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Phospholipase D1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-2-naphthamideIC5021.0 [1], 80.0 [2], 81.0 [3]
HalopemideIC5021.0 [1], 220.0 [2]
CID 25105713IC5011.0 [1], 46.0 [2]
N-[2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl]naphthalene-2-carboxamideIC501000.0 [1], 5100.0 [2]
RaloxifeneIC504000.0 [1], 4300.0 [2], 8500.0 [3]
(1R,2R)-N-[2-[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]-2-phenylcyclopropane-1-carboxamideIC5035.0 [1], 660.0 [2]
FIPI hydrochlorideIC501.0 [1], 9.5 [2]
N-[2-[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]-1-benzothiophene-2-carboxamideIC5014.0 [1], 100.0 [2]
4-Chloro-N-(2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC506.3 [1], 55.0 [2]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)furan-2-carboxamideIC5022.0 [1], 360.0 [2]
4-Methoxy-N-(2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC501000.0 [1], 15000.0 [2]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)palmitamideIC503200.0 [1], 20000.0 [2]
3,4-Difluoro-N-(2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC5017.0 [1], 480.0 [2]
3,4-Dichloro-N-(2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC5019.0 [1], 46.0 [2]
3,5-Dichloro-N-(2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC5085.0 [1], 400.0 [2]
4-Methyl-N-(2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC5032.0 [1], 780.0 [2]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-4-vinylbenzamideIC5079.0 [1], 540.0 [2]
3,4,5-Trimethoxy-N-(2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC5051.0 [1], 59.0 [2]
9-Oxo-N-[2-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]fluorene-4-carboxamideIC5020.0 [1], 260.0 [2]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-9H-carbazole-9-carboxamideIC50300.0 [1], 330.0 [2]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-2-(phenylthio)acetamideIC50380.0 [1], 7400.0 [2]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-1H-pyrrole-2-carboxamideIC5037.0 [1], 316.0 [2]
4,5-Dibromo-N-[2-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]furan-2-carboxamideIC508.9 [1], 79.0 [2]
4-Fluoro-N-(4-fluorobenzoyl)-N-[2-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]benzamideIC5048.0 [1], 1400.0 [2]
2-Chloro-N-(2-(4-(5-chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC50870.0 [1], 1200.0 [2]
4-Chloro-N-(4-chlorobenzoyl)-N-(2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl)benzamideIC503400.0 [1], 20000.0 [2]
(S)-N-(1-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propan-2-yl)-2-naphthamideIC5025.0 [1]
4-Fluoro-N-[2-[1-(3-fluorophenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]benzamideIC5011800.0 [1], 12000.0 [2]
N-[2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propyl]naphthalene-2-carboxamideIC5064.0 [1], 315.0 [2]
4-Fluoro-N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propyl]benzamideIC50290.0 [1], 1490.0 [2]
4-Bromo-N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propyl]benzamideIC50120.0 [1], 230.0 [2]
5-Fluoro-N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propyl]-1H-indole-2-carboxamideIC5018.0 [1], 35.0 [2]
N-[2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propyl]-1H-indole-2-carboxamideIC506.0 [1], 21.0 [2]
3,4-Difluoro-N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propyl]benzamideIC5017.0 [1], 1080.0 [2]
4-Fluoro-N-[2-[2-methyl-4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]benzamideIC50636.0 [1], 7315.0 [2]
(1R,2R)-N-[2-[2-Methyl-4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]-2-phenylcyclopropane-1-carboxamideIC50115.0 [1], 2770.0 [2]
3,4-Difluoro-N-[2-[3-fluoro-4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]benzamideIC5021.0 [1], 100.0 [2]
N-[2-[5-(2-Oxo-3H-benzimidazol-1-yl)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]ethyl]naphthalene-2-carboxamideIC50244.0 [1], 1790.0 [2]
4-Fluoro-N-[2-[5-(2-oxo-3H-benzimidazol-1-yl)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]ethyl]benzamideIC50870.0 [1], 3565.0 [2]
4-Bromo-N-[2-[5-(2-oxo-3H-benzimidazol-1-yl)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]ethyl]benzamideIC50468.0 [1], 2590.0 [2]
5-Fluoro-N-[2-[5-(2-oxo-3H-benzimidazol-1-yl)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]ethyl]-1H-indole-2-carboxamideIC50230.0 [1], 1235.0 [2]
N-[2-[5-(2-Oxo-3H-benzimidazol-1-yl)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]ethyl]-1H-indole-2-carboxamideIC5072.0 [1], 220.0 [2]
3,4-Difluoro-N-[2-[5-(2-oxo-3H-benzimidazol-1-yl)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]ethyl]benzamideIC50820.0 [1], 3250.0 [2]
(1R,2R)-N-[2-[5-(2-Oxo-3H-benzimidazol-1-yl)-3,3a,4,5,6,6a-hexahydro-1H-cyclopenta[c]pyrrol-2-yl]ethyl]-2-phenylcyclopropane-1-carboxamideIC50115.0 [1], 1080.0 [2]
N-[2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl]quinoline-2-carboxamideIC501900.0 [1], 20000.0 [2]
4-Bromo-N-[(2S)-1-[1-(3-methylphenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]propan-2-yl]benzamideIC506.0 [1], 48.0 [2]
N-[2-[1-(3-Fluorophenyl)-2-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]naphthalene-2-carboxamideIC501500.0 [1], 7400.0 [2]
(1R,2S)-N-[(2S)-1-[4-(5-Bromo-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-2-phenylcyclopropane-1-carboxamideIC503.7 [1], 15.0 [2]
(Z)-4-(1-(4-(2-(Dimethylamino)ethoxy)-phenyl)-2-phenylbut-1-en-1-yl)phenolIC504800.0 [1]
1-(2-Pyridyl)piperazineIC503600.0 [1]
Presqualene diphosphateIC501000.0 [1]
N-[2-[1-(3-Fluorophenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]naphthalene-2-carboxamideIC501500.0 [1]
