyl-benzofuran-6-yloxy)-propylsulfanyl]-phenyl}-acetic acidIC5040.0 [1]
2-{5-[3-(7-Propyl-3-trifluoromethylbenzo[D]isoxazol-6-yloxy)propoxy]indol-1-YL}ethanoic acidIC5095.94 [1], 96.0 [2]
(2S)-2-Methoxy-3-{4-[5-(4-phenoxy-phenoxy)-pent-1-ynyl]-phenyl}-propionic acidIC504120.98 [1], 4123.0 [2]
2-[4-[3-[1-[(3,4-Dimethylphenyl)methyl]-4-methyl-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acidIC50739.61 [1], 740.0 [2]
(2R)-7-(3-(2-Chloro-4-cyclopentylphenoxy)propoxy)-2-methylchromane-2-carboxylic AcidIC5010495.42 [1], 10500.0 [2]
(S)-2-Ethoxy-3-{4-[3-(4-phenoxy-phenoxy)-propoxy]-phenyl}-propionic acidIC501569.0 [1], 1570.36 [2]
(S)-2-Methoxy-3-{4-[4-(4-phenoxy-phenoxy)-but-1-ynyl]-phenyl}-propionic acidIC503935.5 [1], 3938.0 [2]
(R)-7-[3-(2-Chloro-4-isobutyl-phenoxy)-propoxy]-2-methyl-chroman-2-carboxylic acidIC507600.0 [1], 7603.26 [2]
2-[4-[3-[1-[(4-Tert-butylphenyl)methyl]-4-methyl-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acidIC501698.24 [1], 1700.0 [2]
2-(4-(4-(4-(Trifluoromethyl)benzyloxy)benzylthio)-5-methoxy-2-methylphenoxy)acetic acidIC501.7 [1]
2-[4-[3-[1-[(3-Methoxyphenyl)methyl]-5-oxo-4-propyl-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acidIC501999.86 [1], 2000.0 [2]
(R)-7-[3-(2-Chloro-4-trifluoromethyl-phenoxy)-propoxy]-2-ethyl-chroman-2-carboxylic acidIC502300.0 [1], 2301.44 [2]
(S)-3-{4-[3-(Biphenyl-4-yloxy)-propoxy]-phenyl}-2-methoxy-propionic acidIC501389.95 [1], 1391.0 [2]
(S)-3-{4-[3-(4-Benzoyl-phenoxy)-propoxy]-phenyl}-2-methoxy-propionic acidIC502322.74 [1], 2324.0 [2]
(S)-2-Methoxy-3-{3-methoxy-4-[3-(4-phenoxy-phenoxy)-propoxy]-phenyl}-propionic acidIC507502.0 [1]
3-[2-Ethyl-4-[(3R)-3-(4-ethyl-2-pyridin-2-ylphenoxy)butoxy]phenyl]propanoic acidIC503.0 [1]
3-[4-[(3R)-3-(4-Ethyl-2-pyridin-2-ylphenoxy)butoxy]-2-methylphenyl]propanoic acidIC503.0 [1]
(2S)-3-[4-[2-(2-Cyclohexyl-5-methyl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-methyl-2-phenoxypropanoic acidIC509682.78 [1], 9688.0 [2]
3-[4-[(3R)-3-[4-Ethyl-2-(1,3-oxazol-2-yl)phenoxy]butoxy]-2-methylphenyl]propanoic acidIC505.0 [1]
2-[5-[3-(6-Benzoylnaphthalen-2-yl)oxypropoxy]indol-1-yl]acetic acidIC504425.88 [1], 4430.0 [2]
2-[4-[3-[[[2-Fluoro-4-(trifluoromethyl)benzoyl]amino]methyl]-5-methylphenoxy]-2-methylphenoxy]-2-methylpropanoic acidIC505.0 [1]
2-(6-(3-(4-(4-Fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acidIC507616.0 [1], 7620.79 [2]
2-[4-[3-[4-(2-Hydroxyethyl)-1-[(4-methylphenyl)methyl]-5-oxo-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acidIC504100.0 [1], 4102.04 [2]
2-Methyl-2-[2-methyl-4-[3-[[[2-methyl-4-(trifluoromethyl)benzoyl]amino]methyl]phenoxy]phenoxy]propanoic acidIC503.0 [1]
