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PI3-kinase p110-alpha/p85-alpha Inhibitors (IC50, Ki)
Structure
Compound Name
Standard Type
Standard Values (in nM)
DactolisibIC504.0 [1], 16.4 [2], 35.15 [3], 49.0 [4], 89.0 [5]
CID 46927938IC502.3 [1]
CID 46927938Ki2.3 [1], 2.34 [2]
[3-[4-(2-Aminopyrimidin-5-yl)-2-morpholin-4-yl-5,6-dihydropyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl] N-methylsulfamateKi0.08 [1], 0.23 [2]
4-[4-(2-Aminopyrimidin-5-yl)-7-[3-[methyl(methylsulfamoyl)amino]cyclobutyl]-5,6-dihydropyrrolo[2,3-d]pyrimidin-2-yl]morpholineKi0.19 [1], 0.32 [2], 0.41 [3], 0.47 [4]

References
This online resource may be cited as follows
MLA
"Quest DatabasePI3-kinase p110-alpha/p85-alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc.4 Dec2025https://www.aatbio.com/data-sets/pi3-kinase-p110-alpha-p85-alpha-inhibitors-ic50-ki.
APA
AAT Bioquest, Inc. (2025December 4). Quest DatabasePI3-kinase p110-alpha/p85-alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/pi3-kinase-p110-alpha-p85-alpha-inhibitors-ic50-ki.
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