1-(4-Pyridyl)piperazineIC503600.0 [1]
(1R,2R)-N-[(2S)-1-[4-(5-Bromo-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-2-phenylcyclopropane-1-carboxamideIC503.7 [1]
3,4-Difluoro-N-[2-[1-(3-fluorophenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]benzamideIC5020000.0 [1]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)octanamideIC506000.0 [1]
N-(2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl)-4-(trifluoromethyl)benzamideIC5020000.0 [1]
N-(2-(4-(2-Oxo-2,3-dihydrobenzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)quinoline-3-carboxamideIC508.0 [1]
4-Fluoro-N-[2-[1-(4-fluorophenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]benzamideIC5014000.0 [1]
N-(2-(4-(5-Bromo-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-4-fluorobenzamideIC504.0 [1]
N-[2-[1-(4-Chlorophenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]-4-fluorobenzamideIC505590.0 [1]
N-[2-[1-(4-Bromophenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]-4-fluorobenzamideIC5010000.0 [1]
N-(2-(4-(5-Chloro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-4-methylbenzamideIC5010.0 [1]
4-Chloro-N-[(2S)-1-[4-(5-chloro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]benzamideIC506.4 [1]
(1R,2R)-N-[(2S)-1-[4-(5-Chloro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-2-phenylcyclopropane-1-carboxamideIC508.0 [1]
N-[(2S)-1-[4-(5-Chloro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-3,4-difluorobenzamideIC503.0 [1]
N-[(2S)-1-[4-(5-Bromo-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-3,4-difluorobenzamideIC503.5 [1]
N-[(2S)-1-[4-(5-Bromo-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-4-chlorobenzamideIC504.0 [1]
N-[(2S)-1-[4-(6-Fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]naphthalene-2-carboxamideIC502.0 [1]
N-[(2S)-1-[4-(5-Bromo-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]naphthalene-2-carboxamideIC505.5 [1]
(1R,2R)-N-[(2S)-1-[4-(6-Fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-2-phenylcyclopropane-1-carboxamideIC5012.0 [1]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-3-phenylpropiolamideIC5040.0 [1]
N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)quinoline-6-carboxamideIC5070.0 [1]
N-[2-[4-(2-Oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]-1,4-dihydronaphthalene-2-carboxamideIC50110.0 [1]
6-Fluoro-N-(2-(4-(2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-2-naphthamideIC50120.0 [1]
N-(2-(4-(5-Fluoro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-2-naphthamideIC504.0 [1]
4-Chloro-N-(2-(4-(5-fluoro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC5018.0 [1]
4-Fluoro-N-(2-(4-(5-fluoro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC5012.0 [1]
N-(2-(4-(5-Bromo-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)-4-chlorobenzamideIC503.0 [1]
4-Chloro-N-(2-(4-(6-fluoro-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-1-yl)piperidin-1-yl)ethyl)benzamideIC507.0 [1]
3,4-Difluoro-N-[2-[4-(6-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]ethyl]benzamideIC504.0 [1]
4-Chloro-N-[(2S)-1-[4-(4-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]benzamideIC5043.0 [1]
4-Fluoro-N-[(2S)-1-[4-(4-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]benzamideIC50130.0 [1]
3,4-Difluoro-N-[(2S)-1-[4-(4-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]benzamideIC5038.0 [1]
N-[(2S)-1-[4-(4-Fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]naphthalene-2-carboxamideIC5066.0 [1]
(1R,2R)-N-[(2S)-1-[4-(4-Fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-2-phenylcyclopropane-1-carboxamideIC50100.0 [1]
4-Fluoro-N-[(2S)-1-[4-(5-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]benzamideIC5011.0 [1]
4-Chloro-N-[(2S)-1-[4-(5-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]benzamideIC507.4 [1]
N-[(2S)-1-[4-(5-Chloro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propan-2-yl]-4-fluorobenzamideIC5010.0 [1]
(1S,2S)-N-[2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl]-2-phenylcyclopropane-1-carboxamideIC5020000.0 [1]
N-[2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl]-3-phenylprop-2-ynamideIC502100.0 [1]
(1S,2S)-N-[(2S)-1-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propan-2-yl]-2-phenylcyclopropane-1-carboxamideIC502600.0 [1]
(S)-3,4-Difluoro-N-(1-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propan-2-yl)benzamideIC50150.0 [1]
N-[2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl]-1-benzothiophene-2-carboxamideIC50150.0 [1]
N-[2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl]-1,2,3,4-tetrahydronaphthalene-2-carboxamideIC504250.0 [1]
4-Amino-3-methoxy-N-[2-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl]benzamideIC505900.0 [1]
N-(2-(4-Oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)ethyl)quinoxaline-2-carboxamideIC5020000.0 [1]
(S)-3-Methyl-N-(1-(4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decan-8-yl)propan-2-yl)benzamideIC503400.0 [1]
5-Fluoro-N-[2-[1-(3-fluorophenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]-1H-indole-2-carboxamideIC50210.0 [1]
N-[2-[1-(3-Chlorophenyl)-4-oxo-1,3,8-triazaspiro[4.5]decan-8-yl]ethyl]-5-fluoro-1H-indole-2-carboxamideIC50250.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Phospholipase D1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 9 May. 2024, https://www.aatbio.com/data-sets/phospholipase-d1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, May 9). Quest Database™ Phospholipase D1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/phospholipase-d1-inhibitors-ic50-ki.
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