Structure | Compound Name | Standard Type | Standard Values (in nM) |
|---|---|---|---|
| Dactolisib | IC50 | 4.0 [1], 16.4 [2], 35.15 [3], 49.0 [4], 89.0 [5] | |
| CID 46927938 | IC50 | 2.3 [1] | |
| CID 46927938 | Ki | 2.3 [1], 2.34 [2] | |
| [3-[4-(2-Aminopyrimidin-5-yl)-2-morpholin-4-yl-5,6-dihydropyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl] N-methylsulfamate | Ki | 0.08 [1], 0.23 [2] | |
| 4-[4-(2-Aminopyrimidin-5-yl)-7-[3-[methyl(methylsulfamoyl)amino]cyclobutyl]-5,6-dihydropyrrolo[2,3-d]pyrimidin-2-yl]morpholine | Ki | 0.19 [1], 0.32 [2], 0.41 [3], 0.47 [4] | |
MLA | "Quest Database™ PI3-kinase p110-alpha/p85-alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 4 Dec. 2025, https://www.aatbio.com/data-sets/pi3-kinase-p110-alpha-p85-alpha-inhibitors-ic50-ki. | |
APA | AAT Bioquest, Inc. (2025, December 4). Quest Database™ PI3-kinase p110-alpha/p85-alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/pi3-kinase-p110-alpha-p85-alpha-inhibitors-ic50-ki. | |
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