2-[4-[3-[1-(Cyclohexylmethyl)-5-oxo-4-propyl-1,2,4-triazol-3-yl]propyl]phenoxy]-2-methylpropanoic acidIC50879.02 [1], 880.0 [2]
3-[2-Ethyl-4-[(3R)-3-[2-pyridin-2-yl-4-(trifluoromethyl)phenoxy]butoxy]phenyl]propanoic acidIC503.0 [1]
(2R)-2-Methyl-3-[4-[2-(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)ethoxy]phenyl]-2-phenoxypropanoic acidIC506745.28 [1], 6749.0 [2]
3-(1-(3-(7-Propyl-3-(trifluoromethyl)benzo[d]isoxazol-6-yloxy)propyl)-1H-indol-5-yl)propanoic acidIC5069.98 [1], 70.0 [2]
2-(4-(3-(6-Benzoyl-1-propylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acidIC505377.0 [1], 5382.7 [2]
2-(6-(3-(6-Benzoylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acidIC502568.0 [1], 2570.4 [2]
2-(5-(3-(4-(4-Fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acidIC50648.63 [1], 649.0 [2]
2-(6-(3-(4-(4-Fluorobenzoyl)phenoxy)propoxy)-1H-indol-1-yl)acetic acidIC503153.0 [1], 3155.0 [2]
2-(1-(3-(7-Propyl-3-(trifluoromethyl)benzo[d]isoxazol-6-yloxy)propyl)-1H-indol-5-yl)acetic acidIC5057.0 [1]
2-(6-(3-(6-Benzoyl-1-propylnaphthalen-2-yloxy)propoxy)-1H-indol-1-yl)acetic acidIC502398.0 [1], 2398.83 [2]
2-(4-(3-(4-(4-Fluorobenzoyl)-2-propylphenoxy)propoxy)-1H-indol-1-yl)acetic acidIC503256.0 [1], 3258.37 [2]
3-[4-[(3R)-3-[4-Ethyl-2-(1,3-thiazol-4-yl)phenoxy]butoxy]-2-methylphenyl]propanoic acidIC503.0 [1]
4-[({1-[(E)-{[4-(Morpholin-4-yl)phenyl]imino}methyl]naphthalen-2-yl}oxy)methyl]benzoic acidIC5033962.53 [1], 34000.0 [2]
(R)-3-{4-[3-(4-Ethyl-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acidIC504.0 [1]
(R)-3-{2-Methyl-4-[3-(2-phenoxy-4-trifluoromethoxy-phenoxy)-butoxy]-phenyl}-propionic acidIC505.0 [1]
(R)-3-{4-[3-(4-Chloro-2-phenoxy-phenoxy)-butoxy]-2-trifluoromethyl-phenyl}-propionic acidIC505.0 [1]
2-(4-(3-(2-Benzoyl-4-ethylphenoxy)propoxy)phenoxy)-2-methylpropanoic acidIC506.0 [1]
(R)-3-{4-[3-(4-Chloro-2-phenoxy-phenoxy)-butoxy]-2-methyl-phenyl}-propionic acidIC504.0 [1]
(R)-3-{2-Methyl-4-[3-(2-phenoxy-4-trifluoromethyl-phenoxy)-butoxy]-phenyl}-propionic acidIC505.0 [1]
(r)-3-{4-[3-(4-Chloro-2-phenoxy-phenoxy)-butoxy]-2-fluoro-phenyl}-propionic acidIC504.0 [1]
(R)-3-{4-[3-(4-Chloro-2-phenoxy-phenoxy)-butoxy]-2-ethyl-phenyl}-propionic acidIC504.0 [1]
{7-[4-(4-Methoxy-benzyloxy)-benzylsulfanyl]-indan-4-yloxy}-acetic AcidIC50120.0 [1]
2-(4-(4-(4-(Trifluoromethyl)benzyloxy)benzylthio)-5-chloro-2-methylphenoxy)acetic acidIC5020.0 [1]
2-(8-(4-(4-(Trifluoromethyl)benzyloxy)benzylthio)chroman-5-yloxy)acetic acidIC50136.0 [1]
2-(6-((5-(4-Chlorophenyl)isoxazol-3-yl)methoxy)-4-methylbenzo[b]thiophen-3-yl)acetic acidIC5023.0 [1], 23.01 [2]
Benzoic acid, 2-((3-((5-methoxy-4-methyl-1H-indol-1-yl)sulfonyl)benzoyl)amino)-5-methyl-IC5019.95 [1], 20.0 [2]
