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Phosphodiesterase 11A Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
TadalafilIC5050.0 [1]
SildenafilIC503000.0 [1]
VardenafilIC50130.0 [1], 240.0 [2]
2-Methoxy-6,7-dimethyl-9-propylimidazo[1,5-a]pyrido[3,2-e]pyrazineIC50690.0 [1], 779.0 [2]
N-(12-Methoxy-5-methyl-3-propyl-2,4,8,13-tetrazatricyclo[7.4.0.02,6]trideca-1(9),3,5,7,10,12-hexaen-7-yl)methanesulfonamideIC5068.6 [1], 69.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabasePhosphodiesterase 11A Inhibitors (IC50, Ki)." AAT Bioquest, Inc.20 Dec2025https://www.aatbio.com/data-sets/phosphodiesterase-11a-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 20). Quest DatabasePhosphodiesterase 11A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/phosphodiesterase-11a-inhibitors-ic50-ki.
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