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Phospholipase A2 group IIA Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
VarespladibIC5012.0 [1]
(3-{[3-(2-Amino-2-Oxoethyl)-1-Benzyl-2-Ethyl-1h-Indol-5-Yl]oxy}propyl)phosphonic AcidIC50470.0 [1]
ManoalideIC503900.0 [1], 93200.0 [2], 1500000.0 [3]
2-(1-Benzyl-5-methoxy-2-methyl-1h-indol-3-yl)acetamideIC50540.0 [1], 840.0 [2], 880.0 [3], 1000.0 [4]
1,2,4-Oxadiazol-5(2H)-one, 3-[[4-(tetradecyloxy)phenyl]methyl]-IC503400.0 [1], 4000.0 [2]

References
This online resource may be cited as follows
MLA
"Quest DatabasePhospholipase A2 group IIA Inhibitors (IC50, Ki)." AAT Bioquest, Inc.28 Dec2025https://www.aatbio.com/data-sets/phospholipase-a2-group-iia-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 28). Quest DatabasePhospholipase A2 group IIA Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/phospholipase-a2-group-iia-inhibitors-ic50-ki.
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