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Phosphodiesterase 10A Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
PapaverineIC5040.0 [1]
MardepodectIC501.34 [1]
2-[[4-[4-Pyridin-4-yl-1-(2,2,2-trifluoroethyl)pyrazol-3-yl]phenoxy]methyl]quinolineIC500.3 [1], 1.0 [2], 1.41 [3]
2-Methoxy-6,7-dimethyl-9-propylimidazo[1,5-a]pyrido[3,2-e]pyrazineIC507.0 [1], 7.28 [2], 7.3 [3], 32.0 [4]
SildenafilIC503100.0 [1], 5400.0 [2], 6800.0 [3], 10000.0 [4]

References
This online resource may be cited as follows
MLA
"Quest DatabasePhosphodiesterase 10A Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/phosphodiesterase-10a-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabasePhosphodiesterase 10A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/phosphodiesterase-10a-inhibitors-ic50-ki.
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