5-Chloro-2-[[3-(5-methoxy-4-methylindol-1-yl)sulfonylbenzoyl]amino]benzoic acidIC5015.85 [1], 16.0 [2]
2-[[3-(3,4-Dihydro-1H-isoquinolin-2-ylsulfonyl)benzoyl]amino]-5-methylbenzoic acidIC5012.59 [1], 13.0 [2]
5-Chloro-2-[[3-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)benzoyl]amino]benzoic acidIC507.94 [1], 8.0 [2]
5-Bromo-2-[[3-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)benzoyl]amino]benzoic acidIC507.94 [1], 8.0 [2]
2-[[3-(3,4-Dihydro-1H-isoquinolin-2-ylsulfonyl)benzoyl]amino]-5-fluorobenzoic acidIC5025.0 [1], 25.12 [2]
2-[[3-(3,4-Dihydro-1H-isoquinolin-2-ylsulfonyl)benzoyl]amino]-5-(trifluoromethyl)benzoic acidIC505.0 [1], 5.01 [2]
4-Bromo-2-[[3-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)benzoyl]amino]benzoic acidIC505.0 [1], 5.01 [2]
5-Chloro-2-[[3-[(5-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)sulfonyl]benzoyl]amino]benzoic acidIC5012.59 [1], 13.0 [2]
2-[3-[(2-Carboxy-4-chlorophenyl)carbamoyl]phenyl]sulfonyl-3,4-dihydro-1H-isoquinoline-5-carboxylic acidIC503.98 [1], 4.0 [2]
2-[[3-[[5-(Carboxymethoxy)-3,4-dihydro-1H-isoquinolin-2-yl]sulfonyl]benzoyl]amino]-5-chlorobenzoic acidIC5010.0 [1]
5-Chloro-2-[[3-[(6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl)sulfonyl]benzoyl]amino]benzoic acidIC5010.0 [1]
5-Chloro-2-[[3-[(7-fluoro-3,4-dihydro-1H-isoquinolin-2-yl)sulfonyl]benzoyl]amino]benzoic acidIC5015.85 [1], 16.0 [2]
5-Chloro-2-[[3-[(7-chloro-3,4-dihydro-1H-isoquinolin-2-yl)sulfonyl]benzoyl]amino]benzoic acidIC5025.0 [1], 25.12 [2]
5-Chloro-2-[[3-[(7-chloro-8-methyl-3,4-dihydro-1H-isoquinolin-2-yl)sulfonyl]benzoyl]amino]benzoic acidIC5015.85 [1], 16.0 [2]
5-Methyl-2-[[3-(4-methylindol-1-yl)sulfonylbenzoyl]amino]benzoic acidIC506.0 [1], 6.31 [2]
2-[[3-(4-Bromoindol-1-yl)sulfonylbenzoyl]amino]-5-methylbenzoic acidIC5010.0 [1]
2-[[3-(4-Methoxyindol-1-yl)sulfonylbenzoyl]amino]-5-methylbenzoic acidIC5010.0 [1]
5-Methyl-2-[[3-(5-methylindol-1-yl)sulfonylbenzoyl]amino]benzoic acidIC5010.0 [1]
Items per page: 1 - 10 of 97
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References

This online tool may be cited as follows

MLA

"Quest Database™ Peroxisome proliferator-activated receptor delta Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 10 May. 2024, https://www.aatbio.com/data-sets/peroxisome-proliferator-activated-receptor-delta-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 10). Quest Database™ Peroxisome proliferator-activated receptor delta Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/peroxisome-proliferator-activated-receptor-delta-inhibitors-ic50-ki.
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