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Phosphodiesterase 5A Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
SildenafilIC503.6 [1]
SildenafilKi1.6 [1], 1.87 [2], 1.91 [3], 10.0 [4]
TadalafilIC504.0 [1]
TadalafilKi5.2 [1], 10.0 [2]
ZaprinastIC501000.0 [1]

References
This online resource may be cited as follows
MLA
"Quest DatabasePhosphodiesterase 5A Inhibitors (IC50, Ki)." AAT Bioquest, Inc.5 Dec2025https://www.aatbio.com/data-sets/phosphodiesterase-5a-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 5). Quest DatabasePhosphodiesterase 5A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/phosphodiesterase-5a-inhibitors-ic50-ki.
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