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Phosphodiesterase 4D Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
RolipramIC50403.0 [1]
RolipramKi382.0 [1]
(R)-2-(4-Fluorophenoxy)-N-(1-(thiophen-2-yl)ethyl)nicotinamideIC501.0 [1]
RoflumilastIC500.27 [1], 0.56 [2], 0.7 [3], 1.1 [4], 460.0 [5]
CilomilastIC5011.0 [1], 27.0 [2], 39.0 [3], 63.0 [4], 79.0 [5]

References
This online resource may be cited as follows
MLA
"Quest DatabasePhosphodiesterase 4D Inhibitors (IC50, Ki)." AAT Bioquest, Inc.15 Dec2025https://www.aatbio.com/data-sets/phosphodiesterase-4d-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 15). Quest DatabasePhosphodiesterase 4D Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/phosphodiesterase-4d-inhibitors-ic50-ki.
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