Phosphoenolpyruvate carboxykinase cytosolic Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	1-(2-Fluorobenzyl)-3-butyl-8-(N-acetyl-4-aminobenzyl)-xanthine	IC50	2110.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]acetamide	IC50	690.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-1,2-dimethylimidazole-4-sulfonamide	IC50	340.0 [1]
	N-[4-[[3-Butyl-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-1-methylimidazole-4-sulfonamide	IC50	630.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]methanesulfonamide	IC50	1250.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-2,2,2-trifluoroacetamide	IC50	1800.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide	IC50	790.0 [1]
	2-Amino-N-[4-[[3-(cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-4-methyl-1,3-thiazole-5-sulfonamide	IC50	230.0 [1]
	5-Chloro-N-[4-[[3-(cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-1,3-dimethylpyrazole-4-sulfonamide	IC50	290.0 [1]
	N-[4-[[3-Butyl-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-5-chloro-1,3-dimethylpyrazole-4-sulfonamide	IC50	540.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-1-methylpyrazole-4-sulfonamide	IC50	390.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-2-(dimethylamino)acetamide	IC50	2070.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]quinoline-8-sulfonamide	IC50	450.0 [1]
	1-(2-Fluorobenzyl)-8-(4-aminobenzyl)-3-butyl-1H-purine-2,6(3H,7H)-dione	IC50	2560.0 [1]
	3-Cyclopropylmethyl-8-[4-aminobenzyl]-1-(2-fluorobenzyl)-3,7-dihydro-purine-2,6-dione	IC50	1560.0 [1]
	N-[3-Acetamido-4-[[3-butyl-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]acetamide	IC50	8700.0 [1]
	3-Butyl-8-[(2,4-diaminophenyl)methyl]-1-[(2-fluorophenyl)methyl]-7H-purine-2,6-dione	IC50	5650.0 [1]
	3-(Cyclopropylmethyl)-8-[[4-(dimethylsulfamoylamino)phenyl]methyl]-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purine	IC50	960.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-1,3-dimethylpyrazole-4-sulfonamide	IC50	240.0 [1]
	N-[4-[[3-Butyl-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]-2,2,2-trifluoroacetamide	IC50	2300.0 [1]
	N-[4-[[3-(Cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]-2,6-dioxo-7H-purin-8-yl]methyl]phenyl]pyridine-3-sulfonamide	IC50	1950.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 21 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Phosphoenolpyruvate carboxykinase cytosolic Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/phosphoenolpyruvate-carboxykinase-cytosolic-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, May 9). Quest Database™ Phosphoenolpyruvate carboxykinase cytosolic Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/phosphoenolpyruvate-carboxykinase-cytosolic-inhibitors-ic50-ki.
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